Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 2666
TargetFalcipain 2(malaria parasite P. falciparum)
University of Cape Town

LigandPNGBDBM23157(1-{2-[(7-chloroquinolin-4-yl)amino]ethyl}-3-[(E)-{...)
Affinity DataIC50: 630nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2008
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
University of Cape Town

LigandPNGBDBM23156(1-{2-[(7-chloroquinolin-4-yl)amino]ethyl}-3-[(E)-{...)
Affinity DataIC50: 720nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2008
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
University of Cape Town

LigandPNGBDBM23152([(E)-[(3-{[4-(7-chloroquinolin-4-yl)piperazin-1-yl...)
Affinity DataIC50: 2.25E+3nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2008
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
University of Cape Town

LigandPNGBDBM23155(1-{2-[(7-chloroquinolin-4-yl)amino]ethyl}-3-[(E)-(...)
Affinity DataIC50: 2.60E+3nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2008
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
University of Cape Town

LigandPNGBDBM23160(1-{2-[(7-chloroquinolin-4-yl)amino]ethyl}-3-[(E)-[...)
Affinity DataIC50: 3.16E+3nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2008
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
University of Cape Town

LigandPNGBDBM23149([(E)-{[2,4-dihydroxy-3-(piperidin-1-ylmethyl)pheny...)
Affinity DataIC50: 3.80E+3nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2008
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
University of Cape Town

LigandPNGBDBM23148([(E)-{[2,4-dihydroxy-3-(pyrrolidin-1-ylmethyl)phen...)
Affinity DataIC50: 5.85E+3nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2008
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
University of Cape Town

LigandPNGBDBM23147([(E)-({3-[(diethylamino)methyl]-2,4-dihydroxypheny...)
Affinity DataIC50: 1.11E+4nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2008
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
University of Cape Town

LigandPNGBDBM23151([(E)-({2,4-dihydroxy-3-[(4-methylpiperazin-1-yl)me...)
Affinity DataIC50: 1.82E+4nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2008
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
University of Cape Town

LigandPNGBDBM23153([(E)-[(3-{[4-(7-chloroquinolin-4-yl)piperazin-1-yl...)
Affinity DataIC50: 2.00E+4nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2008
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
University of Cape Town

LigandPNGBDBM23154(2,4-dihydroxybenzaldehyde thiosemicarbazone | [(E)...)
Affinity DataIC50: 2.00E+4nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2008
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
University of Cape Town

LigandPNGBDBM23141(3-[(diethylamino)methyl]-2,4-dihydroxybenzaldehyde...)
Affinity DataIC50: 2.00E+4nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2008
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
University of Cape Town

LigandPNGBDBM23158(1-{2-[(7-chloroquinolin-4-yl)amino]ethyl}-3-[(E)-{...)
Affinity DataIC50: 2.00E+4nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2008
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
University of Cape Town

LigandPNGBDBM23142(2,4-dihydroxy-3-(pyrrolidin-1-ylmethyl)benzaldehyd...)
Affinity DataIC50: 2.00E+4nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2008
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
University of Cape Town

LigandPNGBDBM23159(1-{2-[(7-chloroquinolin-4-yl)amino]ethyl}-3-[(E)-(...)
Affinity DataIC50: 2.00E+4nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2008
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
University of Cape Town

LigandPNGBDBM23143(2,4-dihydroxy-3-(piperidin-1-ylmethyl)benzaldehyde...)
Affinity DataIC50: 2.00E+4nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2008
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
University of Cape Town

LigandPNGBDBM23144(2,4-dihydroxy-3-(morpholin-4-ylmethyl)benzaldehyde...)
Affinity DataIC50: 2.00E+4nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2008
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
University of Cape Town

LigandPNGBDBM23145(2,4-dihydroxy-3-[(4-methylpiperazin-1-yl)methyl]be...)
Affinity DataIC50: 2.00E+4nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2008
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
University of Cape Town

LigandPNGBDBM23146(3-{[4-(7-chloroquinolin-4-yl)piperazin-1-yl]methyl...)
Affinity DataIC50: 2.00E+4nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2008
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
University of Cape Town

LigandPNGBDBM23150([(E)-{[2,4-dihydroxy-3-(morpholin-4-ylmethyl)pheny...)
Affinity DataIC50: 2.00E+4nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2008
Entry Details Article
PubMed