Compile Data Set for Download or QSAR
Report error Found 41 Enz. Inhib. hit(s) with all data for entry = 50035888
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007887BDBM50007887(CHEMBL63742 | 3-Methyl-2-oxo-2,3-dihydro-benzoimid...)
Affinity DataKi:  0.890nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007868BDBM50007868(CHEMBL540017 | 2-Oxo-2,3-dihydro-benzoimidazole-1-...)
Affinity DataKi:  1.5nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007879BDBM50007879(CHEMBL293239 | 3-Methyl-2-oxo-2,3-dihydro-benzoimi...)
Affinity DataKi:  1.70nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50108392BDBM50108392((3-ENDO)-8-METHYL-8-AZABICYCLO[3.2.1]OCT-3-YL 1H-I...)
Affinity DataKi:  1.70nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007884BDBM50007884(CHEMBL64986 | 2-Oxo-2,3-dihydro-benzoimidazole-1-c...)
Affinity DataKi:  2.10nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007870BDBM50007870(CHEMBL539262 | 2-Oxo-2,3-dihydro-benzoimidazole-1-...)
Affinity DataKi:  2.20nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007872BDBM50007872(BIMU 1 | CHEMBL62023 | CHEMBL544755 | 3-Ethyl-2-ox...)
Affinity DataKi:  2.30nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007886BDBM50007886(CHEMBL293468 | 2-Oxo-2,3-dihydro-benzoimidazole-1-...)
Affinity DataKi:  3.80nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007881BDBM50007881(CHEMBL542869 | 4-Methyl-2-oxo-2,3-dihydro-benzoimi...)
Affinity DataKi:  7.90nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007858BDBM50007858(CHEMBL543340 | 3-Methyl-2-oxo-2,3-dihydro-benzoimi...)
Affinity DataKi:  12nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007882BDBM50007882(CHEMBL554389 | 2-Oxo-2,3-dihydro-benzoimidazole-1-...)
Affinity DataKi:  16nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007888BDBM50007888(CHEMBL545449 | 3-Ethyl-2-oxo-2,3-dihydro-benzoimid...)
Affinity DataKi:  18nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007857BDBM50007857(CHEMBL63891 | 2-Oxo-2,3-dihydro-benzoimidazole-1-c...)
Affinity DataKi:  20nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007874BDBM50007874(CHEMBL306003 | 2-Oxo-2,3-dihydro-benzoimidazole-1-...)
Affinity DataKi:  21nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 82561BDBM82561(TROPANYL 3,5-DICHLOROBENZOATE | CAS_40796-97-2 | T...)
Affinity DataKi:  24nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007869BDBM50007869(CHEMBL541040 | 5-Fluoro-2-oxo-2,3-dihydro-benzoimi...)
Affinity DataKi:  26nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007885BDBM50007885(CHEMBL539003 | 6-Fluoro-2-oxo-2,3-dihydro-benzoimi...)
Affinity DataKi:  34nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007893BDBM50007893(CHEMBL63409 | 8,8-Dimethyl-3-(2-oxo-2,3-dihydro-be...)
Affinity DataKi:  34nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007873BDBM50007873(CHEMBL552824 | 2-Oxo-2,3-dihydro-benzoimidazole-1-...)
Affinity DataKi:  72nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007897BDBM50007897(CHEMBL65226 | 2-Oxo-2,3-dihydro-benzoimidazole-1-c...)
Affinity DataKi:  130nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007860BDBM50007860(CHEMBL555995 | 7-Methyl-2-oxo-2,3-dihydro-benzoimi...)
Affinity DataKi:  306nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007866BDBM50007866(CHEMBL418673 | 2-Oxo-2,3-dihydro-benzoimidazole-1-...)
Affinity DataKi:  436nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007875BDBM50007875(CHEMBL67403 | 2-Oxo-2,3-dihydro-benzoimidazole-1-c...)
Affinity DataKi: >1.00E+3nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007863BDBM50007863(DAU 6285 | CHEMBL552854 | 6-Methoxy-2-oxo-2,3-dihy...)
Affinity DataKi: >1.00E+3nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007865BDBM50007865(CHEMBL554844 | 2-Oxo-2,3-dihydro-benzoimidazole-1-...)
Affinity DataKi: >1.00E+3nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007862BDBM50007862(CHEMBL63621 | 2-Oxo-2,3-dihydro-benzoimidazole-1-c...)
Affinity DataKi: >1.00E+3nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007883BDBM50007883(CHEMBL542634 | 2-Oxo-2,3-dihydro-benzoimidazole-1-...)
Affinity DataKi: >1.00E+3nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007890BDBM50007890(CHEMBL538247 | 6-Acetyl-2-oxo-2,3-dihydro-benzoimi...)
Affinity DataKi: >1.00E+3nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007895BDBM50007895(CHEMBL554755 | 5-Chloro-2-oxo-2,3-dihydro-benzoimi...)
Affinity DataKi: >1.00E+3nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007878BDBM50007878(CHEMBL539006 | 2-Oxo-5-trifluoromethyl-2,3-dihydro...)
Affinity DataKi: >1.00E+3nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007864BDBM50007864(CHEMBL541283 | 2-Oxo-2,3-dihydro-benzoimidazole-1-...)
Affinity DataKi: >1.00E+3nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007892BDBM50007892(DAU 6215 | CHEMBL539261 | 2-Oxo-2,3-dihydro-benzoi...)
Affinity DataKi: >1.00E+3nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007859BDBM50007859(CHEMBL540782 | 2-Oxo-2,3-dihydro-benzoimidazole-1-...)
Affinity DataKi: >1.00E+3nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007896BDBM50007896(CHEMBL553266 | 2-Oxo-2,3-dihydro-benzoimidazole-1-...)
Affinity DataKi: >1.00E+3nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007877BDBM50007877(CHEMBL539005 | 2-Oxo-2,3-dihydro-benzoimidazole-1-...)
Affinity DataKi: >1.00E+3nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007867BDBM50007867(CHEMBL555791 | 2-Oxo-2,3-dihydro-benzoimidazole-1-...)
Affinity DataKi: >1.00E+3nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007894BDBM50007894(CHEMBL555088 | 5,6-Dimethyl-2-oxo-2,3-dihydro-benz...)
Affinity DataKi: >1.00E+3nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007891BDBM50007891(CHEMBL66972 | 2-Oxo-2,3-dihydro-benzoimidazole-1-c...)
Affinity DataKi: >1.00E+3nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007880BDBM50007880(CHEMBL303463 | 2-Oxo-2,3-dihydro-benzoimidazole-1-...)
Affinity DataKi: >1.00E+3nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007876BDBM50007876(CHEMBL68348 | 5-Methoxy-2-oxo-2,3-dihydro-benzoimi...)
Affinity DataKi: >1.00E+3nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Istituto De Angeli

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007889BDBM50007889(CHEMBL304382 | 5-Methyl-2-oxo-2,3-dihydro-benzoimi...)
Affinity DataKi: >1.00E+3nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed