Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50014632
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50145451([(S)-1-((S)-2-Oxo-piperidin-3-ylaminooxalyl)-penty...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory concentration against recombinant human cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50138842([(S)-1-(4-Bromo-1H-pyrazol-3-ylaminooxalyl)-pentyl...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibitory concentration against recombinant human cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50145460([(S)-1-(Thiazol-4-ylmethyl)-aminooxalyl]-pentyl)-c...)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibitory concentration against recombinant human cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50145457([(S)-1-(Isoxazol-5-ylmethyl)-aminooxalyl]-pentyl)-...)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibitory concentration against recombinant human cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50145453([(S)-1-(Thiazol-5-ylmethyl)-aminooxalyl]-pentyl)-c...)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibitory concentration against recombinant human cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50145456([(S)-1-(Thiazol-2-ylmethyl)-aminooxalyl]-pentyl)-c...)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibitory concentration against recombinant human cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50145459([(S)-1-([1,3,4]Oxadiazol-2-ylmethyl)-aminooxalyl]-...)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibitory concentration against recombinant human cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50145452([(S)-1-(Pyridin-3-ylmethyl)-aminooxalyl]-pentyl)-c...)
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibitory concentration against recombinant human cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50145454([(S)-1-(Pyridin-4-ylmethyl)-aminooxalyl]-pentyl)-c...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory concentration against recombinant human cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50145458([(S)-1-(Pyridin-2-ylmethyl)-aminooxalyl]-pentyl)-c...)
Affinity DataIC50: 4.40E+4nMAssay Description:Inhibitory concentration against recombinant human cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50145455([(S)-1-((R)-1-[1,3,4]Oxadiazol-2-yl-ethylaminooxal...)
Affinity DataIC50: 5.90E+4nMAssay Description:Inhibitory concentration against recombinant human cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed