Compile Data Set for Download or QSAR
maximum 50k data
Found 23 Enz. Inhib. hit(s) with all data for entry = 50018841
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199575((1-(4-chlorophenoxy)-9-((1-methylpiperidin-4-yl)me...)
Affinity DataIC50:  11nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199586(2-(4-((1-(4-chlorophenoxy)-3-(1-methylpiperazine-4...)
Affinity DataIC50:  14nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199587((1-(4-chlorophenoxy)-9-(piperidin-4-ylmethyl)-9H-c...)
Affinity DataIC50:  16nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199580((1-(4-chlorophenoxy)-9-(((3R,4S)-3-fluoro-1-methyl...)
Affinity DataIC50:  28nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199584((1-(4-chlorophenoxy)-9-((3-fluoro-1,2,5,6-tetrahyd...)
Affinity DataIC50:  43nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199579(1-(4-chlorophenoxy)-N-(2-(dimethylamino)ethyl)-9-(...)
Affinity DataIC50:  50nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199577((1-(4-chlorophenoxy)-9-(3-(piperidin-1-yl)propyl)-...)
Affinity DataIC50:  50nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199585((1-(4-chlorophenoxy)-9-(((3R,4S)-3-fluoropiperidin...)
Affinity DataIC50:  51nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199570((1-(4-chlorophenoxy)-9-(((3S,4S)-3-fluoropiperidin...)
Affinity DataIC50:  53nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199574((1-(4-chlorophenoxy)-9-(((3S,4S)-3-fluoro-1-methyl...)
Affinity DataIC50:  95nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199573((1-(4-chlorophenoxy)-9-(piperidin-3-ylmethyl)-9H-c...)
Affinity DataIC50:  107nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199581((1-(4-chlorophenoxy)-9-(((3R,4S)-1-cyclopropyl-3-f...)
Affinity DataIC50:  186nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199572(1-(4-chlorophenoxy)-N-(2-(dimethylamino)ethyl)-9-(...)
Affinity DataIC50:  191nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199571(1-(4-chlorophenoxy)-N-((1-ethylpyrrolidin-2-yl)met...)
Affinity DataIC50:  263nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199583((1-(4-chlorophenoxy)-9-(((3S,4S)-3-fluoropiperidin...)
Affinity DataIC50:  467nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199588((1-(4-chlorophenoxy)-9-(((3R,4S)-3-fluoropiperidin...)
Affinity DataIC50:  832nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199589((1-(4-chlorophenoxy)-9-(((3S,4S)-3-fluoropiperidin...)
Affinity DataIC50:  871nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199590(1-(4-chlorophenoxy)-9-(((3S,4S)-3-fluoropiperidin-...)
Affinity DataIC50:  1.86E+3nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199578((1-(4-chlorophenoxy)-9-(((3R,4S)-3-fluoropiperidin...)
Affinity DataIC50:  1.91E+3nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199582((1-(4-chlorophenoxy)-9-(((3R,4S)-3-fluoropiperidin...)
Affinity DataIC50:  2.88E+3nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199591((1-(4-chlorophenoxy)-9-(((3R,4S)-3-fluoropiperidin...)
Affinity DataIC50:  7.76E+3nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199576((1-(4-chlorophenoxy)-9-(((3R,4S)-3-fluoropiperidin...)
Affinity DataIC50:  9.77E+3nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199569(1-(4-chlorophenoxy)-9-(((3S,4S)-3-fluoropiperidin-...)
Affinity DataIC50:  1.20E+4nMAssay Description:Displacement of [125]peptide YY from human recombinant Y1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed