TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Inhibitory activity against Farnesyltransferase quantified by modified SPA assay with improved sensitivityMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Inhibitory activity against Ha-Ras processing in COS7 cellsMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against farnesyltransferase quantified by SPA assayMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 4.20nMAssay Description:Inhibitory activity against Ha-Ras processing in COS7 cellsMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 4.20nMAssay Description:Inhibitory activity against Ha-Ras processing in COS7 cellsMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 4.5nMAssay Description:Inhibitory activity against farnesyltransferase quantified by SPA assayMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 4.5nMAssay Description:Inhibitory activity against farnesyltransferase quantified by SPA assayMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Mus musculus)
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Anchorage-independent growth of transformed NIH3T3 cells in soft agarMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Mus musculus)
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 5.20nMAssay Description:Anchorage-independent growth of transformed NIH3T3 cells in soft agarMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 5.5nMAssay Description:Inhibitory activity against farnesyltransferase quantified by SPA assayMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 5.70nMAssay Description:Inhibitory activity against farnesyltransferase quantified by SPA assayMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibitory activity against farnesyltransferase quantified by SPA assayMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibitory activity against farnesyltransferase quantified by SPA assayMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 7.30nMAssay Description:Inhibitory activity against farnesyltransferase quantified by SPA assayMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 7.30nMAssay Description:Inhibitory activity against farnesyltransferase quantified by SPA assayMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 7.90nMAssay Description:Inhibitory activity against farnesyltransferase quantified by SPA assayMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibitory activity against farnesyltransferase quantified by SPA assayMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibitory activity against farnesyltransferase quantified by SPA assayMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibitory activity against farnesyltransferase quantified by SPA assayMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 8.40nMAssay Description:Inhibitory activity against farnesyltransferase quantified by SPA assayMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 8.60nMAssay Description:Inhibitory activity against Ha-Ras processing in COS7 cellsMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 9.10nMAssay Description:Inhibitory activity against farnesyltransferase quantified by SPA assayMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 9.10nMAssay Description:Inhibitory activity against farnesyltransferase quantified by SPA assayMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 9.70nMAssay Description:Inhibitory activity against Ha-Ras processing in COS7 cellsMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against farnesyltransferase quantified by SPA assayMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibitory activity against Ha-Ras processing in COS7 cellsMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibitory activity against farnesyltransferase quantified by SPA assayMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibitory activity against farnesyltransferase quantified by SPA assayMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibitory activity against farnesyltransferase quantified by SPA assayMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibitory activity against farnesyltransferase quantified by SPA assayMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibitory activity against Ha-Ras processing in COS7 cellsMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibitory activity against farnesyltransferase quantified by SPA assayMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibitory activity against farnesyltransferase quantified by SPA assayMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibitory activity against farnesyltransferase quantified by SPA assayMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibitory activity against farnesyltransferase quantified by SPA assayMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibitory activity against farnesyltransferase quantified by SPA assayMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibitory activity against farnesyltransferase quantified by SPA assayMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibitory activity against Ha-Ras processing in COS7 cellsMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibitory activity against farnesyltransferase quantified by SPA assayMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibitory activity against farnesyltransferase quantified by SPA assayMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against Ha-Ras processing in COS7 cellsMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against farnesyltransferase quantified by SPA assayMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against farnesyltransferase quantified by SPA assayMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibitory activity against farnesyltransferase quantified by SPA assayMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibitory activity against farnesyltransferase quantified by SPA assayMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Inhibitory activity against farnesyltransferase quantified by SPA assayMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibitory activity against Ha-Ras processing in COS7 cellsMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 38nMAssay Description:Inhibitory activity against Ha-Ras processing in COS7 cellsMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 45nMAssay Description:Inhibitory activity against farnesyltransferase quantified by SPA assayMore data for this Ligand-Target Pair
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Pharmacopeia
Curated by ChEMBL
Pharmacopeia
Curated by ChEMBL
Affinity DataIC50: 45nMAssay Description:Inhibitory activity against Ha-Ras processing in COS7 cellsMore data for this Ligand-Target Pair