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Found 6 Enz. Inhib. hit(s) with all data for entry = 50003735
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50223597(CHEMBL95777)
Affinity DataIC50:  1.82E+4nMAssay Description:Inhibitory activity against supercoiling activity of DNA gyrase isolated from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50223617(CHEMBL95778)
Affinity DataIC50:  3.10E+4nMAssay Description:Inhibitory activity against supercoiling activity of DNA gyrase isolated from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 4 subunit A(Escherichia coli (strain K12))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50223597(CHEMBL95777)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibitory activity against decatenation of DNA topoisomerase IV isolated from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50475386(CHEMBL194702)
Affinity DataIC50:  3.26E+4nMAssay Description:Inhibitory activity against supercoiling activity of DNA gyrase isolated from Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 4 subunit A(Escherichia coli (strain K12))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50223617(CHEMBL95778)
Affinity DataIC50:  3.54E+4nMAssay Description:Inhibitory activity against decatenation of DNA topoisomerase IV isolated from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 4 subunit A(Escherichia coli (strain K12))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50475386(CHEMBL194702)
Affinity DataIC50:  6.53E+4nMAssay Description:Inhibitory activity against decatenation of DNA topoisomerase IV isolated from Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed