Compile Data Set for Download or QSAR
maximum 50k data
Found 23 Enz. Inhib. hit(s) with all data for entry = 50017510
TargetCytochrome P450 2J2(Homo sapiens (Human))
Universite Paris 5 René

Curated by ChEMBL
LigandPNGBDBM50183079(4-(4-(hydroxydiphenylmethyl)piperidin-1-yl)-1-(4-p...)
Affinity DataKi:  160nMAssay Description:Inhibition of human recombinant CYP2J2 expressed in baculovirus-infected Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2J2(Homo sapiens (Human))
Universite Paris 5 René

Curated by ChEMBL
LigandPNGBDBM50183075(1-(4-allylphenyl)-4-(4-(hydroxydiphenylmethyl)pipe...)
Affinity DataIC50:  400nMAssay Description:Inhibition of human recombinant CYP2J2 expressed in baculovirus-infected Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2J2(Homo sapiens (Human))
Universite Paris 5 René

Curated by ChEMBL
LigandPNGBDBM50183079(4-(4-(hydroxydiphenylmethyl)piperidin-1-yl)-1-(4-p...)
Affinity DataIC50:  400nMAssay Description:Inhibition of human recombinant CYP2J2 expressed in baculovirus-infected Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2J2(Homo sapiens (Human))
Universite Paris 5 René

Curated by ChEMBL
LigandPNGBDBM50183085(1-(4-ethylphenyl)-4-(4-(hydroxydiphenylmethyl)pipe...)
Affinity DataIC50:  600nMAssay Description:Inhibition of human recombinant CYP2J2 expressed in baculovirus-infected Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2J2(Homo sapiens (Human))
Universite Paris 5 René

Curated by ChEMBL
LigandPNGBDBM50183080(1-(4-butylphenyl)-4-(4-(hydroxydiphenylmethyl)pipe...)
Affinity DataIC50:  700nMAssay Description:Inhibition of human recombinant CYP2J2 expressed in baculovirus-infected Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2J2(Homo sapiens (Human))
Universite Paris 5 René

Curated by ChEMBL
LigandPNGBDBM50183082(4-(4-(hydroxydiphenylmethyl)piperidin-1-yl)-1-p-to...)
Affinity DataIC50:  700nMAssay Description:Inhibition of human recombinant CYP2J2 expressed in baculovirus-infected Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2J2(Homo sapiens (Human))
Universite Paris 5 René

Curated by ChEMBL
LigandPNGBDBM50183084(CHEMBL205154 | terfenadone)
Affinity DataIC50:  700nMAssay Description:Inhibition of human recombinant CYP2J2 expressed in baculovirus-infected Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2J2(Homo sapiens (Human))
Universite Paris 5 René

Curated by ChEMBL
LigandPNGBDBM50183077(4-(4-(hydroxydiphenylmethyl)piperidin-1-yl)-1-(4-(...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of human recombinant CYP2J2 expressed in baculovirus-infected Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2J2(Homo sapiens (Human))
Universite Paris 5 René

Curated by ChEMBL
LigandPNGBDBM50183078(4-(4-(hydroxydiphenylmethyl)piperidin-1-yl)-1-(4-(...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of human recombinant CYP2J2 expressed in baculovirus-infected Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2J2(Homo sapiens (Human))
Universite Paris 5 René

Curated by ChEMBL
LigandPNGBDBM50183076(1-(4-(2,2-difluoroethyl)phenyl)-4-(4-(hydroxydiphe...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of human recombinant CYP2J2 expressed in baculovirus-infected Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2J2(Homo sapiens (Human))
Universite Paris 5 René

Curated by ChEMBL
LigandPNGBDBM50183086(3-(4-(4-(4-(hydroxydiphenylmethyl)piperidin-1-yl)b...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of human recombinant CYP2J2 expressed in baculovirus-infected Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2J2(Homo sapiens (Human))
Universite Paris 5 René

Curated by ChEMBL
LigandPNGBDBM50183081(1-(4-bromophenyl)-4-(4-(hydroxydiphenylmethyl)pipe...)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of human recombinant CYP2J2 expressed in baculovirus-infected Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Universite Paris 5 René

Curated by ChEMBL
LigandPNGBDBM50183075(1-(4-allylphenyl)-4-(4-(hydroxydiphenylmethyl)pipe...)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibition of human recombinant CYP3A4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2J2(Homo sapiens (Human))
Universite Paris 5 René

Curated by ChEMBL
LigandPNGBDBM50183087(1-(benzo[d][1,3]dioxol-5-yl)-4-(4-(hydroxydiphenyl...)
Affinity DataIC50:  6.70E+3nMAssay Description:Inhibition of human recombinant CYP2J2 expressed in baculovirus-infected Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2J2(Homo sapiens (Human))
Universite Paris 5 René

Curated by ChEMBL
LigandPNGBDBM50183083(4-(4-(hydroxydiphenylmethyl)piperidin-1-yl)-1-(4-m...)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of human recombinant CYP2J2 expressed in baculovirus-infected Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Universite Paris 5 René

Curated by ChEMBL
LigandPNGBDBM50183079(4-(4-(hydroxydiphenylmethyl)piperidin-1-yl)-1-(4-p...)
Affinity DataIC50:  7.90E+3nMAssay Description:Inhibition of human recombinant CYP3A4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2J2(Homo sapiens (Human))
Universite Paris 5 René

Curated by ChEMBL
LigandPNGBDBM50017376((+/-)1-(4-tert-butylphenyl)-4-(4-(hydroxydiphenylm...)
Affinity DataIC50:  8.10E+3nMAssay Description:Inhibition of human recombinant CYP2J2 expressed in baculovirus-infected Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Universite Paris 5 René

Curated by ChEMBL
LigandPNGBDBM50183075(1-(4-allylphenyl)-4-(4-(hydroxydiphenylmethyl)pipe...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of human recombinant CYP2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2B6(Homo sapiens (Human))
Universite Paris 5 René

Curated by ChEMBL
LigandPNGBDBM50183075(1-(4-allylphenyl)-4-(4-(hydroxydiphenylmethyl)pipe...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of human recombinant CYP2B6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Universite Paris 5 René

Curated by ChEMBL
LigandPNGBDBM50183079(4-(4-(hydroxydiphenylmethyl)piperidin-1-yl)-1-(4-p...)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of human recombinant CYP2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2B6(Homo sapiens (Human))
Universite Paris 5 René

Curated by ChEMBL
LigandPNGBDBM50183079(4-(4-(hydroxydiphenylmethyl)piperidin-1-yl)-1-(4-p...)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of human recombinant CYP2B6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C8(Homo sapiens (Human))
Universite Paris 5 René

Curated by ChEMBL
LigandPNGBDBM50183079(4-(4-(hydroxydiphenylmethyl)piperidin-1-yl)-1-(4-p...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant CYP2C8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C8(Homo sapiens (Human))
Universite Paris 5 René

Curated by ChEMBL
LigandPNGBDBM50183075(1-(4-allylphenyl)-4-(4-(hydroxydiphenylmethyl)pipe...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant CYP2C8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed