Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 5775
TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandChemical structure of BindingDB Monomer ID 50261631BDBM50261631(Tetramic acid, 38 | CHEMBL468168 | 3-(3-(trifluoro...)
Affinity DataIC50: 6.00E+4nMT: 2°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandChemical structure of BindingDB Monomer ID 93272BDBM93272(Tetramic acid, 72)
Affinity DataIC50: 1.05E+5nMT: 2°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandChemical structure of BindingDB Monomer ID 93271BDBM93271(Tetramic acid, 56)
Affinity DataIC50: 1.45E+5nMT: 2°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandChemical structure of BindingDB Monomer ID 93267BDBM93267(Tetramic acid, 25)
Affinity DataIC50: 1.94E+5nMT: 2°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandChemical structure of BindingDB Monomer ID 93277BDBM93277(N-Substituted tetramic acid, 91)
Affinity DataIC50: 2.00E+5nMT: 2°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandChemical structure of BindingDB Monomer ID 93268BDBM93268(Tetramic acid, 30)
Affinity DataIC50: 2.00E+5nMT: 2°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandChemical structure of BindingDB Monomer ID 93270BDBM93270(Tetramic acid, 44)
Affinity DataIC50: 2.00E+5nMT: 2°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandChemical structure of BindingDB Monomer ID 93269BDBM93269(Tetramic acid, 43)
Affinity DataIC50: 2.00E+5nMT: 2°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandChemical structure of BindingDB Monomer ID 93276BDBM93276(N-Substituted tetramic acid, 89)
Affinity DataIC50: 2.00E+5nMT: 2°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandChemical structure of BindingDB Monomer ID 93275BDBM93275(Tetramic acid, 77)
Affinity DataIC50: 2.00E+5nMT: 2°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandChemical structure of BindingDB Monomer ID 93274BDBM93274(Tetramic acid, 76)
Affinity DataIC50: 2.00E+5nMT: 2°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandChemical structure of BindingDB Monomer ID 93273BDBM93273(Tetramic acid, 74)
Affinity DataIC50: 2.00E+5nMT: 2°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandChemical structure of BindingDB Monomer ID 93278BDBM93278(N-Substituted tetramic acid, 92)
Affinity DataIC50: 2.12E+5nMT: 2°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandChemical structure of BindingDB Monomer ID 93286BDBM93286(N-Substituted tetramic acid, 100)
Affinity DataIC50: 1.39E+8nMT: 2°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandChemical structure of BindingDB Monomer ID 93279BDBM93279(N-Substituted tetramic acid, 93)
Affinity DataIC50: 1.84E+8nMT: 2°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandChemical structure of BindingDB Monomer ID 93288BDBM93288(Sulfo-tetramic acid, 109)
Affinity DataIC50: 2.00E+8nMT: 2°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandChemical structure of BindingDB Monomer ID 93287BDBM93287(Sulfo-tetramic acid, 108)
Affinity DataIC50: 2.00E+8nMT: 2°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandChemical structure of BindingDB Monomer ID 93289BDBM93289(N-Substituted tetramic acid, 101)
Affinity DataIC50: 2.00E+8nMT: 2°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandChemical structure of BindingDB Monomer ID 93285BDBM93285(N-Substituted tetramic acid, 99)
Affinity DataIC50: 2.12E+8nMT: 2°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandChemical structure of BindingDB Monomer ID 93282BDBM93282(N-Substituted tetramic acid, 96)
Affinity DataIC50: 2.41E+8nMT: 2°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandChemical structure of BindingDB Monomer ID 93280BDBM93280(N-Substituted tetramic acid, 94)
Affinity DataIC50: 2.58E+8nMT: 2°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandChemical structure of BindingDB Monomer ID 93281BDBM93281(N-Substituted tetramic acid, 95)
Affinity DataIC50: 2.65E+8nMT: 2°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandChemical structure of BindingDB Monomer ID 93284BDBM93284(N-Substituted tetramic acid, 98)
Affinity DataIC50: 4.24E+8nMT: 2°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Darmstadt Technical University

LigandChemical structure of BindingDB Monomer ID 93283BDBM93283(N-Substituted tetramic acid, 97)
Affinity DataIC50: 4.59E+8nMT: 2°CAssay Description:The FRET assay was performed at 20 C on a FLUOstar (BMG Lab Technologies, D-77656 Offenburg) using 96-well microtiter plates (Dynex Microfluor 2, Cha...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2013
Entry Details Article
PubMed