Compile Data Set for Download or QSAR
Report error Found 77 Enz. Inhib. hit(s) with all data for entry = 50017572
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184049BDBM50184049(3-(6-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2...)
Affinity DataIC50: 4nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50183986BDBM50183986(N-(2-aminoethyl)-3-(2-(3,4,5-trimethoxyphenylamino...)
Affinity DataIC50: 29nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50183989BDBM50183989(3-(3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2...)
Affinity DataIC50: 35nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184028BDBM50184028(2-(3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2...)
Affinity DataIC50: 37nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184019BDBM50184019(N-(2-(dimethylamino)ethyl)-3-(2-(3,4,5-trimethoxyp...)
Affinity DataIC50: 38nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184034BDBM50184034(3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-...)
Affinity DataIC50: 38nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184002BDBM50184002(N-(3-(dimethylamino)propyl)-3-(2-(3,4,5-trimethoxy...)
Affinity DataIC50: 54nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184000BDBM50184000(2-(3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2...)
Affinity DataIC50: 63nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184035BDBM50184035(N-isobutyl-3-(3-(2-(3,4,5-trimethoxyphenylamino)-7...)
Affinity DataIC50: 63nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50183979BDBM50183979(N-(2-(pyrrolidin-1-yl)ethyl)-3-(2-(3,4,5-trimethox...)
Affinity DataIC50: 73nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184020BDBM50184020(3-(3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2...)
Affinity DataIC50: 93nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184043BDBM50184043(7-(3-(2H-tetrazol-5-yl)phenyl)-N-(3,4,5-trimethoxy...)
Affinity DataIC50: 115nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184005BDBM50184005(N-cyclopropyl-2-(3-(2-(3,4,5-trimethoxyphenylamino...)
Affinity DataIC50: 117nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50183980BDBM50183980(7-(3-(2-(2H-tetrazol-5-yl)ethyl)phenyl)-N-(3,4,5-t...)
Affinity DataIC50: 119nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184003BDBM50184003(3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-...)
Affinity DataIC50: 126nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184036BDBM50184036(N-(2-aminoethyl)-6-(2-(3,4,5-trimethoxyphenylamino...)
Affinity DataIC50: 182nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50182010BDBM50182010(7-(pyridin-2-yl)-N-(2,4,6-trimethoxyphenyl)-7H-pyr...)
Affinity DataIC50: 212nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184037BDBM50184037(7-m-tolyl-N-(3,4,5-trimethoxyphenyl)-7H-pyrrolo[2,...)
Affinity DataIC50: 221nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184047BDBM50184047(7-(3-((2H-tetrazol-5-yl)methyl)phenyl)-N-(3,4,5-tr...)
Affinity DataIC50: 232nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184041BDBM50184041(7-(3-(trifluoromethyl)phenyl)-N-(3,4,5-trimethoxyp...)
Affinity DataIC50: 235nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184018BDBM50184018(N-(2-(dimethylamino)ethyl)-3-(3-(2-(3,4,5-trimetho...)
Affinity DataIC50: 236nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50183995BDBM50183995(N-(2-cyanoethyl)-6-(2-(3,4,5-trimethoxyphenylamino...)
Affinity DataIC50: 242nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50183984BDBM50183984(N-methyl-3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyr...)
Affinity DataIC50: 262nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184050BDBM50184050(N-(cyanomethyl)-6-(2-(3,4,5-trimethoxyphenylamino)...)
Affinity DataIC50: 278nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50183981BDBM50183981(N-(2-acetamidoethyl)-3-(2-(3,4,5-trimethoxyphenyla...)
Affinity DataIC50: 298nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50183983BDBM50183983(methyl 2-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrro...)
Affinity DataIC50: 314nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184025BDBM50184025(N-cyclopropyl-3-(2-(3,4,5-trimethoxyphenylamino)-7...)
Affinity DataIC50: 322nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184039BDBM50184039(N-methyl-3-(3-(2-(3,4,5-trimethoxyphenylamino)-7H-...)
Affinity DataIC50: 331nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50183987BDBM50183987(methyl 2-(3-(3-(2-(3,4,5-trimethoxyphenylamino)-7H...)
Affinity DataIC50: 339nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184021BDBM50184021(N-methyl-2-(2-(3,4,5-trimethoxyphenylamino)-7H-pyr...)
Affinity DataIC50: 342nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184013BDBM50184013(N-ethyl-3-(3-(2-(3,4,5-trimethoxyphenylamino)-7H-p...)
Affinity DataIC50: 345nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50183991BDBM50183991(N-ethyl-3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrr...)
Affinity DataIC50: 365nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184023BDBM50184023(N-(3-aminopropyl)-6-(2-(3,4,5-trimethoxyphenylamin...)
Affinity DataIC50: 397nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50183998BDBM50183998(N-ethyl-2-(3-(2-(3,4,5-trimethoxyphenylamino)-7H-p...)
Affinity DataIC50: 421nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184033BDBM50184033(N-(2-hydroxyethyl)-3-(2-(3,4,5-trimethoxyphenylami...)
Affinity DataIC50: 434nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184027BDBM50184027(2-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-...)
Affinity DataIC50: 504nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50183977BDBM50183977(7-p-tolyl-N-(3,4,5-trimethoxyphenyl)-7H-pyrrolo[2,...)
Affinity DataIC50: 507nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184038BDBM50184038(methyl 2-(2-(2-(3,4,5-trimethoxyphenylamino)-7H-py...)
Affinity DataIC50: 544nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184046BDBM50184046(N-(2-(dimethylamino)ethyl)-6-(2-(3,4,5-trimethoxyp...)
Affinity DataIC50: 634nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50183976BDBM50183976(methyl 2-(2-(3-(2-(3,4,5-trimethoxyphenylamino)-7H...)
Affinity DataIC50: 635nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184016BDBM50184016((2-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3...)
Affinity DataIC50: 727nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50183978BDBM50183978(N-(2-aminoethyl)-2-(3-(2-(3,4,5-trimethoxyphenylam...)
Affinity DataIC50: 727nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184006BDBM50184006(7-(4-(methylthio)phenyl)-N-(3,4,5-trimethoxyphenyl...)
Affinity DataIC50: 831nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184029BDBM50184029(N-(3-hydroxypropyl)-3-(2-(3,4,5-trimethoxyphenylam...)
Affinity DataIC50: 882nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184042BDBM50184042(N-(4-(dimethylamino)butyl)-3-(2-(3,4,5-trimethoxyp...)
Affinity DataIC50: 983nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184031BDBM50184031(N-(3-aminopropyl)-2-(3-(2-(3,4,5-trimethoxyphenyla...)
Affinity DataIC50: 1.33E+3nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184012BDBM50184012(methyl 3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrro...)
Affinity DataIC50: 1.51E+3nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184030BDBM50184030(7-(4-(trifluoromethyl)phenyl)-N-(3,4,5-trimethoxyp...)
Affinity DataIC50: 1.51E+3nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50183994BDBM50183994(7-(4-ethylphenyl)-N-(3,4,5-trimethoxyphenyl)-7H-py...)
Affinity DataIC50: 1.53E+3nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Genomics Institute of The Novartis Research Foundation

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50183985BDBM50183985(N-methyl-2-(3-(2-(3,4,5-trimethoxyphenylamino)-7H-...)
Affinity DataIC50: 1.81E+3nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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