Compile Data Set for Download or QSAR
maximum 50k data
Found 36 Enz. Inhib. hit(s) with all data for entry = 50017812
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50186938(1-(3-tert-butyl-2-methyl-5-oxo-1-phenyl-2,5-dihydr...)
Affinity DataEC50:  83nMAssay Description:Activity at human FPRL1-mediated calcium mobilization in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM21692(1-(4-chlorophenyl)-3-[1-methyl-3-oxo-2-phenyl-5-(p...)
Affinity DataEC50:  44nMAssay Description:Activity at human FPRL1-mediated calcium mobilization in CHO cellsMore data for this Ligand-Target Pair
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50186940(1-(2,3-dimethyl-5-oxo-1-phenyl-2,5-dihydro-1H-pyra...)
Affinity DataEC50:  1.23E+4nMAssay Description:Activity at human FPRL1-mediated calcium mobilization in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50186942(1-(3-fluoro-4-methylphenyl)-3-(3-isopropyl-2-methy...)
Affinity DataEC50:  81nMAssay Description:Activity at human FPRL1-mediated calcium mobilization in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50186941(1-(4-cyanophenyl)-3-(2,3-dimethyl-5-oxo-1-phenyl-2...)
Affinity DataEC50:  3.70E+3nMAssay Description:Activity at human FPRL1-mediated calcium mobilization in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50186943(1-(4-bromophenyl)-3-(2,3-dimethyl-5-oxo-1-phenyl-2...)
Affinity DataEC50:  90nMAssay Description:Activity at human FPRL1-mediated calcium mobilization in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50186944(1-(1-(4,5-dihydrothiazol-2-yl)-3-isopropyl-2-methy...)
Affinity DataEC50:  5.13E+3nMAssay Description:Activity at human FPRL1-mediated calcium mobilization in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM21693(1-(2-chlorophenyl)-3-[1-methyl-3-oxo-2-phenyl-5-(p...)
Affinity DataEC50: >1.00E+4nMAssay Description:Activity at human FPRL1-mediated calcium mobilization in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50186945(1-(3-ethyl-2-methyl-5-oxo-1-phenyl-2,5-dihydro-1H-...)
Affinity DataEC50:  310nMAssay Description:Activity at human FPRL1-mediated calcium mobilization in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50186950(1-(2,3-dimethyl-5-oxo-1-phenyl-2,5-dihydro-1H-pyra...)
Affinity DataEC50:  4.85E+3nMAssay Description:Activity at human FPRL1-mediated calcium mobilization in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50186947(1-(2,3-dimethyl-5-oxo-1-phenyl-2,5-dihydro-1H-pyra...)
Affinity DataEC50:  770nMAssay Description:Activity at human FPRL1-mediated calcium mobilization in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50186949(1-(2,3-dimethyl-5-oxo-1-phenyl-2,5-dihydro-1H-pyra...)
Affinity DataEC50:  1.26E+3nMAssay Description:Activity at human FPRL1-mediated calcium mobilization in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50186948(1-(2,3-dimethyl-5-oxo-1-phenyl-2,5-dihydro-1H-pyra...)
Affinity DataEC50:  2.73E+3nMAssay Description:Activity at human FPRL1-mediated calcium mobilization in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50186951(1-(3-chlorophenyl)-3-(2,3-dimethyl-5-oxo-1-phenyl-...)
Affinity DataEC50: >1.00E+4nMAssay Description:Activity at human FPRL1-mediated calcium mobilization in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50186953(1-(3-isopropyl-2-methyl-5-oxo-1-(quinolin-3-yl)-2,...)
Affinity DataEC50:  44nMAssay Description:Activity at human FPRL1-mediated calcium mobilization in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50186954(1-(4-chlorophenyl)-3-(3-ethyl-2-methyl-5-oxo-1-phe...)
Affinity DataEC50:  140nMAssay Description:Activity at human FPRL1-mediated calcium mobilization in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50186956(1-(3-isopropyl-2-methyl-5-oxo-1-(pyrimidin-5-yl)-2...)
Affinity DataEC50:  150nMAssay Description:Activity at human FPRL1-mediated calcium mobilization in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50186957(1-(3-tert-butyl-2-methyl-5-oxo-1-phenyl-2,5-dihydr...)
Affinity DataEC50:  23nMAssay Description:Activity at human FPRL1-mediated calcium mobilization in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50186959(1-(2-chlorophenyl)-3-(2,3-dimethyl-5-oxo-1-phenyl-...)
Affinity DataEC50: >1.00E+4nMAssay Description:Activity at human FPRL1-mediated calcium mobilization in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50186958(1-(2-ethyl-3-isopropyl-5-oxo-1-phenyl-2,5-dihydro-...)
Affinity DataEC50:  100nMAssay Description:Activity at human FPRL1-mediated calcium mobilization in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50186955(1-(2,3-dimethyl-5-oxo-1-phenyl-2,5-dihydro-1H-pyra...)
Affinity DataEC50:  170nMAssay Description:Activity at human FPRL1-mediated calcium mobilization in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50186946(1-(1,5-dimethyl-3-oxo-2-phenylpyrazolidin-4-yl)-3-...)
Affinity DataEC50: >1.00E+4nMAssay Description:Activity at human FPRL1-mediated calcium mobilization in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM31710(1-(4-chlorophenyl)-3-(1,5-dimethyl-3-oxidanylidene...)
Affinity DataEC50:  490nMAssay Description:Activity at human FPRL1-mediated calcium mobilization in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50186960(1-(2,3-dimethyl-5-oxo-1-phenyl-2,5-dihydro-1H-pyra...)
Affinity DataEC50:  980nMAssay Description:Activity at human FPRL1-mediated calcium mobilization in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50186965(1-(benzo[d][1,3]dioxol-5-yl)-3-(2,3-dimethyl-5-oxo...)
Affinity DataEC50:  5.88E+3nMAssay Description:Activity at human FPRL1-mediated calcium mobilization in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50186964(1-(2,3-dimethyl-5-oxo-1-phenyl-2,5-dihydro-1H-pyra...)
Affinity DataEC50: >1.00E+4nMAssay Description:Activity at human FPRL1-mediated calcium mobilization in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50186961(1-(3-isopropyl-2-methyl-5-oxo-1-(quinolin-3-yl)-2,...)
Affinity DataEC50:  30nMAssay Description:Activity at human FPRL1-mediated calcium mobilization in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50186962(1-(4-chlorophenyl)-3-(1-(4,5-dihydrothiazol-2-yl)-...)
Affinity DataEC50:  540nMAssay Description:Activity at human FPRL1-mediated calcium mobilization in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50186963(1-(4-chlorophenyl)-3-(3-isopropyl-2-methyl-5-oxo-1...)
Affinity DataEC50:  80nMAssay Description:Activity at human FPRL1-mediated calcium mobilization in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50186968(1-(3-isopropyl-2-methyl-5-oxo-1-(pyrimidin-5-yl)-2...)
Affinity DataEC50:  43nMAssay Description:Activity at human FPRL1-mediated calcium mobilization in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50186969(1-(1-(4,5-dihydrothiazol-2-yl)-3-isopropyl-2-methy...)
Affinity DataEC50:  1.47E+3nMAssay Description:Activity at human FPRL1-mediated calcium mobilization in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50186952(1-(2,3-dimethyl-5-oxo-1-phenyl-2,5-dihydro-1H-pyra...)
Affinity DataEC50:  30nMAssay Description:Activity at human FPRL1-mediated calcium mobilization in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50186967(1-(2,3-dimethyl-5-oxo-1-phenyl-2,5-dihydro-1H-pyra...)
Affinity DataEC50: >1.00E+4nMAssay Description:Activity at human FPRL1-mediated calcium mobilization in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50186966(1-(2,3-dimethyl-5-oxo-1-phenyl-2,5-dihydro-1H-pyra...)
Affinity DataEC50: >1.00E+4nMAssay Description:Activity at human FPRL1-mediated calcium mobilization in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50186970(1-(2,3-dimethyl-5-oxo-1-phenyl-2,5-dihydro-1H-pyra...)
Affinity DataEC50:  100nMAssay Description:Activity at human FPRL1-mediated calcium mobilization in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-formyl peptide receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50186939(1-(4-chlorophenyl)-3-(3-isopropyl-2-methyl-5-oxo-1...)
Affinity DataEC50:  250nMAssay Description:Activity at human FPRL1-mediated calcium mobilization in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed