Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 50014979
LigandChemical structure of BindingDB Monomer ID 50149871BDBM50149871((R)-2-((3-(biphenyl-4-yloxy)-3-(4-fluorophenyl)pro...)
Affinity DataIC50: 26nMAssay Description:Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50149875BDBM50149875({(R)-4-[5-Chloro-2-(4-methoxy-phenylsulfanyl)-phen...)
Affinity DataIC50: 150nMAssay Description:Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50149873BDBM50149873({(2R,5S)-4-[2-(4-Methoxy-phenylsulfanyl)-phenyl]-2...)
Affinity DataIC50: 160nMAssay Description:Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50149865BDBM50149865({4-[5-Chloro-2-(4-methoxy-phenylsulfanyl)-phenyl]-...)
Affinity DataIC50: 290nMAssay Description:Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50149856BDBM50149856({Methyl-[(R)-3-phenyl-3-(4-trifluoromethyl-phenoxy...)
Affinity DataIC50: 320nMAssay Description:Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50149866BDBM50149866({4-[2-(4-Chloro-phenylsulfanyl)-phenyl]-2,5-dimeth...)
Affinity DataIC50: 360nMAssay Description:Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50149862BDBM50149862([2,5-Dimethyl-4-(2-p-tolylsulfanyl-phenyl)-piperaz...)
Affinity DataIC50: 550nMAssay Description:Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50149859BDBM50149859({4-[2-(4-Methoxy-phenylsulfanyl)-phenyl]-2,5-dimet...)
Affinity DataIC50: 580nMAssay Description:Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50149872BDBM50149872({4-[2-(Biphenyl-4-ylsulfanyl)-phenyl]-2,5-dimethyl...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50149868BDBM50149868({(S)-4-[5-Chloro-2-(4-methoxy-phenylsulfanyl)-phen...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50149853BDBM50149853({4-[2-(4-Methoxy-phenylsulfanyl)-phenyl]-2,2-dimet...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50149860BDBM50149860({4-[2-(4-Methoxy-phenylsulfanyl)-5-methyl-phenyl]-...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50149877BDBM50149877({4-[2-(4-Methoxy-phenylsulfanyl)-phenyl]-2-methyl-...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50149876BDBM50149876({4-[5-Chloro-2-(4-methoxy-phenylsulfanyl)-phenyl]-...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50149861BDBM50149861({4-[2-(4-Fluoro-phenylsulfanyl)-phenyl]-2,5-dimeth...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50149874BDBM50149874([2,5-Dimethyl-4-(2-phenylsulfanyl-phenyl)-piperazi...)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50149864BDBM50149864({4-[2-(4-Hydroxy-phenylsulfanyl)-phenyl]-2,5-dimet...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50149863BDBM50149863({4-[5-Methoxy-2-(4-methoxy-phenylsulfanyl)-phenyl]...)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50149858BDBM50149858({4-[2-(4-Methoxy-phenylsulfanyl)-phenyl]-piperazin...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50149854BDBM50149854({4-[2-(4-Methoxy-phenylsulfanyl)-phenyl]-3-methyl-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50149870BDBM50149870({(2R,5R)-4-[2-(4-Methoxy-phenylsulfanyl)-phenyl]-2...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50149869BDBM50149869({(2S,5S)-4-[2-(4-Methoxy-phenylsulfanyl)-phenyl]-2...)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50149857BDBM50149857({4-[2-(4-Acetylamino-phenylsulfanyl)-phenyl]-2,5-d...)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50149867BDBM50149867({4-[5-Methoxy-2-(4-methoxy-phenylsulfanyl)-phenyl]...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50149855BDBM50149855({(2S,5R)-4-[2-(4-Methoxy-phenylsulfanyl)-phenyl]-2...)
Affinity DataIC50: 5.30E+4nMAssay Description:Inhibition of uptake of [3H]-glycine into cells transfected with human GlyT-1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed