Compile Data Set for Download or QSAR
maximum 50k data
Found 104 Enz. Inhib. hit(s) with all data for entry = 50003771
TargetNeuronal acetylcholine receptor subunit alpha-2/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  0.0200nMAssay Description:Displacement of [3H]epibatidine from rat alpha-2-beta-2 nACHR expressed in human HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  0.0400nMAssay Description:Displacement of [3H]epibatidine from rat alpha-3-beta-2 nACHR expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  0.0600nMAssay Description:Displacement of [3H]epibatidine from rat alpha-4-beta-2 nACHR expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  0.0600nMAssay Description:Displacement of [3H]epibatidine from rat forebrain alpha4beta2 nACHRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-2/beta-4(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  0.0900nMAssay Description:Displacement of [3H]epibatidine from rat alpha-2-beta-4 nACHR expressed in human HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-4(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]epibatidine from rat alpha-4-beta-4 nACHR expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  0.570nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta4 nACHR expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-2/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50475816(CHEMBL205644)
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]epibatidine from rat alpha-2-beta-2 nACHR expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50475816(CHEMBL205644)
Affinity DataKi:  0.730nMAssay Description:Displacement of [3H]epibatidine from rat alpha-4-beta-2 nACHR expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-2/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50143282((-)-cytisine | (1R,5S)-1,2,3,4,5,6-Hexahydro-1,5-m...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]epibatidine from rat alpha-2-beta-2 nACHR expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50143282((-)-cytisine | (1R,5S)-1,2,3,4,5,6-Hexahydro-1,5-m...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]epibatidine from rat alpha-4-beta-2 nACHR expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50475815(CHEMBL379303)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]epibatidine from rat alpha-4-beta-2 nACHR expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50143282((-)-cytisine | (1R,5S)-1,2,3,4,5,6-Hexahydro-1,5-m...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]epibatidine from rat forebrain alpha4beta2 nACHRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-4(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50143282((-)-cytisine | (1R,5S)-1,2,3,4,5,6-Hexahydro-1,5-m...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]epibatidine from rat alpha-4-beta-4 nACHR expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-4(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50475816(CHEMBL205644)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]epibatidine from rat alpha-4-beta-4 nACHR expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50475816(CHEMBL205644)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]epibatidine from rat forebrain alpha4beta2 nACHRMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-2/beta-4(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50143282((-)-cytisine | (1R,5S)-1,2,3,4,5,6-Hexahydro-1,5-m...)
Affinity DataKi:  5.40nMAssay Description:Displacement of [3H]epibatidine from rat alpha-2-beta-4 nACHR expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-2/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50475815(CHEMBL379303)
Affinity DataKi:  7.5nMAssay Description:Displacement of [3H]epibatidine from rat alpha-2-beta-2 nACHR expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-2/beta-4(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50475816(CHEMBL205644)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]epibatidine from rat alpha-2-beta-4 nACHR expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50475814(CHEMBL208438)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]epibatidine from rat alpha-4-beta-2 nACHR expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50475815(CHEMBL379303)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]epibatidine from rat forebrain alpha4beta2 nACHRMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50475816(CHEMBL205644)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]epibatidine from rat alpha-3-beta-2 nACHR expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-2/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50475814(CHEMBL208438)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]epibatidine from rat alpha-2-beta-2 nACHR expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50143282((-)-cytisine | (1R,5S)-1,2,3,4,5,6-Hexahydro-1,5-m...)
Affinity DataKi:  37nMAssay Description:Displacement of [3H]epibatidine from rat alpha-3-beta-2 nACHR expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50475814(CHEMBL208438)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]epibatidine from rat forebrain alpha4beta2 nACHRMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-4(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50475815(CHEMBL379303)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]epibatidine from rat alpha-4-beta-4 nACHR expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-4(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50475814(CHEMBL208438)
Affinity DataKi:  68nMAssay Description:Displacement of [3H]epibatidine from rat alpha-4-beta-4 nACHR expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50475816(CHEMBL205644)
Affinity DataKi:  95nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta4 nACHR expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-2/beta-4(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50475815(CHEMBL379303)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]epibatidine from rat alpha-2-beta-4 nACHR expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50143282((-)-cytisine | (1R,5S)-1,2,3,4,5,6-Hexahydro-1,5-m...)
Affinity DataKi:  217nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta4 nACHR expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-2/beta-4(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50475814(CHEMBL208438)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]epibatidine from rat alpha-2-beta-4 nACHR expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50475822(CHEMBL208066)
Affinity DataKi:  390nMAssay Description:Displacement of [3H]epibatidine from rat alpha-4-beta-2 nACHR expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50475811(CHEMBL382845)
Affinity DataKi:  420nMAssay Description:Displacement of [3H]epibatidine from rat alpha-4-beta-2 nACHR expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50475814(CHEMBL208438)
Affinity DataKi:  467nMAssay Description:Displacement of [3H]epibatidine from rat alpha-3-beta-2 nACHR expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-2/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50475822(CHEMBL208066)
Affinity DataKi:  500nMAssay Description:Displacement of [3H]epibatidine from rat alpha-2-beta-2 nACHR expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50475810(CHEMBL204995)
Affinity DataKi:  540nMAssay Description:Displacement of [3H]epibatidine from rat alpha-4-beta-2 nACHR expressed in human HEK293 cells at 10 uMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50475815(CHEMBL379303)
Affinity DataKi:  540nMAssay Description:Displacement of [3H]epibatidine from rat alpha-3-beta-2 nACHR expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-4(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50475822(CHEMBL208066)
Affinity DataKi:  590nMAssay Description:Displacement of [3H]epibatidine from rat alpha-4-beta-4 nACHR expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-2/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50475811(CHEMBL382845)
Affinity DataKi:  820nMAssay Description:Displacement of [3H]epibatidine from rat alpha-2-beta-2 nACHR expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50475820(CHEMBL380841)
Affinity DataKi:  980nMAssay Description:Displacement of [3H]epibatidine from rat alpha-4-beta-2 nACHR expressed in human HEK293 cells at 10 uMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50475822(CHEMBL208066)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [3H]epibatidine from rat forebrain alpha4beta2 nACHRMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50475813(CHEMBL205230)
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of [3H]epibatidine from rat alpha-4-beta-2 nACHR expressed in human HEK293 cells at 10 uMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-4(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50475810(CHEMBL204995)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [3H]epibatidine from rat alpha-4-beta-4 nACHR expressed in human HEK293 cells at 10 uMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50475818(CHEMBL206887)
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of [3H]epibatidine from rat alpha-4-beta-2 nACHR expressed in human HEK293 cells at 10 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-2/beta-4(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50475822(CHEMBL208066)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [3H]epibatidine from rat alpha-2-beta-4 nACHR expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50475817(CHEMBL205267)
Affinity DataKi:  1.78E+3nMAssay Description:Displacement of [3H]epibatidine from rat alpha-4-beta-2 nACHR expressed in human HEK293 cells at 10 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-4(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50475820(CHEMBL380841)
Affinity DataKi:  2.60E+3nMAssay Description:Displacement of [3H]epibatidine from rat alpha-4-beta-4 nACHR expressed in human HEK293 cells at 10 uMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50475811(CHEMBL382845)
Affinity DataKi:  3.10E+3nMAssay Description:Displacement of [3H]epibatidine from rat forebrain alpha4beta2 nACHRMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-4(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50475811(CHEMBL382845)
Affinity DataKi:  3.30E+3nMAssay Description:Displacement of [3H]epibatidine from rat alpha-4-beta-4 nACHR expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-2/beta-2(Rattus norvegicus (Rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50475818(CHEMBL206887)
Affinity DataKi:  3.60E+3nMAssay Description:Displacement of [3H]epibatidine from rat alpha2beta2 nACHR expressed in human HEK293 cells at 10 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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