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Found 10 Enz. Inhib. hit(s) with all data for entry = 50016689
TargetMu-type opioid receptor(GUINEA PIG)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50172014(CHEMBL371856 | H-Dmt-D-Arg(NO2)-Phe-Lys(Z)-NH2)
Affinity DataIC50:  0.509nMAssay Description:Agonist activity against mu opioid receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50010483(CHEMBL2181202)
Affinity DataIC50:  1.40nMAssay Description:Agonist activity against mu opioid receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50172014(CHEMBL371856 | H-Dmt-D-Arg(NO2)-Phe-Lys(Z)-NH2)
Affinity DataIC50:  1.70nMAssay Description:Agonistic activity against delta opioid receptor of mouse vas deferens assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50010483(CHEMBL2181202)
Affinity DataIC50:  23nMAssay Description:Agonistic activity against delta opioid receptor of mouse vas deferens assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50172013(CHEMBL370701 | H-Dmt-D-Arg(NO2)-Phe-Lys(Z)-OH)
Affinity DataIC50:  63nMAssay Description:Agonist activity against mu opioid receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50172013(CHEMBL370701 | H-Dmt-D-Arg(NO2)-Phe-Lys(Z)-OH)
Affinity DataIC50:  682nMAssay Description:Agonistic activity against delta opioid receptor of mouse vas deferens assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50172017(CHEMBL3143756 | {(S)-5-[(S)-2-({2-[2-Amino-3-(4-hy...)
Affinity DataIC50:  1.89E+3nMAssay Description:Agonist activity against mu opioid receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50172017(CHEMBL3143756 | {(S)-5-[(S)-2-({2-[2-Amino-3-(4-hy...)
Affinity DataIC50: >1.00E+4nMAssay Description:Agonistic activity against delta opioid receptor of mouse vas deferens assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50172015((S)-2-[(S)-2-({2-[2-Amino-3-(4-hydroxy-2,6-dimethy...)
Affinity DataIC50: >1.00E+4nMAssay Description:Agonist activity against mu opioid receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50172015((S)-2-[(S)-2-({2-[2-Amino-3-(4-hydroxy-2,6-dimethy...)
Affinity DataIC50: >1.00E+4nMAssay Description:Agonistic activity against delta opioid receptor of mouse vas deferens assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed