Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50000537
TargetKappa-type opioid receptor(Mouse)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50006994(CHEMBL535347 | 2-(3,4-Dichloro-phenyl)-N-methyl-N-...)
Affinity DataIC50: 5.20nMAssay Description:Binding affinity against opioid receptor kappa using [3H]U-69,593 as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Mouse)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50000296(CHEMBL441765 | CHEMBL482811 | U-50488H | US1149237...)
Affinity DataIC50: 5.40nMAssay Description:Binding affinity against Opioid receptor kappa 1 using [3H]U-69593 as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Mouse)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50007000(CHEMBL294832 | 2-(3,4-Dichloro-phenyl)-N-methyl-N-...)
Affinity DataIC50: 7.30nMAssay Description:Binding affinity against opioid receptor kappa using [3H]U-69,593 as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Mouse)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50006999(CHEMBL293273 | 2-(3,4-Dichloro-phenyl)-N-(2-dimeth...)
Affinity DataIC50: 12nMAssay Description:Binding affinity against opioid receptor kappa using [3H]U-69,593 as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Mouse)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50007002(CHEMBL296184 | 3,4-Dichloro-N-(3-dimethylamino-1,2...)
Affinity DataKi:  21nMAssay Description:Binding affinity against opioid receptor mu using [3H]etorphine as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Mouse)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50006996(CHEMBL55421 | 3,4-Dichloro-N-methyl-N-(3-pyrrolidi...)
Affinity DataIC50: 29nMAssay Description:Binding affinity against opioid receptor kappa using [3H]U-69,593 as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Mouse)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50229403(CHEMBL2311130)
Affinity DataKi:  52nMAssay Description:Binding affinity against Opioid receptor mu 1 using [3H]etorphine as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Mouse)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50007002(CHEMBL296184 | 3,4-Dichloro-N-(3-dimethylamino-1,2...)
Affinity DataIC50: 56nMAssay Description:Binding affinity against opioid receptor kappa using [3H]U-69,593 as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Mouse)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50007001(CHEMBL294231 | 3,4-Dichloro-N-methyl-N-(3-pyrrolid...)
Affinity DataIC50: 85nMAssay Description:Binding affinity against opioid receptor kappa using [3H]U-69,593 as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Mouse)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50006998(CHEMBL55244 | 2-(3,4-Dichloro-phenyl)-N-methyl-N-(...)
Affinity DataIC50: 145nMAssay Description:Binding affinity against opioid receptor kappa using [3H]U-69,593 as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Mouse)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50006997(CHEMBL55705 | 3,4-Dichloro-N-methyl-N-(2-pyrrolidi...)
Affinity DataIC50: 368nMAssay Description:Binding affinity against opioid receptor kappa using [3H]U-69,593 as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Mouse)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50006996(CHEMBL55421 | 3,4-Dichloro-N-methyl-N-(3-pyrrolidi...)
Affinity DataKi:  374nMAssay Description:Binding affinity against opioid receptor mu using [3H]etorphine as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Mouse)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50007004(CHEMBL55809 | 3,4-Dichloro-N-(2-dimethylamino-1,2,...)
Affinity DataKi:  505nMAssay Description:Binding affinity against opioid receptor mu using [3H]etorphine as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Mouse)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50006999(CHEMBL293273 | 2-(3,4-Dichloro-phenyl)-N-(2-dimeth...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against opioid receptor mu using [3H]etorphine as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Mouse)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50006994(CHEMBL535347 | 2-(3,4-Dichloro-phenyl)-N-methyl-N-...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against opioid receptor mu using [3H]etorphine as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Mouse)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50000296(CHEMBL441765 | CHEMBL482811 | U-50488H | US1149237...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against opioid receptor mu using [3H]etorphine as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Mouse)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50006998(CHEMBL55244 | 2-(3,4-Dichloro-phenyl)-N-methyl-N-(...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against opioid receptor mu using [3H]etorphine as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Mouse)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50006997(CHEMBL55705 | 3,4-Dichloro-N-methyl-N-(2-pyrrolidi...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against opioid receptor mu using [3H]etorphine as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Mouse)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50007001(CHEMBL294231 | 3,4-Dichloro-N-methyl-N-(3-pyrrolid...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against opioid receptor mu using [3H]etorphine as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Mouse)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50007000(CHEMBL294832 | 2-(3,4-Dichloro-phenyl)-N-methyl-N-...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against opioid receptor mu using [3H]etorphine as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Mouse)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50007004(CHEMBL55809 | 3,4-Dichloro-N-(2-dimethylamino-1,2,...)
Affinity DataIC50: 2.20E+3nMAssay Description:Binding affinity against opioid receptor kappa using [3H]U-69,593 as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed