Compile Data Set for Download or QSAR
maximum 50k data
Found 52 Enz. Inhib. hit(s) with all data for entry = 50017430
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182065(CHEMBL205996 | N-{2-[2-(5-bromo-2-methoxy-phenyl)-...)
Affinity DataKi:  0.580nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182064(CHEMBL383117 | N-{2-[2-(5-bromo-2-methoxy-phenyl)-...)
Affinity DataKi:  0.830nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182072(CHEMBL205594 | N-{2-[2-(5-bromo-2-methoxy-phenyl)-...)
Affinity DataKi:  2.80nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182077(CHEMBL207946 | N-{2-[2-(5-bromo-2-methoxy-phenyl)-...)
Affinity DataKi:  3.20nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182073(CHEMBL205468 | N-{2-[2-(5-bromo-2-methoxy-phenyl)-...)
Affinity DataKi:  4.30nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182083(CHEMBL380854 | N-[4-(benzyl-methyl-amino)-butyl]-N...)
Affinity DataKi:  5.10nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182068(CHEMBL208376 | N-{2-[2-(5-bromo-2-methoxy-phenyl)-...)
Affinity DataKi:  11nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182067(CHEMBL439158 | N-{2-[2-(5-bromo-2-methoxy-phenyl)-...)
Affinity DataKi:  13nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182078(CHEMBL382833 | N-(4-diethylamino-1-methyl-butyl)-N...)
Affinity DataKi:  14nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182076(CHEMBL383120 | N-{2-[2-(5-bromo-2-methoxy-phenyl)-...)
Affinity DataKi:  21nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182062(CHEMBL205214 | N-{2-[2-(5-bromo-2-methoxy-phenyl)-...)
Affinity DataKi:  26nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182060(CHEMBL204670 | N-{2-[2-(5-bromo-2-methoxy-phenyl)-...)
Affinity DataKi:  57nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182080(CHEMBL206316 | N-{2-[2-(5-bromo-2-methoxy-phenyl)-...)
Affinity DataKi:  64nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182058(CHEMBL206141 | N-{2-[2-(5-bromo-2-methoxy-phenyl)-...)
Affinity DataKi:  80nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182070(CHEMBL205553 | N-(4-diethylamino-1-methyl-butyl)-N...)
Affinity DataKi:  89nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182074(CHEMBL206367 | N-{2-[2-(5-bromo-2-chloro-phenyl)-e...)
Affinity DataKi:  110nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182061(CHEMBL208268 | N-{2-[2-(5-bromo-2-methoxy-phenyl)-...)
Affinity DataKi:  190nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182063(CHEMBL379918 | N-(4-diethylamino-1-methyl-butyl)-N...)
Affinity DataKi:  690nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182069(CHEMBL413931 | N-{2-[2-(5-bromo-2-methoxy-phenyl)-...)
Affinity DataKi:  700nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182075(CHEMBL208366 | N-{2-[2-(5-bromo-2-methoxy-phenyl)-...)
Affinity DataKi:  770nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182085(2-(2-(5-bromo-2-methoxyphenethyl)-3-chlorophenyl)-...)
Affinity DataKi:  840nMAssay Description:Binding affinity to hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182081(CHEMBL205461 | N-[2-(5-bromo-2-methoxy-benzyloxy)-...)
Affinity DataKi:  900nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182066(CHEMBL205552 | N-{2-[2-(5-bromo-2-methoxy-phenyl)-...)
Affinity DataKi:  920nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182071(CHEMBL205898 | N-{2-[2-(5-bromo-2-methoxy-phenyl)-...)
Affinity DataKi:  2.50E+3nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182079(CHEMBL208367 | N-{2-[2-(5-bromo-2-methoxy-phenyl)-...)
Affinity DataKi:  2.60E+3nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182069(CHEMBL413931 | N-{2-[2-(5-bromo-2-methoxy-phenyl)-...)
Affinity DataKi:  3.15E+3nMAssay Description:Binding affinity to hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182082(CHEMBL208329 | N-{2-[2-(5-bromo-2-methoxy-phenyl)-...)
Affinity DataKi:  4.10E+3nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182084(CHEMBL381085 | N-{2-[2-(5-bromo-2-methoxy-phenyl)-...)
Affinity DataKi:  6.30E+3nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182059(CHEMBL205813 | N-{2-[2-(2-chloro-phenyl)-ethyl]-3-...)
Affinity DataKi:  2.60E+4nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182067(CHEMBL439158 | N-{2-[2-(5-bromo-2-methoxy-phenyl)-...)
Affinity DataIC50:  31nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182065(CHEMBL205996 | N-{2-[2-(5-bromo-2-methoxy-phenyl)-...)
Affinity DataIC50:  70nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182072(CHEMBL205594 | N-{2-[2-(5-bromo-2-methoxy-phenyl)-...)
Affinity DataIC50:  97nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182073(CHEMBL205468 | N-{2-[2-(5-bromo-2-methoxy-phenyl)-...)
Affinity DataIC50:  130nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182078(CHEMBL382833 | N-(4-diethylamino-1-methyl-butyl)-N...)
Affinity DataIC50:  170nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182083(CHEMBL380854 | N-[4-(benzyl-methyl-amino)-butyl]-N...)
Affinity DataIC50:  180nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182064(CHEMBL383117 | N-{2-[2-(5-bromo-2-methoxy-phenyl)-...)
Affinity DataIC50:  260nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182068(CHEMBL208376 | N-{2-[2-(5-bromo-2-methoxy-phenyl)-...)
Affinity DataIC50:  260nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182077(CHEMBL207946 | N-{2-[2-(5-bromo-2-methoxy-phenyl)-...)
Affinity DataIC50:  330nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182076(CHEMBL383120 | N-{2-[2-(5-bromo-2-methoxy-phenyl)-...)
Affinity DataIC50:  390nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182081(CHEMBL205461 | N-[2-(5-bromo-2-methoxy-benzyloxy)-...)
Affinity DataIC50:  530nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182062(CHEMBL205214 | N-{2-[2-(5-bromo-2-methoxy-phenyl)-...)
Affinity DataIC50:  650nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182074(CHEMBL206367 | N-{2-[2-(5-bromo-2-chloro-phenyl)-e...)
Affinity DataIC50:  660nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182080(CHEMBL206316 | N-{2-[2-(5-bromo-2-methoxy-phenyl)-...)
Affinity DataIC50:  670nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182060(CHEMBL204670 | N-{2-[2-(5-bromo-2-methoxy-phenyl)-...)
Affinity DataIC50:  1.20E+3nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182070(CHEMBL205553 | N-(4-diethylamino-1-methyl-butyl)-N...)
Affinity DataIC50:  1.50E+3nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182063(CHEMBL379918 | N-(4-diethylamino-1-methyl-butyl)-N...)
Affinity DataIC50:  1.80E+3nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182069(CHEMBL413931 | N-{2-[2-(5-bromo-2-methoxy-phenyl)-...)
Affinity DataIC50:  2.58E+3nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182061(CHEMBL208268 | N-{2-[2-(5-bromo-2-methoxy-phenyl)-...)
Affinity DataIC50:  4.50E+3nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182058(CHEMBL206141 | N-{2-[2-(5-bromo-2-methoxy-phenyl)-...)
Affinity DataIC50:  5.70E+3nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182075(CHEMBL208366 | N-{2-[2-(5-bromo-2-methoxy-phenyl)-...)
Affinity DataIC50:  8.50E+3nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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