Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 50015288
TargetC-C chemokine receptor type 2(Human)
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50236430((R)-N-(2-(1-(4-chlorobenzyl)pyrrolidin-3-ylamino)-...)
Affinity DataEC50:  20nMAssay Description:Inhibition of MCP-1 induced chemotaxis in THP-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153942(N-({[1-(4-Chloro-benzyl)-piperidin-4-ylmethyl]-car...)
Affinity DataEC50:  40nMAssay Description:Inhibition of MCP-1 induced chemotaxis in THP-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50236430((R)-N-(2-(1-(4-chlorobenzyl)pyrrolidin-3-ylamino)-...)
Affinity DataIC50: 180nMAssay Description:Concentration required to inhibit [125I]MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50409951(CHEMBL2096789)
Affinity DataEC50:  360nMAssay Description:Inhibition of MCP-1 induced chemotaxis in THP-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153950(N-{[(R)-1-(4-Chloro-benzyl)-pyrrolidin-3-ylcarbamo...)
Affinity DataIC50: 370nMAssay Description:Concentration required to inhibit [125I]MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50409950(CHEMBL2096788)
Affinity DataIC50: 570nMAssay Description:Concentration required to inhibit [125I]MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50409950(CHEMBL2096788)
Affinity DataIC50: 570nMAssay Description:Concentration required to inhibit [125I]MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153938(N-{[1-(4-Chloro-benzyl)-piperidin-3-ylcarbamoyl]-m...)
Affinity DataEC50:  610nMAssay Description:Inhibition of MCP-1 induced chemotaxis in THP-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153938(N-{[1-(4-Chloro-benzyl)-piperidin-3-ylcarbamoyl]-m...)
Affinity DataIC50: 660nMAssay Description:Concentration required to inhibit [125I]MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153942(N-({[1-(4-Chloro-benzyl)-piperidin-4-ylmethyl]-car...)
Affinity DataIC50: 700nMAssay Description:Concentration required to inhibit [125I]MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153917(3-{1-Hydroxy-3-[4-(4-methanesulfonyl-benzyl)-[1,4]...)
Affinity DataIC50: 710nMAssay Description:Concentration required to inhibit [125I]MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50409950(CHEMBL2096788)
Affinity DataEC50:  810nMAssay Description:Inhibition of MCP-1 induced chemotaxis in THP-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50409950(CHEMBL2096788)
Affinity DataEC50:  810nMAssay Description:Inhibition of MCP-1 induced chemotaxis in THP-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50409951(CHEMBL2096789)
Affinity DataIC50: 1.20E+3nMAssay Description:Concentration required to inhibit [125I]MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153945(N-({[1-(4-Chloro-benzyl)-pyrrolidin-2-ylmethyl]-ca...)
Affinity DataIC50: 2.30E+3nMAssay Description:Concentration required to inhibit [125I]MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153940(N-({[1-(4-Chloro-benzyl)-piperidin-4-ylmethyl]-car...)
Affinity DataIC50: 5.50E+3nMAssay Description:Concentration required to inhibit [125I]MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153955(N-{[1-(4-Chloro-benzyl)-pyrrolidin-3-ylcarbamoyl]-...)
Affinity DataIC50: 6.90E+3nMAssay Description:Concentration required to inhibit [125I]MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153926(4-Methyl-thiophene-2-carboxylic acid N''-{2-[4-(4-...)
Affinity DataIC50: 7.40E+3nMAssay Description:Concentration required to inhibit [125I]MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153954(4-Methyl-thiophene-2-carboxylic acid N''-{2-[3-(4-...)
Affinity DataIC50: 7.80E+3nMAssay Description:Concentration required to inhibit [125I]MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153959(5-Oxo-5-phenyl-pentanoic acid [1-(4-chloro-benzyl)...)
Affinity DataIC50: 1.10E+4nMAssay Description:Concentration required to inhibit [125I]MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153960(N-({[1-(4-Chloro-benzyl)-piperidin-4-ylmethyl]-car...)
Affinity DataIC50: 1.10E+4nMAssay Description:Concentration required to inhibit [125I]MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153952(N-({[1-(4-Chloro-benzyl)-pyrrolidin-2-ylmethyl]-ca...)
Affinity DataIC50: 1.40E+4nMAssay Description:Concentration required to inhibit [125I]MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153951(N-{[1-(4-Chloro-benzyl)-piperidin-3-ylcarbamoyl]-m...)
Affinity DataIC50: 1.70E+4nMAssay Description:Concentration required to inhibit [125I]MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153948(4-Methyl-thiophene-2-carboxylic acid N''-{2-[3-(3,...)
Affinity DataIC50: 1.70E+4nMAssay Description:Concentration required to inhibit [125I]MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153943(5-Oxo-5-phenyl-pentanoic acid [1-(4-chloro-benzyl)...)
Affinity DataIC50: 1.90E+4nMAssay Description:Concentration required to inhibit [125I]MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153939(N-{2-[1-(4-Chloro-benzyl)-pyrrolidin-3-ylcarbamoyl...)
Affinity DataIC50: 2.20E+4nMAssay Description:Concentration required to inhibit [125I]MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153941(4-Methyl-thiophene-2-carboxylic acid N''-(2-{2-[(3...)
Affinity DataIC50: 2.60E+4nMAssay Description:Concentration required to inhibit [125I]MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153946(4-Methyl-thiophene-2-carboxylic acid N''-{2-[1-(3,...)
Affinity DataIC50: 3.30E+4nMAssay Description:Concentration required to inhibit [125I]MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153958(N-(2-{[1-(4-Chloro-benzyl)-pyrrolidin-2-ylmethyl]-...)
Affinity DataIC50: 4.00E+4nMAssay Description:Concentration required to inhibit [125I]MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153949(4-Methyl-thiophene-2-carboxylic acid N''-{2-[1-(4-...)
Affinity DataIC50: 4.10E+4nMAssay Description:Concentration required to inhibit [125I]MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153944(N-{[1-(4-Chloro-benzyl)-pyrrolidin-3-ylcarbamoyl]-...)
Affinity DataIC50: 4.20E+4nMAssay Description:Concentration required to inhibit [125I]MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153957(5-Oxo-5-phenyl-pentanoic acid [1-(4-chloro-benzyl)...)
Affinity DataIC50: 5.00E+4nMAssay Description:Concentration required to inhibit [125I]MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153956(N-(2-{[1-(4-Chloro-benzyl)-piperidin-4-ylmethyl]-c...)
Affinity DataIC50: 6.40E+4nMAssay Description:Concentration required to inhibit [125I]MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153947(N-({[1-(4-Chloro-benzyl)-pyrrolidin-2-ylmethyl]-ca...)
Affinity DataIC50: 6.60E+4nMAssay Description:Concentration required to inhibit [125I]MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153953(N-{2-[1-(4-Chloro-benzyl)-piperidin-3-ylcarbamoyl]...)
Affinity DataIC50: 7.40E+4nMAssay Description:Concentration required to inhibit [125I]MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 2(Human)
Deltagen Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50153961(5-Oxo-5-phenyl-pentanoic acid [1-(4-chloro-benzyl)...)
Affinity DataIC50: 8.70E+4nMAssay Description:Concentration required to inhibit [125I]MCP-1 binding to Chemokine receptor 2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed