Compile Data Set for Download or QSAR
maximum 50k data
Found 146 Enz. Inhib. hit(s) with all data for entry = 50037783
TargetMu-type opioid receptor(GUINEA PIG)
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195673(CHEMBL267027 | N-cyclopropylmethyl-14beta-[3'-(4'-...)
Affinity DataKi:  0.0400nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195666(CHEMBL443311 | N-cyclopropylmethyl-14beta-[3'-(4'-...)
Affinity DataKi:  0.130nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM60212((4R,4aS,7aR,12bS)-3-(cyclopropylmethyl)-4a,9-bis(o...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetMu-type opioid receptor(GUINEA PIG)
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195659(CHEMBL217395 | N-cyclopropylmethyl-14beta-[3'-(4'-...)
Affinity DataKi:  0.240nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195678((1R,5R,13R,17S)-17-{[(2E)-3-(4-chlorophenyl)prop-2...)
Affinity DataKi:  0.320nMAssay Description:Displacement of [3H]diprenorphine from human mu opioid receptor expressed in C6 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM60212((4R,4aS,7aR,12bS)-3-(cyclopropylmethyl)-4a,9-bis(o...)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]U-69593 from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetMu-type opioid receptor(GUINEA PIG)
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM60212((4R,4aS,7aR,12bS)-3-(cyclopropylmethyl)-4a,9-bis(o...)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195660(CHEMBL384497 | N-cyclopropylmethyl-14beta-[3'-(4'-...)
Affinity DataKi:  0.590nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM60212((4R,4aS,7aR,12bS)-3-(cyclopropylmethyl)-4a,9-bis(o...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]U-69593 from kappa opioid receptor in guinea pig brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195673(CHEMBL267027 | N-cyclopropylmethyl-14beta-[3'-(4'-...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]Cl-DPDPE from delta receptor in guinea pig brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195678((1R,5R,13R,17S)-17-{[(2E)-3-(4-chlorophenyl)prop-2...)
Affinity DataKi:  0.630nMAssay Description:Displacement of [3H]diprenorphine from human recombinant delta opioid receptor expressed in C6 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195673(CHEMBL267027 | N-cyclopropylmethyl-14beta-[3'-(4'-...)
Affinity DataKi:  0.650nMAssay Description:Displacement of [3H]U-69593 from kappa opioid receptor in guinea pig brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195677((1R,5R,13R,17S)-17-{[(2E)-3-(4-chlorophenyl)prop-2...)
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195665(CHEMBL448428 | N-cyclopropylmethyl-14beta-[2'-(4''...)
Affinity DataKi:  0.730nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195663(CHEMBL217658 | N-cyclopropylmethyl-14beta-[2'-(4''...)
Affinity DataKi:  0.860nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195678((1R,5R,13R,17S)-17-{[(2E)-3-(4-chlorophenyl)prop-2...)
Affinity DataKi:  0.910nMAssay Description:Displacement of [3H]diprenorphine from human recombinant kappa opioid receptor expressed in C6 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195675(CHEMBL217102 | N-cyclopropylmethyl-14beta-[4'-(4''...)
Affinity DataKi:  0.960nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195665(CHEMBL448428 | N-cyclopropylmethyl-14beta-[2'-(4''...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]U-69593 from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195655(CHEMBL383896 | N-cyclopropylmethyl-14beta-[4'(4''-...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195666(CHEMBL443311 | N-cyclopropylmethyl-14beta-[3'-(4'-...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]Cl-DPDPE from delta receptor in guinea pig brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195669(CHEMBL411089 | N-cyclopropylmethyl-14beta-[4'-(4''...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195658(CHEMBL387101 | N-cyclopropylmethyl-14beta-[2'-(4''...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195676(CHEMBL217479 | N-cyclopropylmethyl-14beta-[4'-(4''...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195656(14beta-4'-Chlorocinnamoylaminodihydronormorphinone...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]U-69593 from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195663(CHEMBL217658 | N-cyclopropylmethyl-14beta-[2'-(4''...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]U-69593 from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195665(CHEMBL448428 | N-cyclopropylmethyl-14beta-[2'-(4''...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]Cl-DPDPE from human recombinant delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195670(CHEMBL216558 | N-cyclopropylmethyl-14beta-[4'-(4''...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195671(CHEMBL217710 | N-cyclopropylmethyl-14beta-[4'-(4''...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195666(CHEMBL443311 | N-cyclopropylmethyl-14beta-[3'-(4'-...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]U-69593 from kappa opioid receptor in guinea pig brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195663(CHEMBL217658 | N-cyclopropylmethyl-14beta-[2'-(4''...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]Cl-DPDPE from human recombinant delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195655(CHEMBL383896 | N-cyclopropylmethyl-14beta-[4'(4''-...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]Cl-DPDPE from human recombinant delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195675(CHEMBL217102 | N-cyclopropylmethyl-14beta-[4'-(4''...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]Cl-DPDPE from human recombinant delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195657(CHEMBL215926 | N-cyclopropylmethyl-14beta-[4'-(4''...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195672(CHEMBL277530 | N-cyclopropylmethyl-14beta-[2'-(4''...)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195672(CHEMBL277530 | N-cyclopropylmethyl-14beta-[2'-(4''...)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]U-69593 from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195656(14beta-4'-Chlorocinnamoylaminodihydronormorphinone...)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]Cl-DPDPE from human recombinant delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195676(CHEMBL217479 | N-cyclopropylmethyl-14beta-[4'-(4''...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]U-69593 from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195656(14beta-4'-Chlorocinnamoylaminodihydronormorphinone...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195671(CHEMBL217710 | N-cyclopropylmethyl-14beta-[4'-(4''...)
Affinity DataKi:  3.30nMAssay Description:Displacement of [3H]Cl-DPDPE from human recombinant delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195670(CHEMBL216558 | N-cyclopropylmethyl-14beta-[4'-(4''...)
Affinity DataKi:  3.70nMAssay Description:Displacement of [3H]U-69593 from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195655(CHEMBL383896 | N-cyclopropylmethyl-14beta-[4'(4''-...)
Affinity DataKi:  3.70nMAssay Description:Displacement of [3H]U-69593 from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195676(CHEMBL217479 | N-cyclopropylmethyl-14beta-[4'-(4''...)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]Cl-DPDPE from human recombinant delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195667(CHEMBL263482 | N-cyclopropylmethyl-14beta-[4'-(4''...)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195674(1N-[4-cyclopropylmethyl-10-methoxy-14-oxo-(17S)-12...)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]Cl-DPDPE from human recombinant delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195674(1N-[4-cyclopropylmethyl-10-methoxy-14-oxo-(17S)-12...)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195671(CHEMBL217710 | N-cyclopropylmethyl-14beta-[4'-(4''...)
Affinity DataKi:  4.90nMAssay Description:Displacement of [3H]U-69593 from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195659(CHEMBL217395 | N-cyclopropylmethyl-14beta-[3'-(4'-...)
Affinity DataKi:  5.10nMAssay Description:Displacement of [3H]Cl-DPDPE from delta receptor in guinea pig brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195675(CHEMBL217102 | N-cyclopropylmethyl-14beta-[4'-(4''...)
Affinity DataKi:  5.30nMAssay Description:Displacement of [3H]U-69593 from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM60212((4R,4aS,7aR,12bS)-3-(cyclopropylmethyl)-4a,9-bis(o...)
Affinity DataKi:  6.5nMAssay Description:Displacement of [3H]Cl-DPDPE from delta receptor in guinea pig brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50195659(CHEMBL217395 | N-cyclopropylmethyl-14beta-[3'-(4'-...)
Affinity DataKi:  6.5nMAssay Description:Displacement of [3H]U-69593 from kappa opioid receptor in guinea pig brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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