Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50024447
TargetGlucagon receptor(Human)
Boehringer Ingelheim Pharma Gmbh And

Curated by ChEMBL
LigandPNGBDBM50269746(methyl (1S,5S,11S,17S,20S,23S,29S,32S,35S,38R,43R,...)
Affinity DataIC50: 320nMAssay Description:Antagonist activity at human glucagon receptor expressed in BHK21 cells assessed as inhibition of glucagon-induced cAMP elevation by RIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Boehringer Ingelheim Pharma Gmbh And

Curated by ChEMBL
LigandPNGBDBM50269738(BI-32169 | CHEMBL526383)
Affinity DataIC50: 440nMAssay Description:Antagonist activity at human glucagon receptor expressed in BHK21 cells assessed as inhibition of glucagon-induced cAMP elevation by RIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Boehringer Ingelheim Pharma Gmbh And

Curated by ChEMBL
LigandPNGBDBM50269745(cid_160115 | CHEMBL463175 | Cephalochromin)
Affinity DataIC50: 2.00E+4nMAssay Description:Antagonist activity at human glucagon receptor expressed in BHK21 cells assessed as inhibition of glucagon-induced cAMP elevation by RIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed