Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50017877
LigandChemical structure of BindingDB Monomer ID 50187877BDBM50187877((S)-1-{2-[3-(3-fluoro-phenylsulfanyl)-biphenyl-4-y...)
Affinity DataIC50: 59nMAssay Description:Inhibition of [3H]glycine uptake at human GlyT1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50187888BDBM50187888((S)-1-{2-[3-(3-fluoro-phenylsulfanyl)-4'-methoxy-b...)
Affinity DataIC50: 160nMAssay Description:Inhibition of [3H]glycine uptake at human GlyT1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50187875BDBM50187875(2-(methyl(2-(2-(phenylthio)phenoxy)ethyl)amino)ace...)
Affinity DataIC50: 160nMAssay Description:Inhibition of [3H]glycine uptake at human GlyT1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50187869BDBM50187869((S)-1-{2-[3-(3-fluoro-phenylsulfanyl)-3'-methoxy-b...)
Affinity DataIC50: 300nMAssay Description:Inhibition of [3H]glycine uptake at human GlyT1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50187882BDBM50187882((S)-1-(2-(2-(3-chlorophenylthio)phenoxy)ethyl)pyrr...)
Affinity DataIC50: 380nMAssay Description:Inhibition of [3H]glycine uptake at human GlyT1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50187874BDBM50187874((S)-1-(2-(4-chloro-2-(3-fluorophenylthio)phenoxy)e...)
Affinity DataIC50: 400nMAssay Description:Inhibition of [3H]glycine uptake at human GlyT1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50187872BDBM50187872((2S)-1-(2-(2-(3-fluorophenylthio)-4-(thiophen-3-yl...)
Affinity DataIC50: 520nMAssay Description:Inhibition of [3H]glycine uptake at human GlyT1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50187890BDBM50187890((S)-1-(2-(5-chloro-2-(3-fluorophenylthio)phenoxy)e...)
Affinity DataIC50: 600nMAssay Description:Inhibition of [3H]glycine uptake at human GlyT1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50187889BDBM50187889((S)-1-{2-[4-(3-fluoro-phenylsulfanyl)-biphenyl-3-y...)
Affinity DataIC50: 950nMAssay Description:Inhibition of [3H]glycine uptake at human GlyT1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50187868BDBM50187868((S)-1-(2-(3-chloro-2-(3-fluorophenylthio)phenoxy)e...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of [3H]glycine uptake at human GlyT1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50187881BDBM50187881((S)-1-{2-[4'-chloro-3-(3-fluoro-phenylsulfanyl)-bi...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of [3H]glycine uptake at human GlyT1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50187886BDBM50187886(2-((2-(2-(3-chlorophenylthio)phenoxy)ethyl)(methyl...)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of [3H]glycine uptake at human GlyT1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50187873BDBM50187873(2-((2-(2-(3-fluorophenylthio)phenoxy)ethyl)(methyl...)
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of [3H]glycine uptake at human GlyT1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50187879BDBM50187879(2-((2-(2-(3-chlorophenylthio)phenoxy)ethyl)(ethyl)...)
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of [3H]glycine uptake at human GlyT1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50187871BDBM50187871(2-((2-(2-(4-chlorophenylthio)phenoxy)ethyl)(methyl...)
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibition of [3H]glycine uptake at human GlyT1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50187863BDBM50187863((S)-2-((1-(2-(3-fluorophenylthio)phenoxy)propan-2-...)
Affinity DataIC50: 8.90E+3nMAssay Description:Inhibition of [3H]glycine uptake at human GlyT1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50187866BDBM50187866(2-((2-(2-(4-tert-butylphenylthio)phenoxy)ethyl)(me...)
Affinity DataIC50: 9.20E+3nMAssay Description:Inhibition of [3H]glycine uptake at human GlyT1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50187864BDBM50187864(2-((1-(2-(3-fluorophenylthio)phenoxy)butan-2-yl)(m...)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of [3H]glycine uptake at human GlyT1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50187870BDBM50187870((R)-2-((1-(2-(3-fluorophenylthio)phenoxy)propan-2-...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of [3H]glycine uptake at human GlyT1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50187883BDBM50187883(2-((2-(2-(4-fluorophenylthio)phenoxy)ethyl)(methyl...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of [3H]glycine uptake at human GlyT1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50187885BDBM50187885(2-((1-(2-(3-fluorophenylthio)phenoxy)-3-methylbuta...)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of [3H]glycine uptake at human GlyT1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50187884BDBM50187884((S)-1-(2-(2-chloro-6-(3-fluorophenylthio)phenoxy)e...)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of [3H]glycine uptake at human GlyT1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50187878BDBM50187878((R)-1-(2-(2-(3-chlorophenylthio)phenoxy)ethyl)pyrr...)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of [3H]glycine uptake at human GlyT1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50187867BDBM50187867(2-((2-(2-(3-chlorophenylthio)phenoxy)ethyl)(methyl...)
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of [3H]glycine uptake at human GlyT1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50187865BDBM50187865(2-((2-(2-(4-methoxyphenylthio)phenoxy)ethyl)(methy...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of [3H]glycine uptake at human GlyT1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50187876BDBM50187876(2-(methyl(2-(2-(p-tolylthio)phenoxy)ethyl)amino)ac...)
Affinity DataIC50: 4.70E+4nMAssay Description:Inhibition of [3H]glycine uptake at human GlyT1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50187880BDBM50187880(2-((2-(2-(3-chlorophenylthio)phenoxy)ethyl)(ethyl)...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of [3H]glycine uptake at human GlyT1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50187887BDBM50187887(2-((2-(2-(4-acetamidophenylthio)phenoxy)ethyl)(met...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of [3H]glycine uptake at human GlyT1b transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed