Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50017385
TargetCholecystokinin receptor type A(Rat)
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50181434((S)-2-{3-[3-(4-Benzoylphenyl)ureido]-2,4-dioxo-5-p...)
Affinity DataIC50: 61nMAssay Description:Displacement of [125I]D-Tyr-Gly-[(Nle28,31)CCK-26-33] from rat CCK receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50181434((S)-2-{3-[3-(4-Benzoylphenyl)ureido]-2,4-dioxo-5-p...)
Affinity DataEC50:  150nMAssay Description:Intrinsic agonistic activity at CCK receptor in SD rat at 1 uM expressed in pancreatic acinar cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50181435((R)-2-{3-[3-(4-Benzoylphenyl)ureido]-2,4-dioxo-5-p...)
Affinity DataIC50: 470nMAssay Description:Displacement of [125I]D-Tyr-Gly-[(Nle28,31)CCK-26-33] from rat CCK receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50181433((S)-2-{3-[3-(4-Benzoylphenyl)ureido]-2,4-dioxo-5-p...)
Affinity DataIC50: 490nMAssay Description:Displacement of [125I]D-Tyr-Gly-[(Nle28,31)CCK-26-33] from rat CCK receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50181436((R)-2-{3-[3-(4-Benzoylphenyl)ureido]-2,4-dioxo-5-p...)
Affinity DataIC50: 710nMAssay Description:Displacement of [125I]D-Tyr-Gly-[(Nle28,31)CCK-26-33] from rat CCK receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed