Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50037461
TargetGlucocorticoid receptor(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM18627(Mifeprex | (10S,11S,14S,15S,17R)-17-[4-(dimethylam...)
Affinity DataIC50: 0.00800nMAssay Description:Inhibition of CHO-K1 cells expressing glucocorticoid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50154006(17-Hydroxy-13-methyl-11-pentyl-1,2,6,7,8,11,12,13,...)
Affinity DataIC50: 0.00900nMAssay Description:Inhibition of AR-dimerization in CHO-K1 cells expressing human androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50154006(17-Hydroxy-13-methyl-11-pentyl-1,2,6,7,8,11,12,13,...)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of human androgen receptor expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50422635(CHEMBL2311179)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of human androgen receptor expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50154003(11-Dodecyl-17-hydroxy-13-methyl-1,2,6,7,8,11,12,13...)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of human androgen receptor expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50154004(11-Decyl-17-hydroxy-13-methyl-1,2,6,7,8,11,12,13,1...)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human androgen receptor expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50154009(Acetic acid 17-acetyl-6-chloro-10,13-dimethyl-3-ox...)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of CHO-K1 cells expressing glucocorticoid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50154005(17-Hydroxy-13-methyl-11-octyl-1,2,6,7,8,11,12,13,1...)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of AR-dimerization in CHO-K1 cells expressing human androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50154007(11-Ethyl-17-hydroxy-13-methyl-1,2,6,7,8,11,12,13,1...)
Affinity DataIC50: 2nMAssay Description:Inhibition of human androgen receptor expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM18627(Mifeprex | (10S,11S,14S,15S,17R)-17-[4-(dimethylam...)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of human androgen receptor expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM8885(Testosterone, 1 | (1S,2R,10R,11S,14S,15S)-14-hydro...)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of human androgen receptor expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAndrogen receptor(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50154009(Acetic acid 17-acetyl-6-chloro-10,13-dimethyl-3-ox...)
Affinity DataIC50: 4.70nMAssay Description:Inhibition of AR-dimerization in CHO-K1 cells expressing human androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50154005(17-Hydroxy-13-methyl-11-octyl-1,2,6,7,8,11,12,13,1...)
Affinity DataIC50: 6.60nMAssay Description:Inhibition of human androgen receptor expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM18627(Mifeprex | (10S,11S,14S,15S,17R)-17-[4-(dimethylam...)
Affinity DataIC50: 7.80nMAssay Description:Inhibition of AR-dimerization in CHO-K1 cells expressing human androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50154004(11-Decyl-17-hydroxy-13-methyl-1,2,6,7,8,11,12,13,1...)
Affinity DataIC50: 17nMAssay Description:Inhibition of human lymph node carcinoma of prostate (LNCaP) cell proliferationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50154006(17-Hydroxy-13-methyl-11-pentyl-1,2,6,7,8,11,12,13,...)
Affinity DataIC50: 17nMAssay Description:Inhibition of human lymph node carcinoma of prostate (LNCaP) cell proliferationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50154005(17-Hydroxy-13-methyl-11-octyl-1,2,6,7,8,11,12,13,1...)
Affinity DataIC50: 17nMAssay Description:Inhibition of human lymph node carcinoma of prostate (LNCaP) cell proliferationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50154003(11-Dodecyl-17-hydroxy-13-methyl-1,2,6,7,8,11,12,13...)
Affinity DataIC50: 19nMAssay Description:Inhibition of human lymph node carcinoma of prostate (LNCaP) cell proliferationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50154009(Acetic acid 17-acetyl-6-chloro-10,13-dimethyl-3-ox...)
Affinity DataIC50: 22nMAssay Description:Inhibition of human androgen receptor expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM18627(Mifeprex | (10S,11S,14S,15S,17R)-17-[4-(dimethylam...)
Affinity DataIC50: 23nMAssay Description:Inhibition of human lymph node carcinoma of prostate (LNCaP) cell proliferationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50154007(11-Ethyl-17-hydroxy-13-methyl-1,2,6,7,8,11,12,13,1...)
Affinity DataIC50: 55nMAssay Description:Inhibition of human lymph node carcinoma of prostate (LNCaP) cell proliferationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50154009(Acetic acid 17-acetyl-6-chloro-10,13-dimethyl-3-ox...)
Affinity DataIC50: 61nMAssay Description:Inhibition of human lymph node carcinoma of prostate (LNCaP) cell proliferationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50154004(11-Decyl-17-hydroxy-13-methyl-1,2,6,7,8,11,12,13,1...)
Affinity DataIC50: 85nMAssay Description:Inhibition of AR-dimerization in CHO-K1 cells expressing human androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50422635(CHEMBL2311179)
Affinity DataIC50: 100nMAssay Description:Inhibition of human lymph node carcinoma of prostate (LNCaP) cell proliferationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50154006(17-Hydroxy-13-methyl-11-pentyl-1,2,6,7,8,11,12,13,...)
Affinity DataIC50: 125nMAssay Description:Inhibition of CHO-K1 cells expressing glucocorticoid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50422635(CHEMBL2311179)
Affinity DataIC50: 133nMAssay Description:Inhibition of CHO-K1 cells expressing glucocorticoid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50154003(11-Dodecyl-17-hydroxy-13-methyl-1,2,6,7,8,11,12,13...)
Affinity DataIC50: 870nMAssay Description:Inhibition of CHO-K1 cells expressing glucocorticoid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50154005(17-Hydroxy-13-methyl-11-octyl-1,2,6,7,8,11,12,13,1...)
Affinity DataIC50: 979nMAssay Description:Inhibition of CHO-K1 cells expressing glucocorticoid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50154007(11-Ethyl-17-hydroxy-13-methyl-1,2,6,7,8,11,12,13,1...)
Affinity DataIC50: 1.29E+3nMAssay Description:Inhibition of CHO-K1 cells expressing glucocorticoid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50154004(11-Decyl-17-hydroxy-13-methyl-1,2,6,7,8,11,12,13,1...)
Affinity DataIC50: 1.81E+3nMAssay Description:Inhibition of CHO-K1 cells expressing glucocorticoid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed