Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50015417
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155833BDBM50155833(3-[4-(2,4-Bis-trifluoromethyl-benzyloxy)-3-methoxy...)
Affinity DataIC50: 370nMAssay Description:Inhibition of estrogen-related receptor alpha Gal4 activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155821BDBM50155821(3-[4-(2,4-Bis-trifluoromethyl-benzyloxy)-3-methoxy...)
Affinity DataIC50: 400nMAssay Description:Inhibition of estrogen-related receptor alpha Gal4 activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155821BDBM50155821(3-[4-(2,4-Bis-trifluoromethyl-benzyloxy)-3-methoxy...)
Affinity DataIC50: 400nMAssay Description:Inhibition of estrogen-related receptor alpha Gal4 activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155832BDBM50155832(3-[4-(2,4-Bis-trifluoromethyl-benzyloxy)-3-methoxy...)
Affinity DataIC50: 440nMAssay Description:Inhibition of estrogen-related receptor alpha Gal4 activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155822BDBM50155822(3-[4-(2,4-Bis-trifluoromethyl-benzyloxy)-3-methoxy...)
Affinity DataIC50: 500nMAssay Description:Inhibition of estrogen-related receptor alpha Gal4 activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155821BDBM50155821(3-[4-(2,4-Bis-trifluoromethyl-benzyloxy)-3-methoxy...)
Affinity DataIC50: 610nMAssay Description:Inhibition of estrogen-related receptor alpha Gal4 activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155825BDBM50155825(3-[4-(2,4-Bis-trifluoromethyl-benzyloxy)-3-methoxy...)
Affinity DataIC50: 750nMAssay Description:Inhibition of estrogen-related receptor alpha Gal4 activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155820BDBM50155820(2-Cyano-N-(5-ethyl-[1,3,4]thiadiazol-2-yl)-3-[4-(5...)
Affinity DataIC50: 800nMAssay Description:Inhibition of estrogen-related receptor alpha Gal4 activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155820BDBM50155820(2-Cyano-N-(5-ethyl-[1,3,4]thiadiazol-2-yl)-3-[4-(5...)
Affinity DataIC50: 800nMAssay Description:Inhibition of estrogen-related receptor alpha Gal4 activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155830BDBM50155830(2-Cyano-N-(5-ethyl-[1,3,4]thiadiazol-2-yl)-3-[4-(4...)
Affinity DataIC50: 920nMAssay Description:Inhibition of estrogen-related receptor alpha Gal4 activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155830BDBM50155830(2-Cyano-N-(5-ethyl-[1,3,4]thiadiazol-2-yl)-3-[4-(4...)
Affinity DataIC50: 920nMAssay Description:Inhibition of estrogen-related receptor alpha Gal4 activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155828BDBM50155828(6-[1-{4-[2-(2,6-Dimethyl-phenoxy)-ethoxy]-3-methox...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of estrogen-related receptor alpha in FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155815BDBM50155815(2-Cyano-3-{4-[2-(2,6-dimethyl-phenoxy)-ethoxy]-3-m...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of estrogen-related receptor alpha Gal4 activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155817BDBM50155817(2-Cyano-3-{4-[2-(2,6-dimethyl-phenoxy)-ethoxy]-3-m...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of estrogen-related receptor alpha Gal4 activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155819BDBM50155819(N-(5-tert-Butyl-[1,3,4]thiadiazol-2-yl)-2-cyano-3-...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of estrogen-related receptor alpha Gal4 activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155831BDBM50155831(2-Cyano-N-(5-ethyl-[1,3,4]thiadiazol-2-yl)-3-[3-me...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of estrogen-related receptor alpha Gal4 activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155824BDBM50155824(2-Cyano-N-(5-ethyl-[1,3,4]thiadiazol-2-yl)-3-[3-me...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of estrogen-related receptor alpha Gal4 activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155823BDBM50155823(2-Cyano-3-{4-[2-(2,6-dimethyl-phenoxy)-ethoxy]-3-m...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of estrogen-related receptor alpha Gal4 activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155829BDBM50155829(2-Cyano-N-[5-(4-dimethylamino-phenyl)-[1,3,4]thiad...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of estrogen-related receptor alpha Gal4 activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155816BDBM50155816(3-[4-(2-Bromo-benzyloxy)-3-methoxy-phenyl]-2-cyano...)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of estrogen-related receptor alpha Gal4 activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155828BDBM50155828(6-[1-{4-[2-(2,6-Dimethyl-phenoxy)-ethoxy]-3-methox...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of estrogen-related receptor alpha Gal4 activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155827BDBM50155827(2-Cyano-3-{4-[2-(2,6-dimethyl-phenoxy)-ethoxy]-3-m...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of estrogen-related receptor alpha Gal4 activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155826BDBM50155826(2-Cyano-3-{4-[2-(2,6-dimethyl-phenoxy)-ethoxy]-3-m...)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of estrogen-related receptor alpha Gal4 activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155818BDBM50155818(3-[4-(2,4-Bis-trifluoromethyl-benzyloxy)-3-methoxy...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of estrogen-related receptor alpha Gal4 activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed