Compile Data Set for Download or QSAR
Report error Found 73 Enz. Inhib. hit(s) with all data for entry = 50037927
TargetGlucocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM18207(dexamethasone (tetramethyl-rhodamine conjugated ) ...)
Affinity DataIC50: 3.40nMAssay Description:Inhibition of human GRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198964((S)-N-(1-(1H-indol-3-yl)propan-2-yl)-2,4,6-trimeth...)
Affinity DataIC50: 29nMAssay Description:Inhibition of human GRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM18207(dexamethasone (tetramethyl-rhodamine conjugated ) ...)
Affinity DataIC50: 33nMAssay Description:Inhibition of human MRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198946(N-(1-(1H-indol-3-yl)propan-2-yl)-2,4,6-trimethylbe...)
Affinity DataIC50: 40nMAssay Description:Inhibition of human GRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198950(N-(1-(1H-indol-3-yl)butan-2-yl)-2,4,6-trichloroben...)
Affinity DataIC50: 64nMAssay Description:Inhibition of human GRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198973(N-(1-(1H-indol-3-yl)propan-2-yl)-2,4,6-trichlorobe...)
Affinity DataIC50: 64nMAssay Description:Inhibition of human GRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198991(N-(1-(5-fluoro-1H-indol-3-yl)propan-2-yl)-2,4,6-tr...)
Affinity DataIC50: 65nMAssay Description:Inhibition of human GRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198956(N-(1-(1H-indol-3-yl)propan-2-yl)-2,4,6-triisopropy...)
Affinity DataIC50: 67nMAssay Description:Inhibition of human GRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198961(N-(1-(6-fluoro-1H-indol-3-yl)propan-2-yl)-2,4,6-tr...)
Affinity DataIC50: 79nMAssay Description:Inhibition of human GRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198974(2,4,6-trimethyl-N-(1-(7-methyl-1H-indol-3-yl)propa...)
Affinity DataIC50: 120nMAssay Description:Inhibition of human GRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198973(N-(1-(1H-indol-3-yl)propan-2-yl)-2,4,6-trichlorobe...)
Affinity DataIC50: 130nMAssay Description:Inhibition of human MRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198945(N-(1-(1H-indol-3-yl)propan-2-yl)-2,6-dichlorobenze...)
Affinity DataIC50: 170nMAssay Description:Inhibition of human PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198945(N-(1-(1H-indol-3-yl)propan-2-yl)-2,6-dichlorobenze...)
Affinity DataIC50: 240nMAssay Description:Inhibition of human GRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198943(N-(1-(1H-indol-3-yl)propan-2-yl)-2-chloro-6-methyl...)
Affinity DataIC50: 280nMAssay Description:Inhibition of human GRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198946(N-(1-(1H-indol-3-yl)propan-2-yl)-2,4,6-trimethylbe...)
Affinity DataIC50: 290nMAssay Description:Inhibition of human MRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198959(N-(1-(1H-indol-3-yl)propan-2-yl)-2,4,5-trichlorobe...)
Affinity DataIC50: 440nMAssay Description:Inhibition of human PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198953(N-(1-(1H-indol-3-yl)propan-2-yl)-2,4-dichlorobenze...)
Affinity DataIC50: 480nMAssay Description:Inhibition of human GRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198971(2,4,6-trimethyl-N-(1-(6-methyl-1H-indol-3-yl)propa...)
Affinity DataIC50: 490nMAssay Description:Inhibition of human GRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198978((R)-N-(1-(1H-indol-3-yl)propan-2-yl)-2,4,6-trimeth...)
Affinity DataIC50: 520nMAssay Description:Inhibition of human MRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198965(2,4,6-trichloro-N-(1-(2-methyl-1H-indol-3-yl)propa...)
Affinity DataIC50: 570nMAssay Description:Inhibition of human GRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198973(N-(1-(1H-indol-3-yl)propan-2-yl)-2,4,6-trichlorobe...)
Affinity DataIC50: 570nMAssay Description:Inhibition of human PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198947(N-(1-(1H-indol-3-yl)propan-2-yl)-4-tert-butylbenze...)
Affinity DataIC50: 735nMAssay Description:Inhibition of human GRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198968(N-(1-(1H-indol-3-yl)propan-2-yl)-4-isopropylbenzen...)
Affinity DataIC50: 750nMAssay Description:Inhibition of human GRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198989(N-(1-(1H-indol-3-yl)propan-2-yl)-3-chloro-2-methyl...)
Affinity DataIC50: 820nMAssay Description:Inhibition of human GRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198953(N-(1-(1H-indol-3-yl)propan-2-yl)-2,4-dichlorobenze...)
Affinity DataIC50: 850nMAssay Description:Inhibition of human MRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198959(N-(1-(1H-indol-3-yl)propan-2-yl)-2,4,5-trichlorobe...)
Affinity DataIC50: 990nMAssay Description:Inhibition of human GRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198959(N-(1-(1H-indol-3-yl)propan-2-yl)-2,4,5-trichlorobe...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human MRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198964((S)-N-(1-(1H-indol-3-yl)propan-2-yl)-2,4,6-trimeth...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human MRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198968(N-(1-(1H-indol-3-yl)propan-2-yl)-4-isopropylbenzen...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198947(N-(1-(1H-indol-3-yl)propan-2-yl)-4-tert-butylbenze...)
Affinity DataIC50: 1.07E+3nMAssay Description:Inhibition of human MRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198966(N-(1-(1H-indol-3-yl)propan-2-yl)-2,3-dichlorobenze...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human GRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198964((S)-N-(1-(1H-indol-3-yl)propan-2-yl)-2,4,6-trimeth...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198987(N-(1-(1H-indol-3-yl)propan-2-yl)-N,2,4,6-tetrameth...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human GRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198949(N-(1-(1H-indol-3-yl)propan-2-yl)-2,5-dichlorobenze...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human GRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198968(N-(1-(1H-indol-3-yl)propan-2-yl)-4-isopropylbenzen...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human MRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198946(N-(1-(1H-indol-3-yl)propan-2-yl)-2,4,6-trimethylbe...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198944(N-(1-(1H-indol-3-yl)propan-2-yl)-4-propylbenzenesu...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human GRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198945(N-(1-(1H-indol-3-yl)propan-2-yl)-2,6-dichlorobenze...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human MRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198986(N-(1-(1H-indol-3-yl)propan-2-yl)-4-chloro-2,5-dime...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of human GRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198975(N-(1-(1H-indol-3-yl)propan-2-yl)-2,3,4-trichlorobe...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of human GRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198969(1-(1-(1H-indol-3-yl)propan-2-yl)-3-(2,4,6-trichlor...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human GRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198988([2-(1H-indol-3-yl)-1-methyl-ethyl]-(2,4,6-trimethy...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human GRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198978((R)-N-(1-(1H-indol-3-yl)propan-2-yl)-2,4,6-trimeth...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human GRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198956(N-(1-(1H-indol-3-yl)propan-2-yl)-2,4,6-triisopropy...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198956(N-(1-(1H-indol-3-yl)propan-2-yl)-2,4,6-triisopropy...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human MRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM18207(dexamethasone (tetramethyl-rhodamine conjugated ) ...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198990(2,4,6-trichloro-N-(1-(5-methoxy-1H-indol-3-yl)prop...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human GRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198948(2,4,6-trichloro-N-(1-(1-methyl-1H-indol-3-yl)propa...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human GRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198980(N-(1-(1H-indol-2-yl)propan-2-yl)-2,4,6-trimethylbe...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human GRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50198947(N-(1-(1H-indol-3-yl)propan-2-yl)-4-tert-butylbenze...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human PRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
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