Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 50003830
TargetUrotensin-2 receptor(Human)
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50476310(CHEMBL228470)
Affinity DataEC50:  129nMAssay Description:Agonist activity at human urotensin-2 receptor transfected in NIH3T3 cells after 5 days by R-SAT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50476328(CHEMBL229713)
Affinity DataEC50:  135nMAssay Description:Agonist activity at human urotensin-2 receptor transfected in NIH3T3 cells after 5 days by R-SAT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50476307(CHEMBL229710)
Affinity DataEC50:  372nMAssay Description:Agonist activity at human urotensin-2 receptor transfected in NIH3T3 cells after 5 days by R-SAT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50476311(CHEMBL229714)
Affinity DataEC50:  380nMAssay Description:Agonist activity at human urotensin-2 receptor transfected in NIH3T3 cells after 5 days by R-SAT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50476318(CHEMBL228471)
Affinity DataEC50:  398nMAssay Description:Agonist activity at human urotensin-2 receptor transfected in NIH3T3 cells after 5 days by R-SAT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50476308(CHEMBL374817)
Affinity DataEC50:  427nMAssay Description:Agonist activity at human urotensin-2 receptor transfected in NIH3T3 cells after 5 days by R-SAT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50476321(CHEMBL229923)
Affinity DataEC50:  437nMAssay Description:Agonist activity at human urotensin-2 receptor transfected in NIH3T3 cells after 5 days by R-SAT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50476309(CHEMBL229764)
Affinity DataEC50:  457nMAssay Description:Agonist activity at human urotensin-2 receptor transfected in NIH3T3 cells after 5 days by R-SAT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50476315(CHEMBL387661)
Affinity DataEC50:  513nMAssay Description:Agonist activity at human urotensin-2 receptor transfected in NIH3T3 cells after 5 days by R-SAT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50476329(CHEMBL390792)
Affinity DataEC50:  575nMAssay Description:Agonist activity at human urotensin-2 receptor transfected in NIH3T3 cells after 5 days by R-SAT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50476325(CHEMBL387694)
Affinity DataEC50:  589nMAssay Description:Agonist activity at human urotensin-2 receptor transfected in NIH3T3 cells after 5 days by R-SAT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50476332(CHEMBL229709)
Affinity DataEC50:  603nMAssay Description:Agonist activity at human urotensin-2 receptor transfected in NIH3T3 cells after 5 days by R-SAT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50476316(CHEMBL228411)
Affinity DataEC50:  871nMAssay Description:Agonist activity at human urotensin-2 receptor transfected in NIH3T3 cells after 5 days by R-SAT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50476327(CHEMBL228525)
Affinity DataEC50:  1.12E+3nMAssay Description:Agonist activity at human urotensin-2 receptor transfected in NIH3T3 cells after 5 days by R-SAT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50476320(CHEMBL228413)
Affinity DataEC50:  1.12E+3nMAssay Description:Agonist activity at human urotensin-2 receptor transfected in NIH3T3 cells after 5 days by R-SAT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50476313(CHEMBL413787)
Affinity DataEC50:  1.41E+3nMAssay Description:Agonist activity at human urotensin-2 receptor transfected in NIH3T3 cells after 5 days by R-SAT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50476319(CHEMBL375275)
Affinity DataEC50:  1.51E+3nMAssay Description:Agonist activity at human urotensin-2 receptor transfected in NIH3T3 cells after 5 days by R-SAT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50476312(CHEMBL376582)
Affinity DataEC50:  1.55E+3nMAssay Description:Agonist activity at human urotensin-2 receptor transfected in NIH3T3 cells after 5 days by R-SAT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50476333(CHEMBL228412)
Affinity DataEC50:  1.66E+3nMAssay Description:Agonist activity at human urotensin-2 receptor transfected in NIH3T3 cells after 5 days by R-SAT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50476324(CHEMBL442230)
Affinity DataEC50:  1.74E+3nMAssay Description:Agonist activity at human urotensin-2 receptor transfected in NIH3T3 cells after 5 days by R-SAT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50475729(CHEMBL206596)
Affinity DataEC50:  1.86E+3nMAssay Description:Agonist activity at human urotensin-2 receptor transfected in NIH3T3 cells after 5 days by R-SAT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50476330(CHEMBL229924)
Affinity DataEC50:  2.00E+3nMAssay Description:Agonist activity at human urotensin-2 receptor transfected in NIH3T3 cells after 5 days by R-SAT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50476306(CHEMBL229868)
Affinity DataEC50:  2.29E+3nMAssay Description:Agonist activity at human urotensin-2 receptor transfected in NIH3T3 cells after 5 days by R-SAT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50476326(CHEMBL228461)
Affinity DataEC50:  2.95E+3nMAssay Description:Agonist activity at human urotensin-2 receptor transfected in NIH3T3 cells after 5 days by R-SAT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50476331(CHEMBL229659)
Affinity DataEC50:  3.09E+3nMAssay Description:Agonist activity at human urotensin-2 receptor transfected in NIH3T3 cells after 5 days by R-SAT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50476323(CHEMBL228472)
Affinity DataEC50:  4.17E+3nMAssay Description:Agonist activity at human urotensin-2 receptor transfected in NIH3T3 cells after 5 days by R-SAT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50476314(CHEMBL376581)
Affinity DataEC50:  4.57E+3nMAssay Description:Agonist activity at human urotensin-2 receptor transfected in NIH3T3 cells after 5 days by R-SAT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50476317(CHEMBL229922)
Affinity DataEC50:  5.37E+3nMAssay Description:Agonist activity at human urotensin-2 receptor transfected in NIH3T3 cells after 5 days by R-SAT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
G£Teborg University

Curated by ChEMBL
LigandPNGBDBM50476322(CHEMBL228526)
Affinity DataEC50:  5.89E+3nMAssay Description:Agonist activity at human urotensin-2 receptor transfected in NIH3T3 cells after 5 days by R-SAT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed