Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50003804
TargetIntegrin alpha-V/beta-3(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50237601([5-Benzyl-11-(3-guanidino-propyl)-8-isopropyl-3,6,...)
Affinity DataIC50: 0.487nMAssay Description:Inhibition of human alpha-v-beta-3 integrin receptor by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50063140((2R)-[(4-biphenylylsulfonyl) amino]-N-hydroxy-3-ph...)
Affinity DataIC50: 7.06nMAssay Description:Inhibition of human MMP9 by quenched fluorescense assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetCathepsin K(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50213272(CHEBI:6426 | Leupeptin)
Affinity DataIC50: 42.2nMAssay Description:Inhibition of human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetCathepsin K(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50323210(2,3-dihydroamentoflavone | CHEMBL220741)
Affinity DataIC50: 1.42E+3nMAssay Description:Inhibition of human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetCathepsin K(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50323196(4'-methylamentoflavone | bilobetin | CHEMBL378188)
Affinity DataIC50: 1.52E+3nMAssay Description:Inhibition of human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetCathepsin K(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50323214(CHEMBL291426 | 6-[4-(5,7-Dihydroxy-4-oxo-4H-chrome...)
Affinity DataIC50: 1.54E+3nMAssay Description:Inhibition of human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetCathepsin K(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50323204(7'',4'''-dimethylamentoflavone | CHEMBL374055)
Affinity DataIC50: 1.57E+3nMAssay Description:Inhibition of human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetCathepsin K(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50129952(cid_5281600 | CHEMBL63354 | 8-[5-(5,7-Dihydroxy-4-...)
Affinity DataIC50: 1.85E+3nMAssay Description:Inhibition of human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetCathepsin K(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50476091(CHEMBL434383 | 8,8''-Biskoenigine)
Affinity DataIC50: 1.94E+3nMAssay Description:Inhibition of human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetCathepsin K(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50323198(4'''-methylamentoflavone | podocarpusflavone A | C...)
Affinity DataIC50: 2.53E+3nMAssay Description:Inhibition of human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50476092(Aniasatin)
Affinity DataIC50: 1.76E+4nMAssay Description:Inhibition of human MMP9 by quenched fluorescense assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50476090(MELILOTOSIDE | CHEBI:17531)
Affinity DataIC50: 1.83E+4nMAssay Description:Inhibition of human alpha-v-beta-3 integrin receptor by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50131046(CHEMBL85139 | cid_65752 | rutaecarpine | 8,13-Dihy...)
Affinity DataIC50: 2.78E+4nMAssay Description:Inhibition of human MMP9 by quenched fluorescense assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed