Compile Data Set for Download or QSAR
Report error Found 62 Enz. Inhib. hit(s) with all data for entry = 1074
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8686BDBM8686(4-[(1E)-{2-[1-(3-methoxyphenyl)-1H-pyrazolo[3,4-d]...)
Affinity DataIC50: 2.51nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8688BDBM8688((1E)-1-[(4-methanesulfonylphenyl)methylidene]-2-[1...)
Affinity DataIC50: 2.51nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8674BDBM8674(4-{4-[(2E)-2-(pyridin-4-ylmethylidene)hydrazin-1-y...)
Affinity DataIC50: 3.16nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8695BDBM8695(ethyl({4-[(1E)-{2-[1-(3-methoxyphenyl)-1H-pyrazolo...)
Affinity DataIC50: 3.98nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8687BDBM8687((1E)-1-[(3-methanesulfonylphenyl)methylidene]-2-[1...)
Affinity DataIC50: 3.98nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8694BDBM8694(({4-[(1E)-{2-[1-(3-methoxyphenyl)-1H-pyrazolo[3,4-...)
Affinity DataIC50: 5.01nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8698BDBM8698(3-(dimethylamino)-N-{4-[(1E)-{2-[1-(3-methoxypheny...)
Affinity DataIC50: 5.01nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8692BDBM8692((2-{4-[(1E)-{2-[1-(3-methoxyphenyl)-1H-pyrazolo[3,...)
Affinity DataIC50: 6.31nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8682BDBM8682((1E)-1-[(3-fluorophenyl)methylidene]-2-[1-(3-metho...)
Affinity DataIC50: 7.94nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8683BDBM8683((1E)-1-[(4-fluorophenyl)methylidene]-2-[1-(3-metho...)
Affinity DataIC50: 7.94nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8704BDBM8704(N-(2-methanesulfonylethyl)-4-[(1E)-{2-[1-(3-methox...)
Affinity DataIC50: 7.94nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8708BDBM8708(4-[(1E)-{2-[1-(3-methoxyphenyl)-3-propyl-1H-pyrazo...)
Affinity DataIC50: 10nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8677BDBM8677((2E)-1-[1-(3-methoxyphenyl)-1H-pyrazolo[3,4-d]pyri...)
Affinity DataIC50: 10nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8685BDBM8685(3-[(1E)-{2-[1-(3-methoxyphenyl)-1H-pyrazolo[3,4-d]...)
Affinity DataIC50: 10nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8705BDBM8705(N-[2-(dimethylamino)ethyl]-4-[(1E)-{2-[1-(3-methox...)
Affinity DataIC50: 10nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8706BDBM8706(4-[(1E)-{2-[1-(3-methoxyphenyl)-3-methyl-1H-pyrazo...)
Affinity DataIC50: 10nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8707BDBM8707(4-[(1E)-{2-[3-ethyl-1-(3-methoxyphenyl)-1H-pyrazol...)
Affinity DataIC50: 12.6nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8696BDBM8696(N-{4-[(1E)-{2-[1-(3-methoxyphenyl)-1H-pyrazolo[3,4...)
Affinity DataIC50: 12.6nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8689BDBM8689(4-[(1E)-{2-[1-(3-methoxyphenyl)-1H-pyrazolo[3,4-d]...)
Affinity DataIC50: 12.6nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8697BDBM8697(N-{4-[(1E)-{2-[1-(3-methoxyphenyl)-1H-pyrazolo[3,4...)
Affinity DataIC50: 15.8nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8684BDBM8684((1E)-1-[(3,4-difluorophenyl)methylidene]-2-[1-(3-m...)
Affinity DataIC50: 15.8nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8701BDBM8701(4-[(1E)-{2-[1-(3-methoxyphenyl)-1H-pyrazolo[3,4-d]...)
Affinity DataIC50: 15.8nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8703BDBM8703(N-[2-(dimethylamino)ethyl]-4-[(1E)-{2-[1-(3-methox...)
Affinity DataIC50: 15.8nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8679BDBM8679((2E)-1-[1-(3-methoxyphenyl)-1H-pyrazolo[3,4-d]pyri...)
Affinity DataIC50: 25.1nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8709BDBM8709(4-[(1E)-{2-[1-(3-methoxyphenyl)-3-(propan-2-yl)-1H...)
Affinity DataIC50: 31.6nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8680BDBM8680((2E)-1-[1-(3-methoxyphenyl)-1H-pyrazolo[3,4-d]pyri...)
Affinity DataIC50: 31.6nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8702BDBM8702(4-[(1E)-{2-[1-(3-methoxyphenyl)-1H-pyrazolo[3,4-d]...)
Affinity DataIC50: 31.6nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8673BDBM8673(3-{4-[(2E)-2-(pyridin-4-ylmethylidene)hydrazin-1-y...)
Affinity DataIC50: 31.6nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8675BDBM8675(2-methoxy-6-{4-[(2E)-2-(pyridin-4-ylmethylidene)hy...)
Affinity DataIC50: 39.8nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8676BDBM8676(2-{4-[(2E)-2-(pyridin-4-ylmethylidene)hydrazin-1-y...)
Affinity DataIC50: 39.8nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8710BDBM8710(4-[(1E)-1-{2-[1-(3-methoxyphenyl)-1H-pyrazolo[3,4-...)
Affinity DataIC50: 63.1nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8663BDBM8663(4-[(1E)-{2-[1-(3-ethoxyphenyl)-1H-pyrazolo[3,4-d]p...)
Affinity DataIC50: 100nMpH: 7.2 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8649BDBM8649(2-methoxy-4-[(1E)-(2-{1-phenyl-1H-pyrazolo[3,4-d]p...)
Affinity DataIC50: 100nMpH: 7.2 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8656BDBM8656(4-[(1E)-(2-{1-phenyl-1H-pyrazolo[3,4-d]pyrimidin-4...)
Affinity DataIC50: 100nMpH: 7.2 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8681BDBM8681((1E)-1-[(2-fluorophenyl)methylidene]-2-[1-(3-metho...)
Affinity DataIC50: 126nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8667BDBM8667(N-(3-{4-[(2E)-2-(pyridin-4-ylmethylidene)hydrazin-...)
Affinity DataIC50: 159nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8657BDBM8657(4-[(1E)-{2-[1-(2-methylphenyl)-1H-pyrazolo[3,4-d]p...)
Affinity DataIC50: 159nMpH: 7.2 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8658BDBM8658(4-[(1E)-{2-[1-(3-methylphenyl)-1H-pyrazolo[3,4-d]p...)
Affinity DataIC50: 159nMpH: 7.2 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8690BDBM8690((2E)-1-[1-(3-methoxyphenyl)-1H-pyrazolo[3,4-d]pyri...)
Affinity DataIC50: 159nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8670BDBM8670(4-[(1E)-{2-[1-(3-bromophenyl)-1H-pyrazolo[3,4-d]py...)
Affinity DataIC50: 251nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8669BDBM8669(4-[(1E)-{2-[1-(3-fluorophenyl)-1H-pyrazolo[3,4-d]p...)
Affinity DataIC50: 316nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8664BDBM8664(4-[(1E)-(2-{1-[3-(trifluoromethoxy)phenyl]-1H-pyra...)
Affinity DataIC50: 316nMpH: 7.2 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8668BDBM8668(N-(3-{4-[(2E)-2-(pyridin-4-ylmethylidene)hydrazin-...)
Affinity DataIC50: 631nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8662BDBM8662(4-[(1E)-{2-[1-(4-methoxyphenyl)-1H-pyrazolo[3,4-d]...)
Affinity DataIC50: 1.00E+3nMpH: 7.2 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8672BDBM8672(2-{4-[(2E)-2-(pyridin-4-ylmethylidene)hydrazin-1-y...)
Affinity DataIC50: 1.26E+3nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8666BDBM8666(N-(cyclopropylmethyl)-3-{4-[(2E)-2-(pyridin-4-ylme...)
Affinity DataIC50: 2.00E+3nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8660BDBM8660(4-[(1E)-{2-[1-(2-methoxyphenyl)-1H-pyrazolo[3,4-d]...)
Affinity DataIC50: 2.51E+3nMpH: 7.2 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8654BDBM8654(2-methoxy-4-[(1E)-{2-[1-(propan-2-yl)-1H-pyrazolo[...)
Affinity DataIC50: 2.51E+3nMpH: 7.2 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8691BDBM8691((1E)-1-({4-[(4-fluorophenyl)methoxy]phenyl}methyli...)
Affinity DataIC50: 2.51E+3nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Glaxosmithkline

LigandChemical structure of BindingDB Monomer ID 8693BDBM8693(N,N-diethyl-4-[(1E)-{2-[1-(3-methoxyphenyl)-1H-pyr...)
Affinity DataIC50: 2.51E+3nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 2.5 uM ATP/ [gamma-33P] ATP. Af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2006
Entry Details Article
PubMed
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