Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 1545
TargetFalcipain-2(malaria parasite P. falciparum)
Universidad Central De Venezuela

LigandPNGBDBM12041(Acetyl-Leu-Leu-Arg-CHO | (2S)-2-({5-[(diaminomethy...)
Affinity DataIC50: 5.80nMpH: 5.5 T: 2°CAssay Description:The substrate peptide terminating in AMC is processed by falcipain-2 with or without inhibitors, and the accumulation of AMC was monitored in a Labsy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2006
Entry Details Article
PubMed
TargetFalcipain-2(malaria parasite P. falciparum)
Universidad Central De Venezuela

LigandPNGBDBM12042(L-trans-3-Carboxyoxiran-2-carbonyl-L-leucylagmatin...)
Affinity DataIC50: 58nMpH: 5.5 T: 2°CAssay Description:The substrate peptide terminating in AMC is processed by falcipain-2 with or without inhibitors, and the accumulation of AMC was monitored in a Labsy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2006
Entry Details Article
PubMed
TargetFalcipain-2(malaria parasite P. falciparum)
Universidad Central De Venezuela

LigandPNGBDBM12037(3-(4-chlorophenyl)-1-{4-[(2E)-3-(3,4,5-trimethoxyp...)
Affinity DataIC50: 1.80E+3nMpH: 5.5 T: 2°CAssay Description:The substrate peptide terminating in AMC is processed by falcipain-2 with or without inhibitors, and the accumulation of AMC was monitored in a Labsy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2006
Entry Details Article
PubMed
TargetFalcipain-2(malaria parasite P. falciparum)
Universidad Central De Venezuela

LigandPNGBDBM12032(1-{4-[(2E)-3-(2H-1,3-benzodioxol-5-yl)prop-2-enoyl...)
Affinity DataIC50: 2.50E+3nMpH: 5.5 T: 2°CAssay Description:The substrate peptide terminating in AMC is processed by falcipain-2 with or without inhibitors, and the accumulation of AMC was monitored in a Labsy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2006
Entry Details Article
PubMed
TargetFalcipain-2(malaria parasite P. falciparum)
Universidad Central De Venezuela

LigandPNGBDBM12035(3-(4-chlorophenyl)-1-{4-[(2E)-3-(2,4-dichloropheny...)
Affinity DataIC50: 2.50E+3nMpH: 5.5 T: 2°CAssay Description:The substrate peptide terminating in AMC is processed by falcipain-2 with or without inhibitors, and the accumulation of AMC was monitored in a Labsy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2006
Entry Details Article
PubMed
TargetFalcipain-2(malaria parasite P. falciparum)
Universidad Central De Venezuela

LigandPNGBDBM12034(3-(4-chlorophenyl)-1-{4-[(2E)-3-(4-chlorophenyl)pr...)
Affinity DataIC50: 2.60E+3nMpH: 5.5 T: 2°CAssay Description:The substrate peptide terminating in AMC is processed by falcipain-2 with or without inhibitors, and the accumulation of AMC was monitored in a Labsy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2006
Entry Details Article
PubMed
TargetFalcipain-2(malaria parasite P. falciparum)
Universidad Central De Venezuela

LigandPNGBDBM12036(3-(4-chlorophenyl)-1-{4-[(2E)-3-(2,4-difluoropheny...)
Affinity DataIC50: 2.60E+3nMpH: 5.5 T: 2°CAssay Description:The substrate peptide terminating in AMC is processed by falcipain-2 with or without inhibitors, and the accumulation of AMC was monitored in a Labsy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2006
Entry Details Article
PubMed
TargetFalcipain-2(malaria parasite P. falciparum)
Universidad Central De Venezuela

LigandPNGBDBM12039(3-(4-chlorophenyl)-1-{4-[(2E)-3-(pyridin-3-yl)prop...)
Affinity DataIC50: 3.40E+3nMpH: 5.5 T: 2°CAssay Description:The substrate peptide terminating in AMC is processed by falcipain-2 with or without inhibitors, and the accumulation of AMC was monitored in a Labsy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2006
Entry Details Article
PubMed
TargetFalcipain-2(malaria parasite P. falciparum)
Universidad Central De Venezuela

LigandPNGBDBM12038(3-(4-chlorophenyl)-1-{4-[(2E)-3-phenylprop-2-enoyl...)
Affinity DataIC50: 3.80E+3nMpH: 5.5 T: 2°CAssay Description:The substrate peptide terminating in AMC is processed by falcipain-2 with or without inhibitors, and the accumulation of AMC was monitored in a Labsy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2006
Entry Details Article
PubMed
TargetFalcipain-2(malaria parasite P. falciparum)
Universidad Central De Venezuela

LigandPNGBDBM12040(3-(4-methoxyphenyl)-1-{4-[(2E)-3-(pyridin-3-yl)pro...)
Affinity DataIC50: 1.25E+4nMpH: 5.5 T: 2°CAssay Description:The substrate peptide terminating in AMC is processed by falcipain-2 with or without inhibitors, and the accumulation of AMC was monitored in a Labsy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2006
Entry Details Article
PubMed