Compile Data Set for Download or QSAR
Report error Found 70 Enz. Inhib. hit(s) with all data for entry = 1572
LigandChemical structure of BindingDB Monomer ID 12255BDBM12255(CHEMBL217092 | N-(5-chloro-2H-1,3-benzodioxol-4-yl...)
Affinity DataIC50: 2.70nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandChemical structure of BindingDB Monomer ID 12241BDBM12241(N-(5-chloro-2H-1,3-benzodioxol-4-yl)-5-(oxan-4-ylo...)
Affinity DataIC50: 3nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12243BDBM12243(N-(2-chloro-5-methoxyphenyl)-7-[3-(4-methylpiperaz...)
Affinity DataIC50: 4nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12231BDBM12231(N-(2-chloro-5-methoxyphenyl)-7-[3-(morpholin-4-yl)...)
Affinity DataIC50: 4nMpH: 7.4 T: 2°CAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12247BDBM12247(N-(5-chloro-2H-1,3-benzodioxol-4-yl)-7-[3-(4-methy...)
Affinity DataIC50: 4nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12250BDBM12250(N-(5-Chloro-1,3-benzodioxol-4-yl)-7-(2-fluoroethox...)
Affinity DataIC50: 4nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12252BDBM12252(N-(5-chloro-2H-1,3-benzodioxol-4-yl)-5-(propan-2-y...)
Affinity DataIC50: 4nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12237BDBM12237(N-(5-chloro-2H-1,3-benzodioxol-4-yl)-5-(oxan-4-ylo...)
Affinity DataIC50: 4nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6218BDBM6218(AZD0530 analogue 34 | N-(5-chloro-2H-1,3-benzodiox...)
Affinity DataIC50: 5nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12259BDBM12259(N-(5-chloro-2H-1,3-benzodioxol-4-yl)-6-methoxy-7-[...)
Affinity DataIC50: 5nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12253BDBM12253(N-(5-chloro-2H-1,3-benzodioxol-4-yl)-7-[2-(morphol...)
Affinity DataIC50: 5nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12240BDBM12240(N-(5-chloro-2H-1,3-benzodioxol-4-yl)-7-[(1-methylp...)
Affinity DataIC50: 6nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12238BDBM12238(N-(5-chloro-2H-1,3-benzodioxol-4-yl)-5-(oxan-4-ylo...)
Affinity DataIC50: 6nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12251BDBM12251(N-(5-chloro-2H-1,3-benzodioxol-4-yl)-5-[(1-methylp...)
Affinity DataIC50: 7nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12246BDBM12246(N-(5-Chloro-1,3-benzodioxol-4-yl)-7-methoxy-5-(pip...)
Affinity DataIC50: 9.5nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6198BDBM6198(AZD0530 analogue 35 | M475271 | N-(2-Chloro-5-meth...)
Affinity DataIC50: 10nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12228BDBM12228(N-(5-chloro-2H-1,3-benzodioxol-4-yl)-7-methoxy-5-[...)
Affinity DataIC50: 10nMpH: 7.4 T: 2°CAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12258BDBM12258(N-(5-chloro-2H-1,3-benzodioxol-4-yl)-5-methoxy-7-[...)
Affinity DataIC50: 15nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12229BDBM12229(N-(2-chloro-5-methoxyphenyl)-7-[3-(morpholin-4-yl)...)
Affinity DataIC50: 20nMpH: 7.4 T: 2°CAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12230BDBM12230(N-(2-chloro-5-methoxyphenyl)-5-(cyclohexyloxy)-7-[...)
Affinity DataIC50: 20nMpH: 7.4 T: 2°CAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12254BDBM12254(1-{4-[2-({4-[(5-fluoro-2H-1,3-benzodioxol-4-yl)ami...)
Affinity DataIC50: 20nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12227BDBM12227(N-(2-chloro-5-methoxyphenyl)-7-methoxy-5-[(1-methy...)
Affinity DataIC50: 30nMpH: 7.4 T: 2°CAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12232BDBM12232(N-(2-chloro-5-methoxyphenyl)-7-[3-(morpholin-4-yl)...)
Affinity DataIC50: 30nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12232BDBM12232(N-(2-chloro-5-methoxyphenyl)-7-[3-(morpholin-4-yl)...)
Affinity DataIC50: 40nMpH: 7.4 T: 2°CAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12233BDBM12233(N-(2H-1,3-benzodioxol-4-yl)-5-(oxan-4-yloxy)-7-[3-...)
Affinity DataIC50: 40nMpH: 7.4 T: 2°CAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12243BDBM12243(N-(2-chloro-5-methoxyphenyl)-7-[3-(4-methylpiperaz...)
Affinity DataIC50: 40nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12239BDBM12239(N-(2,3-dihydro-1,4-benzodioxin-5-yl)-5-(oxan-4-ylo...)
Affinity DataIC50: 50nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12231BDBM12231(N-(2-chloro-5-methoxyphenyl)-7-[3-(morpholin-4-yl)...)
Affinity DataIC50: 50nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12245BDBM12245(N-(5-chloro-2H-1,3-benzodioxol-4-yl)-5-(piperidin-...)
Affinity DataIC50: 55nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12264BDBM12264(N-(6-chloro-2,3-dihydro-1,4-benzodioxin-5-yl)-7-[2...)
Affinity DataIC50: 65nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12242BDBM12242(N-(5-chloro-2H-1,3-benzodioxol-4-yl)-5-(morpholin-...)
Affinity DataIC50: 75nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12236BDBM12236(N-(2H-1,3-benzodioxol-4-yl)-5-(oxan-4-yloxy)-7-[2-...)
Affinity DataIC50: 80nMpH: 7.4 T: 2°CAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12239BDBM12239(N-(2,3-dihydro-1,4-benzodioxin-5-yl)-5-(oxan-4-ylo...)
Affinity DataIC50: 85nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12233BDBM12233(N-(2H-1,3-benzodioxol-4-yl)-5-(oxan-4-yloxy)-7-[3-...)
Affinity DataIC50: 100nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12225BDBM12225(N-(5-chloro-2H-1,3-benzodioxol-4-yl)-5-[(1-methylp...)
Affinity DataIC50: 100nMpH: 7.4 T: 2°CAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12249BDBM12249(N-(5-Chloro-1,3-benzodioxol-4-yl)-7-isopropoxy-5-[...)
Affinity DataIC50: 100nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12263BDBM12263(N-(6-chloro-2,3-dihydro-1,4-benzodioxin-5-yl)-5-(o...)
Affinity DataIC50: 110nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12234BDBM12234(N-(2H-1,3-benzodioxol-4-yl)-7-methoxy-5-[(1-methyl...)
Affinity DataIC50: 150nMpH: 7.4 T: 2°CAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12226BDBM12226(N-(2-Chloro-5-methoxyphenyl)-7-methoxy-5-(3-morpho...)
Affinity DataIC50: 230nMpH: 7.4 T: 2°CAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12244BDBM12244(N-(2-chloro-5-methoxyphenyl)-6,7-dimethoxyquinazol...)
Affinity DataIC50: 250nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12223BDBM12223(N-(2-Chloro-5-methoxyphenyl)-5-[(1-methylpiperidin...)
Affinity DataIC50: 300nMpH: 7.4 T: 2°CAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12224BDBM12224(N-(2-chloro-5-methoxyphenyl)-5-(oxan-4-yloxy)quina...)
Affinity DataIC50: 400nMpH: 7.4 T: 2°CAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12229BDBM12229(N-(2-chloro-5-methoxyphenyl)-7-[3-(morpholin-4-yl)...)
Affinity DataIC50: 400nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12235BDBM12235(N-(2,3-dihydro-1,4-benzodioxin-5-yl)-7-methoxy-5-[...)
Affinity DataIC50: 500nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12248BDBM12248(N-(5-chloro-2H-1,3-benzodioxol-4-yl)-5-[(1-methylp...)
Affinity DataIC50: 500nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12260BDBM12260(N-(2-Chloro-5-methoxyphenyl)-6-methoxy-5-[(1-methy...)
Affinity DataIC50: 540nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12235BDBM12235(N-(2,3-dihydro-1,4-benzodioxin-5-yl)-7-methoxy-5-[...)
Affinity DataIC50: 570nMpH: 7.4 T: 2°CAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12262BDBM12262(N-(2-Chloro-5-methoxyphenyl)-6-[3-(4-methylpiperaz...)
Affinity DataIC50: 600nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 12236BDBM12236(N-(2H-1,3-benzodioxol-4-yl)-5-(oxan-4-yloxy)-7-[2-...)
Affinity DataIC50: 650nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6198BDBM6198(AZD0530 analogue 35 | M475271 | N-(2-Chloro-5-meth...)
Affinity DataIC50: 670nMAssay Description:This assay determines the ability of test compounds to inhibit Src kinase activity that catalyzes the transfer of the terminal phosphate to the immob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2006
Entry Details Article
PubMed
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