Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50003730
TargetKappa-type opioid receptor(Human)
University of Bath

Curated by ChEMBL
LigandPNGBDBM82551(C18130 | CAS_105618-26-6 | NORBNI | NOR-BNI (HCI)2)
Affinity DataKi:  0.400nMAssay Description:Inhibition of [3H]diprenorphine binding to human opioid receptor kappa 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50475335(CHEMBL2113078)
Affinity DataKi:  0.700nMAssay Description:Inhibition of [3H]diprenorphine binding to human opioid receptor kappa 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bath

Curated by ChEMBL
LigandPNGBDBM82551(C18130 | CAS_105618-26-6 | NORBNI | NOR-BNI (HCI)2)
Affinity DataKi:  1.20nMAssay Description:Inhibition of [3H]diprenorphine binding to rat Opioid receptor mu 1 expressed in C6 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Bath

Curated by ChEMBL
LigandPNGBDBM82551(C18130 | CAS_105618-26-6 | NORBNI | NOR-BNI (HCI)2)
Affinity DataKi:  5.80nMAssay Description:Inhibition of [3H]diprenorphine binding to rat Opioid receptor delta 1 expressed in C6 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50475334(CHEMBL2113073)
Affinity DataKi:  6.40nMAssay Description:Inhibition of [3H]diprenorphine binding to rat Opioid receptor mu 1 expressed in C6 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50475336(CHEMBL606959)
Affinity DataKi:  7.70nMAssay Description:Inhibition of [3H]diprenorphine binding to human opioid receptor kappa 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50475335(CHEMBL2113078)
Affinity DataKi:  8.60nMAssay Description:Inhibition of [3H]diprenorphine binding to rat Opioid receptor delta 1 expressed in C6 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50475335(CHEMBL2113078)
Affinity DataKi:  10nMAssay Description:Inhibition of [3H]diprenorphine binding to rat Opioid receptor mu 1 expressed in C6 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50475334(CHEMBL2113073)
Affinity DataKi:  25nMAssay Description:Inhibition of [3H]diprenorphine binding to human opioid receptor kappa 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50475336(CHEMBL606959)
Affinity DataKi:  64nMAssay Description:Inhibition of [3H]diprenorphine binding to rat Opioid receptor mu 1 expressed in C6 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50475336(CHEMBL606959)
Affinity DataKi:  98nMAssay Description:Inhibition of [3H]diprenorphine binding to rat Opioid receptor delta 1 expressed in C6 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50475335(CHEMBL2113078)
Affinity DataEC50:  187nMAssay Description:Agonist activity against rat Opioid receptor mu 1 expressed in C6 cells in [35S]-GTP-gamma S binding assay More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50475334(CHEMBL2113073)
Affinity DataKi:  207nMAssay Description:Inhibition of [3H]diprenorphine binding to rat Opioid receptor delta 1 expressed in C6 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50475334(CHEMBL2113073)
Affinity DataEC50:  526nMAssay Description:Agonist activity against rat Opioid receptor mu 1 expressed in C6 cells in [35S]-GTP-gamma S binding assay More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50475336(CHEMBL606959)
Affinity DataEC50:  1.39E+3nMAssay Description:Agonist activity against rat Opioid receptor mu 1 expressed in C6 cells in [35S]-GTP-gamma S binding assay More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50475335(CHEMBL2113078)
Affinity DataEC50:  1.91E+3nMAssay Description:Agonist activity against human Opioid receptor kappa 1 expressed in CHO cells in [35S]-GTP-gamma S binding assay More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed