Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50018550
TargetDipeptidyl peptidase 4(Human)
Tufts University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50050513(Ketopyrrolidine derivative | (R)-1-((S)-2-amino-3-...)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Tufts University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50196928((R)-1-((S)-2,4-diaminobutanamido)pentylboronic aci...)
Affinity DataIC50: 0.480nMAssay Description:Inhibition of human DPP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Tufts University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50196929((S)-2,4-diamino-1-((3aR,6aR)-hexahydrocyclopenta[b...)
Affinity DataIC50: 0.880nMAssay Description:Inhibition of human DPP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Tufts University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50050513(Ketopyrrolidine derivative | (R)-1-((S)-2-amino-3-...)
Affinity DataIC50: 2nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Tufts University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50050513(Ketopyrrolidine derivative | (R)-1-((S)-2-amino-3-...)
Affinity DataIC50: 17nMAssay Description:Inhibition of human DPP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProlyl endopeptidase FAP(Human)
Tufts University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50050513(Ketopyrrolidine derivative | (R)-1-((S)-2-amino-3-...)
Affinity DataIC50: 24nMAssay Description:Inhibition of human FAPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Tufts University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50050513(Ketopyrrolidine derivative | (R)-1-((S)-2-amino-3-...)
Affinity DataIC50: 30nMAssay Description:Inhibition of human DPP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Tufts University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50196928((R)-1-((S)-2,4-diaminobutanamido)pentylboronic aci...)
Affinity DataIC50: 800nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Tufts University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50196928((R)-1-((S)-2,4-diaminobutanamido)pentylboronic aci...)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of human DPP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProlyl endopeptidase(Human)
Tufts University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50050513(Ketopyrrolidine derivative | (R)-1-((S)-2-amino-3-...)
Affinity DataIC50: 7.96E+3nMAssay Description:Inhibition of prolyl oligopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProlyl endopeptidase(Human)
Tufts University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50196929((S)-2,4-diamino-1-((3aR,6aR)-hexahydrocyclopenta[b...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of prolyl oligopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProlyl endopeptidase(Human)
Tufts University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50196928((R)-1-((S)-2,4-diaminobutanamido)pentylboronic aci...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of prolyl oligopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Tufts University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50196929((S)-2,4-diamino-1-((3aR,6aR)-hexahydrocyclopenta[b...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human DPP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Tufts University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50196929((S)-2,4-diamino-1-((3aR,6aR)-hexahydrocyclopenta[b...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Tufts University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50196928((R)-1-((S)-2,4-diaminobutanamido)pentylboronic aci...)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Tufts University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50196929((S)-2,4-diamino-1-((3aR,6aR)-hexahydrocyclopenta[b...)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProlyl endopeptidase FAP(Human)
Tufts University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50196928((R)-1-((S)-2,4-diaminobutanamido)pentylboronic aci...)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of human FAPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProlyl endopeptidase FAP(Human)
Tufts University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50196929((S)-2,4-diamino-1-((3aR,6aR)-hexahydrocyclopenta[b...)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of human FAPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed