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Found 136 Enz. Inhib. hit(s) with all data for entry = 50017041
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176751(8-(1-((3-phenyl-1,2,4-oxadiazol-5-yl)methyl)-1H-py...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50233091(8-(1-((5-phenylisoxazol-3-yl)methyl)-1H-pyrazol-4-...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176739(4-(3-((4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydr...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176757(4-(5-((4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydr...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176769(8-(1-((3-(2-chlorophenyl)-1,2,4-oxadiazol-5-yl)met...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176740(8-(1-((3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl)met...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50233109(8-(1-((5-phenyl-1,2,4-oxadiazol-3-yl)methyl)-1H-py...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176738(1,3-dipropyl-8-(1-((5-(4-(trifluoromethyl)phenyl)-...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176736(CHEMBL200780 | N-(2-chlorophenyl)-2-(4-(2,6-dioxo-...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176752(8-(1-((3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl)met...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176768(8-(1-((5-(2-chlorophenyl)-1,2,4-oxadiazol-3-yl)met...)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176748(8-(1-((5-(4-chlorophenyl)-1,2,4-oxadiazol-3-yl)met...)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176737(1,3-dipropyl-8-(1-((3-(3-(trifluoromethyl)phenyl)-...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176755(1,3-dipropyl-8-(1-((5-(4-(trifluoromethyl)phenyl)i...)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176767(1,3-dipropyl-8-(1-((3-p-tolyl-1,2,4-oxadiazol-5-yl...)
Affinity DataKi:  54nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176756(1,3-dipropyl-8-(1-((3-(4-(trifluoromethyl)phenyl)-...)
Affinity DataKi:  55nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176763(8-(1-((5-(4-methoxyphenyl)isoxazol-3-yl)methyl)-1H...)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176759(1,3-dipropyl-8-(1-((5-(3-(trifluoromethyl)phenyl)-...)
Affinity DataKi:  64nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176742(1,3-dipropyl-8-(1-((3-(2-(trifluoromethyl)phenyl)-...)
Affinity DataKi:  74nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176749(8-(1-((3-(3-methoxyphenyl)-1,2,4-oxadiazol-5-yl)me...)
Affinity DataKi:  82nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176745(8-(1-((3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl)me...)
Affinity DataKi:  82nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176754(8-(1-((5-(4-chlorophenyl)isoxazol-3-yl)methyl)-1H-...)
Affinity DataKi:  82nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176762(8-(1-((5-(2-methoxyphenyl)-1,2,4-oxadiazol-3-yl)me...)
Affinity DataKi:  83nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176743(1,3-dipropyl-8-(1-((5-(2-(trifluoromethyl)phenyl)-...)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176736(CHEMBL200780 | N-(2-chlorophenyl)-2-(4-(2,6-dioxo-...)
Affinity DataKi:  102nMAssay Description:Displacement of [3H]CPX from Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176744(8-(1-((3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl)me...)
Affinity DataKi:  106nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176761(8-(1-((5-(2-chlorophenyl)isoxazol-3-yl)methyl)-1H-...)
Affinity DataKi:  111nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176750(1,3-dipropyl-8-(1-((5-(2-(trifluoromethyl)phenyl)i...)
Affinity DataKi:  121nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176747(8-(1-((5-(4-methoxyphenyl)-1,2,4-oxadiazol-3-yl)me...)
Affinity DataKi:  123nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176766(1,3-dipropyl-8-(1-((3-m-tolyl-1,2,4-oxadiazol-5-yl...)
Affinity DataKi:  128nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176765(8-(1-((5-(3-methoxyphenyl)isoxazol-3-yl)methyl)-1H...)
Affinity DataKi:  131nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176746(8-(1-((5-(3-chlorophenyl)-1,2,4-oxadiazol-3-yl)met...)
Affinity DataKi:  134nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176741(8-(1-((5-(3-methoxyphenyl)-1,2,4-oxadiazol-3-yl)me...)
Affinity DataKi:  136nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176764(8-(1-((5-(3-chlorophenyl)isoxazol-3-yl)methyl)-1H-...)
Affinity DataKi:  163nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176753(8-(1-((5-(2-methoxyphenyl)isoxazol-3-yl)methyl)-1H...)
Affinity DataKi:  195nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176768(8-(1-((5-(2-chlorophenyl)-1,2,4-oxadiazol-3-yl)met...)
Affinity DataKi:  330nMAssay Description:Displacement of [125I]AB-MECA from Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176742(1,3-dipropyl-8-(1-((3-(2-(trifluoromethyl)phenyl)-...)
Affinity DataKi:  340nMAssay Description:Displacement of [125I]AB-MECA from Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176751(8-(1-((3-phenyl-1,2,4-oxadiazol-5-yl)methyl)-1H-py...)
Affinity DataKi:  370nMAssay Description:Displacement of [3H]CPX from Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176740(8-(1-((3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl)met...)
Affinity DataKi:  400nMAssay Description:Displacement of [125I]AB-MECA from Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176745(8-(1-((3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl)me...)
Affinity DataKi:  410nMAssay Description:Displacement of [125I]AB-MECA from Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50233091(8-(1-((5-phenylisoxazol-3-yl)methyl)-1H-pyrazol-4-...)
Affinity DataKi:  420nMAssay Description:Displacement of [3H]ZM241385 from Adenosine A2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176751(8-(1-((3-phenyl-1,2,4-oxadiazol-5-yl)methyl)-1H-py...)
Affinity DataKi:  480nMAssay Description:Displacement of [125I]AB-MECA from Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176769(8-(1-((3-(2-chlorophenyl)-1,2,4-oxadiazol-5-yl)met...)
Affinity DataKi:  490nMAssay Description:Displacement of [125I]AB-MECA from Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176752(8-(1-((3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl)met...)
Affinity DataKi:  490nMAssay Description:Displacement of [125I]AB-MECA from Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176742(1,3-dipropyl-8-(1-((3-(2-(trifluoromethyl)phenyl)-...)
Affinity DataKi:  530nMAssay Description:Displacement of [3H]CPX from Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176754(8-(1-((5-(4-chlorophenyl)isoxazol-3-yl)methyl)-1H-...)
Affinity DataKi:  540nMAssay Description:Displacement of [3H]CPX from Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176739(4-(3-((4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydr...)
Affinity DataKi:  570nMAssay Description:Displacement of [3H]CPX from Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176749(8-(1-((3-(3-methoxyphenyl)-1,2,4-oxadiazol-5-yl)me...)
Affinity DataKi:  600nMAssay Description:Displacement of [125I]AB-MECA from Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50176743(1,3-dipropyl-8-(1-((5-(2-(trifluoromethyl)phenyl)-...)
Affinity DataKi:  620nMAssay Description:Displacement of [125I]AB-MECA from Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50233109(8-(1-((5-phenyl-1,2,4-oxadiazol-3-yl)methyl)-1H-py...)
Affinity DataKi:  630nMAssay Description:Displacement of [125I]AB-MECA from Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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