Compile Data Set for Download or QSAR
maximum 50k data
Found 46 Enz. Inhib. hit(s) with all data for entry = 50016744
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173019(4-(4-(4-tert-butylphenylamino)phthalazin-1-yl)benz...)
Affinity DataIC50:  78nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173031(4-(4-(4-bromophenylamino)phthalazin-1-yl)benzamide...)
Affinity DataIC50:  100nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173045(4-(4-(4-tert-butylphenylamino)phthalazin-1-yl)-N-m...)
Affinity DataIC50:  130nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173049(4-(4-(4-(chlorodifluoromethoxy)phenylamino)phthala...)
Affinity DataIC50:  190nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173007(4-[4-(4-Chloro-phenylamino)-phthalazin-1-yl]-benzo...)
Affinity DataIC50:  360nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173022(3-(4-(4-tert-butylphenylamino)phthalazin-1-yl)benz...)
Affinity DataIC50:  400nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173034(4-(4-(3-tert-butylphenylamino)phthalazin-1-yl)benz...)
Affinity DataIC50:  470nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173021(4-{4-[4-(Chloro-difluoro-methoxy)-phenylamino]-pht...)
Affinity DataIC50:  630nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173051(4-(4-(3,4-dichlorophenylamino)phthalazin-1-yl)benz...)
Affinity DataIC50:  840nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173024(4-(4-(4-(chlorodifluoromethoxy)phenylamino)phthala...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173041(3,5-dimethoxy-N-(1-(naphthalen-2-ylmethyl)piperidi...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173011(4-(4-(4-chlorophenylamino)phthalazin-1-yl)benzamid...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173029(4-(4-(m-tolylamino)phthalazin-1-yl)benzamide | 4-(...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173012(4-(4-(3-chlorophenylamino)phthalazin-1-yl)benzamid...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173017(4-(4-(p-tolylamino)phthalazin-1-yl)benzamide | 4-(...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173043(4-(4-(4-methoxyphenylamino)phthalazin-1-yl)benzami...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173025(4-[4-(4-Carbamoyl-phenyl)-phthalazin-1-ylamino]-be...)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173013(4-(4-(4-chlorophenylamino)phthalazin-1-yl)-N-methy...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173047(3-(4-(4-(chlorodifluoromethoxy)phenylamino)phthala...)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173020((4-(4-(4-(chlorodifluoromethoxy)phenylamino)phthal...)
Affinity DataIC50:  4.90E+3nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173040(4-[4-(2,4-Dimethyl-phenylamino)-phthalazin-1-yl]-b...)
Affinity DataIC50:  6.90E+3nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173048(5-{4-[4-(Chloro-difluoro-methoxy)-phenylamino]-pht...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173050(4-(4-(4-(trifluoromethoxy)phenylthio)phthalazin-1-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173052(5-{4-[4-(Chloro-difluoro-methoxy)-phenylamino]-pht...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173042(4-(4-(4-carbamoylphenyl)phthalazin-1-ylamino)benza...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173014(CHEMBL364974 | N-(4-(chlorodifluoromethoxy)phenyl)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173038((3,4-Dichloro-phenyl)-(4-p-tolyl-phthalazin-1-yl)-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173046(CHEMBL196657 | [4-(4-Ethoxy-phenyl)-phthalazin-1-y...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173044(CHEMBL194138 | [4-(Chloro-difluoro-methoxy)-phenyl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173036(4-[4-(4-Pyridin-1-yl-phenylamino)-phthalazin-1-yl]...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173039((4-Chloro-phenyl)-(4-p-tolyl-phthalazin-1-yl)-amin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173037(CHEMBL195727 | N-(4-(chlorodifluoromethoxy)phenyl)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173035((4-Chloro-phenyl)-[4-(4-ethoxy-phenyl)-phthalazin-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173033((3,4-Dichloro-phenyl)-[4-(4-methoxy-phenyl)-phthal...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173027(CHEMBL196940 | N,N-Dimethyl-4-(4-p-tolylamino-phth...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173028(4-(4-(4-(benzyloxy)phenylamino)phthalazin-1-yl)ben...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173030(4-[4-(4-Sulfamoyl-phenylamino)-phthalazin-1-yl]-be...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173032(4-[4-(4-Morpholin-4-yl-phenylamino)-phthalazin-1-y...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173026(CHEMBL370206 | [4-(4-Ethoxy-phenyl)-phthalazin-1-y...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173023((4-Methoxy-phenyl)-(4-phenyl-phthalazin-1-yl)-amin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173018(CHEMBL195829 | N-(4-(chlorodifluoromethoxy)phenyl)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173015(CHEMBL196422 | N-tert-Butyl-4-{4-[4-(chloro-difluo...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173010((4-Chloro-phenyl)-[4-(4-methoxy-phenyl)-phthalazin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173008(4-(4-(4-(trifluoromethoxy)phenoxy)phthalazin-1-yl)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173016(4-(4-(phenylamino)phthalazin-1-yl)benzamide | 4-(4...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173009(4-(4-(4-(chlorodifluoromethoxy)phenylamino)phthala...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed