Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) with all data for entry = 50016843
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50174266(CHEMBL198525 | N-(2-(4-(1H-indol-3-yl)-5,6-dihydro...)
Affinity DataIC50:  2nMAssay Description:Inhibitory activity against human SERT transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50174266(CHEMBL198525 | N-(2-(4-(1H-indol-3-yl)-5,6-dihydro...)
Affinity DataIC50:  30nMAssay Description:Inhibitory activity of compound bound to streptavidin-conjugated quantum dots against human SERT transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50174265(2-(2-(2-(3-(2-aminoethyl)-1H-indol-5-yloxy)ethoxy)...)
Affinity DataIC50:  9.90E+4nMAssay Description:Inhibitory activity of compound bound to streptavidin-conjugated quantum dots against human SERT transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50174265(2-(2-(2-(3-(2-aminoethyl)-1H-indol-5-yloxy)ethoxy)...)
Affinity DataIC50:  1.15E+5nMAssay Description:Inhibitory activity against human SERT transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed