Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50017612
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184576BDBM50184576(2-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-4-p...)
Affinity DataKi:  38.5nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A serotonergic receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184568BDBM50184568(2-(4-(4-(2-ethoxyphenyl)piperazin-1-yl)butyl)-4-p-...)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A serotonergic receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184571BDBM50184571(4-p-tolyl-2-(4-(4-(3-(trifluoromethyl)phenyl)piper...)
Affinity DataKi:  71.8nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A serotonergic receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184578BDBM50184578(2-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)butyl)-...)
Affinity DataKi:  81nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A serotonergic receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184579BDBM50184579(2-(7-(4-(2-methoxyphenyl)piperazin-1-yl)heptyl)-4-...)
Affinity DataKi:  101nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A serotonergic receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184569BDBM50184569(2-(4-(4-(3-chlorophenyl)piperazin-1-yl)butyl)-4-p-...)
Affinity DataKi:  116nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A serotonergic receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184583BDBM50184583(2-(7-(4-(2-ethoxyphenyl)piperazin-1-yl)heptyl)-4-p...)
Affinity DataKi:  207nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A serotonergic receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184574BDBM50184574(2-(4-(4-phenylpiperazin-1-yl)butyl)-4-p-tolylphtha...)
Affinity DataKi:  450nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A serotonergic receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184581BDBM50184581(2-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-4-p...)
Affinity DataKi:  473nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A serotonergic receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184570BDBM50184570(2-(7-(4-(3-chlorophenyl)piperazin-1-yl)heptyl)-4-p...)
Affinity DataKi:  673nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A serotonergic receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184575BDBM50184575(4-p-tolyl-2-(7-(4-(3-(trifluoromethyl)phenyl)piper...)
Affinity DataKi:  722nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A serotonergic receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184573BDBM50184573(2-(2-(4-(2-ethoxyphenyl)piperazin-1-yl)ethyl)-4-p-...)
Affinity DataKi:  951nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A serotonergic receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184580BDBM50184580(2-(4-(4-(pyrimidin-2-yl)piperazin-1-yl)butyl)-4-p-...)
Affinity DataKi:  1.18E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A serotonergic receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184572BDBM50184572(2-(2-(4-(2-isopropoxyphenyl)piperazin-1-yl)ethyl)-...)
Affinity DataKi:  1.29E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A serotonergic receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184577BDBM50184577(2-(4-(4-((2,3-dihydrobenzo[b][1,4]dioxin-2-yl)meth...)
Affinity DataKi:  1.93E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A serotonergic receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184582BDBM50184582(2-(2-(4-phenylpiperazin-1-yl)ethyl)-4-p-tolylphtha...)
Affinity DataKi:  6.20E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A serotonergic receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed