Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 5517
TargetAlpha-1A adrenergic receptor(Human)
University of Dublin

Curated by PDSP Ki Database
LigandPNGBDBM81444(NSC_185453 | CAS_185453 | WB 4101 | WB-4101)
Affinity DataKi:  0.160nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Dublin

Curated by PDSP Ki Database
LigandPNGBDBM29568([3H]-Minipress | [3H]-Furazosin | PRAZOSIN HYDROCH...)
Affinity DataKi:  0.200nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Mouse)
University of Dublin

Curated by PDSP Ki Database
LigandPNGBDBM29568([3H]-Minipress | [3H]-Furazosin | PRAZOSIN HYDROCH...)
Affinity DataKi:  0.25nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Dublin

Curated by PDSP Ki Database
LigandPNGBDBM81444(NSC_185453 | CAS_185453 | WB 4101 | WB-4101)
Affinity DataKi:  0.25nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Dublin

Curated by PDSP Ki Database
LigandPNGBDBM29568([3H]-Minipress | [3H]-Furazosin | PRAZOSIN HYDROCH...)
Affinity DataKi:  0.320nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Dublin

Curated by PDSP Ki Database
LigandPNGBDBM50160165(CHEMBL88272 | RS-17053 | [2-(2-Cyclopropylmethoxy-...)
Affinity DataKi:  0.600nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Dublin

Curated by PDSP Ki Database
LigandPNGBDBM50033112(Urapidil-5-methyl | CHEMBL420060 | 6-{3-[4-(2-Meth...)
Affinity DataKi:  0.630nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Mouse)
University of Dublin

Curated by PDSP Ki Database
LigandPNGBDBM86731(UK 33,274 | CAS_74191-85-8 | Doxazosin)
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Dublin

Curated by PDSP Ki Database
LigandPNGBDBM50160152(CHEMBL24777 | 3-(3-{4-[4-Fluoro-2-(2,2,2-trifluoro...)
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Mouse)
University of Dublin

Curated by PDSP Ki Database
LigandPNGBDBM50033111(6,7-dimethoxy-2-[4-(tetrahydrofuran-2-ylcarbonyl)p...)
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Mouse)
University of Dublin

Curated by PDSP Ki Database
LigandPNGBDBM81444(NSC_185453 | CAS_185453 | WB 4101 | WB-4101)
Affinity DataKi:  2.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Dublin

Curated by PDSP Ki Database
LigandPNGBDBM50033111(6,7-dimethoxy-2-[4-(tetrahydrofuran-2-ylcarbonyl)p...)
Affinity DataKi:  2.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Dublin

Curated by PDSP Ki Database
LigandPNGBDBM86731(UK 33,274 | CAS_74191-85-8 | Doxazosin)
Affinity DataKi:  3.16nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Dublin

Curated by PDSP Ki Database
LigandPNGBDBM50033110(N-{3-[(4-amino-6,7-dimethoxyquinazolin-2-yl)(methy...)
Affinity DataKi:  3.16nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Dublin

Curated by PDSP Ki Database
LigandPNGBDBM86731(UK 33,274 | CAS_74191-85-8 | Doxazosin)
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Dublin

Curated by PDSP Ki Database
LigandPNGBDBM50033111(6,7-dimethoxy-2-[4-(tetrahydrofuran-2-ylcarbonyl)p...)
Affinity DataKi:  6.30nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Mouse)
University of Dublin

Curated by PDSP Ki Database
LigandPNGBDBM50033110(N-{3-[(4-amino-6,7-dimethoxyquinazolin-2-yl)(methy...)
Affinity DataKi:  10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Dublin

Curated by PDSP Ki Database
LigandPNGBDBM50033112(Urapidil-5-methyl | CHEMBL420060 | 6-{3-[4-(2-Meth...)
Affinity DataKi:  10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Mouse)
University of Dublin

Curated by PDSP Ki Database
LigandPNGBDBM50160165(CHEMBL88272 | RS-17053 | [2-(2-Cyclopropylmethoxy-...)
Affinity DataKi:  16nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Dublin

Curated by PDSP Ki Database
LigandPNGBDBM50160165(CHEMBL88272 | RS-17053 | [2-(2-Cyclopropylmethoxy-...)
Affinity DataKi:  16nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Mouse)
University of Dublin

Curated by PDSP Ki Database
LigandPNGBDBM50033112(Urapidil-5-methyl | CHEMBL420060 | 6-{3-[4-(2-Meth...)
Affinity DataKi:  40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Mouse)
University of Dublin

Curated by PDSP Ki Database
LigandPNGBDBM50160152(CHEMBL24777 | 3-(3-{4-[4-Fluoro-2-(2,2,2-trifluoro...)
Affinity DataKi:  79nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Dublin

Curated by PDSP Ki Database
LigandPNGBDBM50160152(CHEMBL24777 | 3-(3-{4-[4-Fluoro-2-(2,2,2-trifluoro...)
Affinity DataKi:  100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed