Compile Data Set for Download or QSAR
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Found 29 Enz. Inhib. hit(s) with all data for entry = 50037442
TargetEukaryotic translation initiation factor 4E(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50410170(CHEMBL2079703)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 4E(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50370488(CHEMBL607618)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 4E(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50410173(CHEMBL2079719)
Affinity DataIC50:  4.50E+4nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 4E(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50370490(CHEMBL610599)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 4E(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50410172(CHEMBL2079724)
Affinity DataIC50:  5.50E+4nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 4E(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50410171(CHEMBL2079700)
Affinity DataIC50:  7.00E+4nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 4E(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50410174(CHEMBL2079702)
Affinity DataIC50:  8.50E+4nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 4E(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50370482(CHEMBL610852)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 4E(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50370491(CHEMBL611110)
Affinity DataIC50:  1.30E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 4E(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50165117(2-amino-6-hydroxy-9-[(2R,4S,5R)-5-[(phosphinatooxy...)
Affinity DataIC50:  1.80E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 4E(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50370487(CHEMBL609052)
Affinity DataIC50:  2.00E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 4E(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50370492(CHEMBL607905)
Affinity DataIC50:  2.20E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 4E(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50370481(CHEMBL611113)
Affinity DataIC50:  2.20E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 4E(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50165135(CHEMBL193790 | disodium 2-amino-9-[(2R,4S,5R)-5-[(...)
Affinity DataIC50:  4.00E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 4E(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50370484(CHEMBL611105)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 4E(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50370483(CHEMBL607903)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 4E(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50370489(CHEMBL607902)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 4E(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50165127(2-Amino-9-((2R,4S,5R)-5-hydroxymethyl-3,4-diisopro...)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 4E(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50165122(CHEMBL195283 | disodium 2-amino-9-[(2R,4S,5R)-5-[(...)
Affinity DataIC50:  4.00E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 4E(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50165142(CHEMBL194978 | disodium 2-amino-9-[(2R,4S,5R)-5-[(...)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 4E(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50165141(CHEMBL436762 | disodium 2-amino-9-[(2R,4S,5R)-5-{[...)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 4E(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50370493(CHEMBL609636)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 4E(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50410169(CHEMBL2021409)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 4E(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50165119(2-Amino-9-((2R,4S,5R)-5-hydroxymethyl-3,4-diisopro...)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 4E(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50165118(2-Amino-7-benzyl-9-((2R,4S,5R)-5-hydroxymethyl-3,4...)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 4E(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50165116(CHEMBL194007 | tetrasodium ({[(2R,3R,5R)-5-(2-amin...)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 4E(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50165134(2-Amino-7-ethyl-9-((2R,4S,5R)-5-hydroxymethyl-3,4-...)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 4E(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50370485(CHEMBL611114)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 4E(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50370486(CHEMBL611097)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibitory concentration against 7-methyl-GTP binding to eukaryotic translation initiation factor 4EMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed