Compile Data Set for Download or QSAR
maximum 50k data
Found 18 Enz. Inhib. hit(s) with all data for entry = 50016585
TargetSubstance-K receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50170969((S)-1-(1-Cyclopropyl-cyclopentyl)-5-(3,4-dichloro-...)
Affinity DataKi:  9.50E+3nMAssay Description:Ki for human Neurokinin 2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50170967((S)-1-(1-Cyclopropyl-cyclopentyl)-5-(3,4-dichloro-...)
Affinity DataKi:  1.00E+4nMAssay Description:Ki for human Neurokinin 2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50170968((S)-5-(3,4-Dichloro-phenyl)-1-(4,4-difluoro-cycloh...)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of human Neurokinin 2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50409627(CHEMBL185572)
Affinity DataIC50:  0.790nMAssay Description:Inhibition of human Neurokinin 2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50410049(CHEMBL434142)
Affinity DataIC50:  1nMAssay Description:Inhibition of human Neurokinin 2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50410051(CHEMBL185182)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of human Neurokinin 2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50410048(CHEMBL434548)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of human Neurokinin 2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50410054(CHEMBL185133)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of human Neurokinin 2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50410052(CHEMBL367815)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of human Neurokinin 2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50410047(CHEMBL365613 | UK-224671)
Affinity DataIC50:  4nMAssay Description:Inhibition of human Neurokinin 2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50410046(CHEMBL367348)
Affinity DataIC50:  6.30nMAssay Description:Inhibition of human Neurokinin 2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50410058(CHEMBL185452)
Affinity DataIC50:  7.90nMAssay Description:Inhibition of human Neurokinin 2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50410057(CHEMBL359655)
Affinity DataIC50:  7.90nMAssay Description:Inhibition of human Neurokinin 2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50410050(CHEMBL359903)
Affinity DataIC50:  10nMAssay Description:Inhibition of human Neurokinin 2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50410056(CHEMBL185007)
Affinity DataIC50:  16nMAssay Description:Inhibition of human Neurokinin 2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50410055(CHEMBL180049)
Affinity DataIC50:  16nMAssay Description:Inhibition of human Neurokinin 2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50410053(CHEMBL360721)
Affinity DataIC50:  79nMAssay Description:Inhibition of human Neurokinin 2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50170968((S)-5-(3,4-Dichloro-phenyl)-1-(4,4-difluoro-cycloh...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory concentration for Tachykinin 1 receptor of human IM9 cells More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed