Compile Data Set for Download or QSAR
maximum 50k data
Found 53 Enz. Inhib. hit(s) with all data for entry = 50003765
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475698(CHEMBL206748)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]5-HT from the cloned human 5-HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475694(CHEMBL204269)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]5-HT from the cloned human 5-HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50357995(CHEMBL202780)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]5-HT from the cloned human 5-HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50297894(2-(3-(1-(phenylsulfonyl)cyclobutyl)propyl)-1,2,3,4...)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]5-HT from the cloned human 5-HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475691(CHEMBL206563)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]5-HT from the cloned human 5-HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475700(CHEMBL206305)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]5-HT from the cloned human 5-HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475692(CHEMBL379238)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]5-HT from the cloned human 5-HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475705(CHEMBL206747)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]5-HT from the cloned human 5-HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475693(CHEMBL203400)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]5-HT from the cloned human 5-HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475699(CHEMBL380613)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]5-HT from the cloned human 5-HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50297894(2-(3-(1-(phenylsulfonyl)cyclobutyl)propyl)-1,2,3,4...)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]5-HT from the cloned human 5-HT1A receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475703(CHEMBL382163)
Affinity DataKi:  53nMAssay Description:Displacement of [3H]5-HT from the cloned human 5-HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475695(CHEMBL380511)
Affinity DataKi:  54nMAssay Description:Displacement of [3H]5-HT from the cloned human 5-HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50297894(2-(3-(1-(phenylsulfonyl)cyclobutyl)propyl)-1,2,3,4...)
Affinity DataKi:  65nMAssay Description:Displacement of [3H]ketanserin from the cloned human 5-HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475696(CHEMBL206667)
Affinity DataKi:  96nMAssay Description:Displacement of [3H]5-HT from the cloned human 5-HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475698(CHEMBL206748)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]5-HT from the cloned human 5-HT1A receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475694(CHEMBL204269)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]spiperone from the cloned human D2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475694(CHEMBL204269)
Affinity DataKi:  400nMAssay Description:Displacement of [3H]5-HT from the cloned human 5-HT1A receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475701(CHEMBL204174)
Affinity DataKi:  455nMAssay Description:Displacement of [3H]5-HT from the cloned human 5-HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475694(CHEMBL204269)
Affinity DataKi:  540nMAssay Description:Displacement of [3H]prazosin from alpha-1 adrenergic receptor in rat cortexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475707(CHEMBL206269)
Affinity DataKi:  550nMAssay Description:Displacement of [3H]5-HT from the cloned human 5-HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475698(CHEMBL206748)
Affinity DataKi:  570nMAssay Description:Displacement of [3H]ketanserin from the cloned human 5-HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475693(CHEMBL203400)
Affinity DataKi:  710nMAssay Description:Displacement of [3H]spiperone from the cloned human D2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50357995(CHEMBL202780)
Affinity DataKi:  900nMAssay Description:Displacement of [3H]spiperone from the cloned human D2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475695(CHEMBL380511)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]spiperone from the cloned human D2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475692(CHEMBL379238)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]ketanserin from the cloned human 5-HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50357995(CHEMBL202780)
Affinity DataKi:  1.50E+3nMAssay Description:Displacement of [3H]5-HT from the cloned human 5-HT1A receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475692(CHEMBL379238)
Affinity DataKi:  1.50E+3nMAssay Description:Displacement of [3H]spiperone from the cloned human D2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475694(CHEMBL204269)
Affinity DataKi:  1.80E+3nMAssay Description:Displacement of [3H]ketanserin from the cloned human 5-HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475693(CHEMBL203400)
Affinity DataKi:  1.87E+3nMAssay Description:Displacement of [3H]ketanserin from the cloned human 5-HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50357995(CHEMBL202780)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [3H]ketanserin from the cloned human 5-HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475695(CHEMBL380511)
Affinity DataKi: >2.00E+3nMAssay Description:Displacement of [3H]ketanserin from the cloned human 5-HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475693(CHEMBL203400)
Affinity DataKi:  2.40E+3nMAssay Description:Displacement of [3H]5-HT from the cloned human 5-HT1A receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475702(CHEMBL380863)
Affinity DataKi:  2.70E+3nMAssay Description:Displacement of [3H]5-HT from the cloned human 5-HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50357995(CHEMBL202780)
Affinity DataKi:  3.90E+3nMAssay Description:Displacement of [3H]prazosin from alpha-1 adrenergic receptor in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475695(CHEMBL380511)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]prazosin from alpha-1 adrenergic receptor in rat cortexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50357995(CHEMBL202780)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [35S]-labeled MK-499 from cloned human ERG receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475692(CHEMBL379238)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]prazosin from alpha-1 adrenergic receptor in rat cortexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475693(CHEMBL203400)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]prazosin from alpha-1 adrenergic receptor in rat cortexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475693(CHEMBL203400)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [35S]-labeled MK-499 from cloned human ERG receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475695(CHEMBL380511)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [35S]-labeled MK-499 from cloned human ERG receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475694(CHEMBL204269)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [35S]-labeled MK-499 from cloned human ERG receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475692(CHEMBL379238)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [3H]5-HT from the cloned human 5-HT1B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475706(CHEMBL425767)
Affinity DataKi:  5.80E+3nMAssay Description:Displacement of [3H]5-HT from the cloned human 5-HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475693(CHEMBL203400)
Affinity DataKi: >7.00E+3nMAssay Description:Displacement of [3H]5-HT from the cloned human 5-HT1B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475697(CHEMBL380114)
Affinity DataKi: >7.00E+3nMAssay Description:Displacement of [3H]5-HT from the cloned human 5-HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50357995(CHEMBL202780)
Affinity DataKi: >7.00E+3nMAssay Description:Displacement of [3H]5-HT from the cloned human 5-HT1B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475695(CHEMBL380511)
Affinity DataKi: >7.00E+3nMAssay Description:Displacement of [3H]5-HT from the cloned human 5-HT1B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475704(CHEMBL383232)
Affinity DataKi: >7.00E+3nMAssay Description:Displacement of [3H]5-HT from the cloned human 5-HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50475695(CHEMBL380511)
Affinity DataKi: >7.00E+3nMAssay Description:Displacement of [3H]5-HT from the cloned human 5-HT1A receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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