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Found 26 Enz. Inhib. hit(s) with all data for entry = 50017181
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50031704((2S,4R)-2-Amino-4-methyl-pentanedioic acid | (2S,4...)
Affinity DataKi:  6.60E+3nMAssay Description:Binding affinity to human EAAT3 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50178688((2S,4R)-4-benzylglutamic acid | CHEMBL198618)
Affinity DataKi:  1.30E+4nMAssay Description:Binding affinity to human EAAT1 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50031704((2S,4R)-2-Amino-4-methyl-pentanedioic acid | (2S,4...)
Affinity DataKi:  1.30E+4nMAssay Description:Binding affinity to human EAAT2 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50088230((2S,4R)-4-propylglutamic acid | 2-Amino-4-propyl-p...)
Affinity DataKi:  1.30E+4nMAssay Description:Binding affinity to human EAAT1 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50178684((2S,4R)-4-ethylglutamic acid | CHEMBL372124)
Affinity DataKi:  1.40E+4nMAssay Description:Binding affinity to human EAAT2 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50178683((2S,4S)-4-isopropylglutamic acid | CHEMBL199564)
Affinity DataKi:  1.90E+4nMAssay Description:Binding affinity to human EAAT2 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50088230((2S,4R)-4-propylglutamic acid | 2-Amino-4-propyl-p...)
Affinity DataKi:  2.20E+4nMAssay Description:Binding affinity to human EAAT2 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50178687((2S,4R)-4-isobutylglutamic acid | CHEMBL199617)
Affinity DataKi:  2.20E+4nMAssay Description:Binding affinity to human EAAT2 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50178684((2S,4R)-4-ethylglutamic acid | CHEMBL372124)
Affinity DataKi:  2.30E+4nMAssay Description:Binding affinity to human EAAT1 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50178686((2S,4R)-4-isopentylglutamic acid | CHEMBL197176)
Affinity DataKi:  2.60E+4nMAssay Description:Binding affinity to human EAAT2 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50178686((2S,4R)-4-isopentylglutamic acid | CHEMBL197176)
Affinity DataKi:  2.90E+4nMAssay Description:Binding affinity to human EAAT1 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50088230((2S,4R)-4-propylglutamic acid | 2-Amino-4-propyl-p...)
Affinity DataKi:  3.20E+4nMAssay Description:Binding affinity to human EAAT3 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50178683((2S,4S)-4-isopropylglutamic acid | CHEMBL199564)
Affinity DataKi:  3.50E+4nMAssay Description:Binding affinity to human EAAT1 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50178688((2S,4R)-4-benzylglutamic acid | CHEMBL198618)
Affinity DataKi:  3.60E+4nMAssay Description:Binding affinity to human EAAT2 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50178684((2S,4R)-4-ethylglutamic acid | CHEMBL372124)
Affinity DataKi:  3.80E+4nMAssay Description:Binding affinity to human EAAT3 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50178685((2S,4R)-4-butylglutamic acid | CHEMBL381004)
Affinity DataKi:  4.20E+4nMAssay Description:Binding affinity to human EAAT2 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50178685((2S,4R)-4-butylglutamic acid | CHEMBL381004)
Affinity DataKi:  5.00E+4nMAssay Description:Binding affinity to human EAAT1 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50178683((2S,4S)-4-isopropylglutamic acid | CHEMBL199564)
Affinity DataKi:  5.10E+4nMAssay Description:Binding affinity to human EAAT3 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50178687((2S,4R)-4-isobutylglutamic acid | CHEMBL199617)
Affinity DataKi:  5.50E+4nMAssay Description:Binding affinity to human EAAT1 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50178688((2S,4R)-4-benzylglutamic acid | CHEMBL198618)
Affinity DataKi:  6.60E+4nMAssay Description:Binding affinity to human EAAT3 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50088220((2S,4R)-4-pentylglutamic acid | 2-Amino-4-pentyl-p...)
Affinity DataKi:  7.70E+4nMAssay Description:Binding affinity to human EAAT2 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50178685((2S,4R)-4-butylglutamic acid | CHEMBL381004)
Affinity DataKi:  8.00E+4nMAssay Description:Binding affinity to human EAAT3 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50178686((2S,4R)-4-isopentylglutamic acid | CHEMBL197176)
Affinity DataKi:  8.10E+4nMAssay Description:Binding affinity to human EAAT3 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50088220((2S,4R)-4-pentylglutamic acid | 2-Amino-4-pentyl-p...)
Affinity DataKi:  9.80E+4nMAssay Description:Binding affinity to human EAAT3 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50088220((2S,4R)-4-pentylglutamic acid | 2-Amino-4-pentyl-p...)
Affinity DataKi:  1.20E+5nMAssay Description:Binding affinity to human EAAT1 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50178687((2S,4R)-4-isobutylglutamic acid | CHEMBL199617)
Affinity DataKi:  3.00E+5nMAssay Description:Binding affinity to human EAAT3 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed