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Found 94 Enz. Inhib. hit(s) with all data for entry = 50014833
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148090((R)-7-{3-[2-Chloro-4-(4-fluoro-phenoxy)-phenoxy]-p...)
Affinity DataIC50:  60nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor alpha using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148110((R)-7-[3-(2-Chloro-4-phenoxy-phenoxy)-propoxy]-2-m...)
Affinity DataIC50:  60nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor alpha using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148097(7-[3-(2-Chloro-4-phenoxy-phenoxy)-propoxy]-2-ethyl...)
Affinity DataIC50:  120nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor alpha using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148092(7-[3-(2-Chloro-4-phenoxy-phenoxy)-propoxy]-2-methy...)
Affinity DataIC50:  120nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor alpha using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM28681(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)
Affinity DataIC50:  200nMAssay Description:In vitro binding affinity for human PPAR gamma receptor using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148110((R)-7-[3-(2-Chloro-4-phenoxy-phenoxy)-propoxy]-2-m...)
Affinity DataIC50:  250nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor gamma using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148090((R)-7-{3-[2-Chloro-4-(4-fluoro-phenoxy)-phenoxy]-p...)
Affinity DataIC50:  260nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor gamma using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148094(2-Ethyl-7-[3-(4-phenoxy-2-propyl-phenoxy)-propoxy]...)
Affinity DataIC50:  360nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor alpha using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148107(2-Ethyl-7-{3-[4-(4-methanesulfonyl-phenoxy)-2-prop...)
Affinity DataIC50:  370nMAssay Description:In vitro binding affinity for human PPAR gamma receptor using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148109(7-[3-(4-Phenoxy-2-propyl-phenoxy)-propoxy]-2-propy...)
Affinity DataIC50:  370nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor gamma using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148096(2-Ethyl-7-[3-(2-fluoro-4-phenoxy-phenoxy)-propoxy]...)
Affinity DataIC50:  370nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor alpha using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148094(2-Ethyl-7-[3-(4-phenoxy-2-propyl-phenoxy)-propoxy]...)
Affinity DataIC50:  440nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor gamma using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148105(2-Ethyl-7-{3-[4-(4-methoxy-phenoxy)-2-propyl-pheno...)
Affinity DataIC50:  630nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor gamma using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148097(7-[3-(2-Chloro-4-phenoxy-phenoxy)-propoxy]-2-ethyl...)
Affinity DataIC50:  690nMAssay Description:In vitro binding affinity for human PPAR gamma receptor using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148089(2-Methyl-7-[3-(4-phenoxy-2-propyl-phenoxy)-propoxy...)
Affinity DataIC50:  750nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor gamma using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148106(2-Ethyl-7-{3-[4-(4-fluoro-phenoxy)-2-propyl-phenox...)
Affinity DataIC50:  970nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor alpha using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148108(7-[3-(4-Phenoxy-2-propyl-phenoxy)-propoxy]-chroman...)
Affinity DataIC50:  980nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor gamma using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148100(2-tert-Butyl-7-[3-(4-phenoxy-2-propyl-phenoxy)-pro...)
Affinity DataIC50:  1.20E+3nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor gamma using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148106(2-Ethyl-7-{3-[4-(4-fluoro-phenoxy)-2-propyl-phenox...)
Affinity DataIC50:  1.20E+3nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor gamma using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148092(7-[3-(2-Chloro-4-phenoxy-phenoxy)-propoxy]-2-methy...)
Affinity DataIC50:  1.40E+3nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor gamma using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148098((S)-7-[3-(2-Chloro-4-phenoxy-phenoxy)-propoxy]-2-m...)
Affinity DataIC50:  1.40E+3nMAssay Description:In vitro binding affinity for human PPAR gamma receptor using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148102(7-{3-[4-(4-Chloro-phenoxy)-2-propyl-phenoxy]-propo...)
Affinity DataIC50:  1.40E+3nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor gamma using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148108(7-[3-(4-Phenoxy-2-propyl-phenoxy)-propoxy]-chroman...)
Affinity DataIC50:  1.50E+3nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor alpha using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148101(2-Methyl-6-[3-(4-phenoxy-2-propyl-phenoxy)-propoxy...)
Affinity DataIC50:  1.70E+3nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor gamma using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148104(2-Ethyl-7-[3-(4-phenoxy-phenoxy)-propoxy]-chroman-...)
Affinity DataIC50:  1.70E+3nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor alpha using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148099(7-[4-(4-Phenoxy-2-propyl-phenoxy)-butoxy]-chroman-...)
Affinity DataIC50:  1.80E+3nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor gamma using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148089(2-Methyl-7-[3-(4-phenoxy-2-propyl-phenoxy)-propoxy...)
Affinity DataIC50:  1.90E+3nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor alpha using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148095(2-Methyl-6-[4-(4-phenoxy-2-propyl-phenoxy)-butoxy]...)
Affinity DataIC50:  2.00E+3nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor alpha using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148109(7-[3-(4-Phenoxy-2-propyl-phenoxy)-propoxy]-2-propy...)
Affinity DataIC50:  2.10E+3nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor alpha using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148095(2-Methyl-6-[4-(4-phenoxy-2-propyl-phenoxy)-butoxy]...)
Affinity DataIC50:  2.30E+3nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor gamma using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148103(6-[3-(4-Phenoxy-2-propyl-phenoxy)-propoxy]-chroman...)
Affinity DataIC50:  2.90E+3nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor gamma using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148100(2-tert-Butyl-7-[3-(4-phenoxy-2-propyl-phenoxy)-pro...)
Affinity DataIC50:  3.00E+3nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor alpha using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148091(6-[4-(4-Phenoxy-2-propyl-phenoxy)-butoxy]-chroman-...)
Affinity DataIC50:  3.00E+3nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor gamma using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148101(2-Methyl-6-[3-(4-phenoxy-2-propyl-phenoxy)-propoxy...)
Affinity DataIC50:  3.30E+3nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor alpha using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148102(7-{3-[4-(4-Chloro-phenoxy)-2-propyl-phenoxy]-propo...)
Affinity DataIC50:  4.00E+3nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor alpha using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148111((S)-7-{3-[2-Chloro-4-(4-fluoro-phenoxy)-phenoxy]-p...)
Affinity DataIC50:  4.40E+3nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor gamma using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148096(2-Ethyl-7-[3-(2-fluoro-4-phenoxy-phenoxy)-propoxy]...)
Affinity DataIC50:  4.70E+3nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor gamma using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148093(2-Methyl-7-[4-(4-phenoxy-2-propyl-phenoxy)-butoxy]...)
Affinity DataIC50:  5.10E+3nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor gamma using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148091(6-[4-(4-Phenoxy-2-propyl-phenoxy)-butoxy]-chroman-...)
Affinity DataIC50:  5.80E+3nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor alpha using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148093(2-Methyl-7-[4-(4-phenoxy-2-propyl-phenoxy)-butoxy]...)
Affinity DataIC50: >1.50E+4nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor alpha using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148111((S)-7-{3-[2-Chloro-4-(4-fluoro-phenoxy)-phenoxy]-p...)
Affinity DataIC50: >1.50E+4nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor alpha using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148105(2-Ethyl-7-{3-[4-(4-methoxy-phenoxy)-2-propyl-pheno...)
Affinity DataIC50: >1.50E+4nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor alpha using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148098((S)-7-[3-(2-Chloro-4-phenoxy-phenoxy)-propoxy]-2-m...)
Affinity DataIC50: >1.50E+4nMAssay Description:In vitro binding affinity for human Peroxisome proliferator activated receptor gamma using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148107(2-Ethyl-7-{3-[4-(4-methanesulfonyl-phenoxy)-2-prop...)
Affinity DataIC50: >1.50E+4nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor alpha using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148098((S)-7-[3-(2-Chloro-4-phenoxy-phenoxy)-propoxy]-2-m...)
Affinity DataIC50: >1.50E+4nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor alpha using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148099(7-[4-(4-Phenoxy-2-propyl-phenoxy)-butoxy]-chroman-...)
Affinity DataIC50: >1.50E+4nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor alpha using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148104(2-Ethyl-7-[3-(4-phenoxy-phenoxy)-propoxy]-chroman-...)
Affinity DataIC50: >1.50E+4nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor gamma using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148103(6-[3-(4-Phenoxy-2-propyl-phenoxy)-propoxy]-chroman...)
Affinity DataIC50: >1.50E+4nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor alpha using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM28681(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)
Affinity DataIC50:  1.50E+4nMAssay Description:In vitro binding affinity for human peroxisome proliferator activated receptor alpha using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50148110((R)-7-[3-(2-Chloro-4-phenoxy-phenoxy)-propoxy]-2-m...)
Affinity DataEC50:  80nMAssay Description:In vitro transcriptional activation by human PPAR gamma Gal4 chimeraMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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