Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50018754
TargetVitamin D3 receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50198707((2Z)-(20S)-1alpha,25-dihydroxy-2-[2''''-(fluoroeth...)
Affinity DataEC50:  0.0700nMAssay Description:Inhibition of human VDR induced-transcriptional transactivation of luciferase reporter gene in COS7 cells after 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50198705(CHEMBL226435 | (2Z)-(20R)-1alpha,25-dihydroxy-2-[(...)
Affinity DataEC50:  0.5nMAssay Description:Inhibition of human VDR induced-transcriptional transactivation of luciferase reporter gene in COS7 cells after 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50198707((2Z)-(20S)-1alpha,25-dihydroxy-2-[2''''-(fluoroeth...)
Affinity DataEC50:  1.10nMAssay Description:Inhibition of human VDR induced-transcriptional transactivation of luciferase reporter gene in COS7 cells after 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50198705(CHEMBL226435 | (2Z)-(20R)-1alpha,25-dihydroxy-2-[(...)
Affinity DataEC50:  2.20nMAssay Description:Inhibition of human VDR induced-transcriptional transactivation of luciferase reporter gene in COS7 cells after 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed