Compile Data Set for Download or QSAR
Report error Found 61 Enz. Inhib. hit(s) with all data for entry = 50017049
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176833(methyl 4-(4-methoxyphenethylamino)-1-(2-chloro-2-p...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176833(methyl 4-(4-methoxyphenethylamino)-1-(2-chloro-2-p...)
Affinity DataKi:  6.30nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranes in absence of GTPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176822(isopropyl 4-(4-methoxyphenethylamino)-1-(2-chloro-...)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176822(isopropyl 4-(4-methoxyphenethylamino)-1-(2-chloro-...)
Affinity DataKi:  7.20nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranes in absence of GTPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176833(methyl 4-(4-methoxyphenethylamino)-1-(2-chloro-2-p...)
Affinity DataKi:  7.30nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranes in presence of GTPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176822(isopropyl 4-(4-methoxyphenethylamino)-1-(2-chloro-...)
Affinity DataKi:  7.70nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranes in presence of GTPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176835(ethyl 4-(4-methoxyphenethylamino)-1-(2-chloro-2-ph...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176815(ethyl 4-(4-fluorophenethylamino)-1-(2-chloro-2-phe...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176838(1-(2-chloro-2-phenyl-ethyl)-4-(2-p-tolyl-ethylamin...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176842(ethyl 4-(2-fluorophenethylamino)-1-(2-chloro-2-phe...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50176815(ethyl 4-(4-fluorophenethylamino)-1-(2-chloro-2-phe...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50176822(isopropyl 4-(4-methoxyphenethylamino)-1-(2-chloro-...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176832(ethyl 4-(4-chlorophenethylamino)-1-(2-chloro-2-phe...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176855(1-(2-chloro-2-phenyl-ethyl)-4-(2-p-tolyl-ethylamin...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176844(isopropyl 1-(2-chloro-2-phenylethyl)-4-(propylamin...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50176835(ethyl 4-(4-methoxyphenethylamino)-1-(2-chloro-2-ph...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50176842(ethyl 4-(2-fluorophenethylamino)-1-(2-chloro-2-phe...)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176849(isopropyl 1-(2-chloro-2-phenylethyl)-4-(phenethyla...)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176828(ethyl 4-(3-fluorophenethylamino)-1-(2-chloro-2-phe...)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176840(isopropyl 1-(2-chloro-2-phenylethyl)-4-(cyclopropy...)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176825(isopropyl 4-(4-chlorophenethylamino)-1-(2-chloro-2...)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176839(isopropyl 4-(2-chlorophenethylamino)-1-(2-chloro-2...)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176848(1-(2-chloro-2-phenyl-ethyl)-4-(2-p-tolyl-ethylamin...)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176834(cyclopropylmethyl 1-(2-chloro-2-phenylethyl)-4-(ph...)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176850(sec-butyl 1-(2-chloro-2-phenylethyl)-4-(propylamin...)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176843(sec-butyl 1-(2-chloro-2-phenylethyl)-4-(phenethyla...)
Affinity DataKi:  62nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176852(1-(2-chloro-2-phenyl-ethyl)-4-(2-p-tolyl-ethylamin...)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176847(ethyl 4-(2-chlorophenethylamino)-1-(2-chloro-2-phe...)
Affinity DataKi:  76nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176830(methyl 1-(2-chloro-2-phenylethyl)-4-(phenethylamin...)
Affinity DataKi:  88nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50176833(methyl 4-(4-methoxyphenethylamino)-1-(2-chloro-2-p...)
Affinity DataKi:  94nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176845(isopropyl 4-(3-chlorophenethylamino)-1-(2-chloro-2...)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176820(4-butyl-5-(4-cyclopropylbut-1-en-2-yl)-1-(2-phenyl...)
Affinity DataKi:  109nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176826(propyl 1-(2-chloro-2-phenylethyl)-4-(phenethylamin...)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176819(methyl 4-(benzylamino)-1-(2-chloro-2-phenylethyl)-...)
Affinity DataKi:  141nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176818(propyl 1-(2-chloro-2-phenylethyl)-4-(propylamino)-...)
Affinity DataKi:  145nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50176838(1-(2-chloro-2-phenyl-ethyl)-4-(2-p-tolyl-ethylamin...)
Affinity DataKi:  148nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50176832(ethyl 4-(4-chlorophenethylamino)-1-(2-chloro-2-phe...)
Affinity DataKi:  153nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176831(propyl 1-(2-chloro-2-phenylethyl)-4-(cyclopropylam...)
Affinity DataKi:  156nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176836(methyl 1-(2-chloro-2-phenylethyl)-4-(propylamino)-...)
Affinity DataKi:  170nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176841(ethyl 4-(3-chlorophenethylamino)-1-(2-chloro-2-phe...)
Affinity DataKi:  178nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176853(sec-butyl 1-(2-chloro-2-phenylethyl)-4-(cyclopropy...)
Affinity DataKi:  197nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176816(methyl 1-(2-chloro-2-phenylethyl)-4-(cyclopropylam...)
Affinity DataKi:  251nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176851(isopropyl 4-(benzylamino)-1-(2-chloro-2-phenylethy...)
Affinity DataKi:  559nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176827(butyl 1-(2-chloro-2-phenylethyl)-4-(cyclopropylami...)
Affinity DataKi:  895nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176846(butyl 1-(2-chloro-2-phenylethyl)-4-(propylamino)-1...)
Affinity DataKi:  959nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176823(isopropyl 1-(2-chloro-2-phenylethyl)-4-(pyrrolidin...)
Affinity DataKi:  1.08E+3nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50176830(methyl 1-(2-chloro-2-phenylethyl)-4-(phenethylamin...)
Affinity DataKi:  1.23E+3nMAssay Description:Displacement of [3H]CGS-21680 from adenosine A2A receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50176826(propyl 1-(2-chloro-2-phenylethyl)-4-(phenethylamin...)
Affinity DataKi:  1.36E+3nMAssay Description:Displacement of [3H]CGS-21680 from adenosine A2A receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50176854(propyl 4-(benzylamino)-1-(2-chloro-2-phenylethyl)-...)
Affinity DataKi:  1.37E+3nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50176818(propyl 1-(2-chloro-2-phenylethyl)-4-(propylamino)-...)
Affinity DataKi:  1.39E+3nMAssay Description:Displacement of [3H]CGS-21680 from adenosine A2A receptor in bovine cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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