Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50018928
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184359(MT-II | CHEMBL430239 | Ac-Nle-c[Asp-His-DPhe-Arg-T...)
Affinity DataIC50: 0.200nMAssay Description:Displacement of [125I]NDP-alphaMSH from human MC1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184359(MT-II | CHEMBL430239 | Ac-Nle-c[Asp-His-DPhe-Arg-T...)
Affinity DataEC50:  0.300nMAssay Description:Activity at hMC1R transfected in HEK293 cells assessed as intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50200356(Ac-c[Cys-His-D-Phe-Cys]-N-alpha-guanidinylbutyl-D-...)
Affinity DataIC50: 0.700nMAssay Description:Displacement of [125I]NDP-alphaMSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184359(MT-II | CHEMBL430239 | Ac-Nle-c[Asp-His-DPhe-Arg-T...)
Affinity DataIC50: 1.10nMAssay Description:Displacement of [125I]NDP-alphaMSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50200360(Ac-c[Cys-His-D-Phe-N-alpha-guanidinylbutyl-Cys]-Tr...)
Affinity DataIC50: 1.80nMAssay Description:Displacement of [125I]NDP-alphaMSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184359(MT-II | CHEMBL430239 | Ac-Nle-c[Asp-His-DPhe-Arg-T...)
Affinity DataEC50:  1.90nMAssay Description:Activity at hMC3R transfected in HEK293 cells assessed as intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184359(MT-II | CHEMBL430239 | Ac-Nle-c[Asp-His-DPhe-Arg-T...)
Affinity DataIC50: 2nMAssay Description:Displacement of [125I]NDP-alphaMSH from human MC3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184359(MT-II | CHEMBL430239 | Ac-Nle-c[Asp-His-DPhe-Arg-T...)
Affinity DataEC50:  2.90nMAssay Description:Displacement of [125I]NDP-alphaMSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184359(MT-II | CHEMBL430239 | Ac-Nle-c[Asp-His-DPhe-Arg-T...)
Affinity DataEC50:  3.30nMAssay Description:Displacement of [125I]NDP-alphaMSH from human MC5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50200361(Ac-c[Cys-His-D-Phe-Cys]-N-alpha-guanidinylbutyl-Tr...)
Affinity DataIC50: 4.10nMAssay Description:Displacement of [125I]NDP-alphaMSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184359(MT-II | CHEMBL430239 | Ac-Nle-c[Asp-His-DPhe-Arg-T...)
Affinity DataIC50: 7.5nMAssay Description:Displacement of [125I]NDP-alphaMSH from human MC5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50200358(Ac-c[Glu-His-D-Phe-N-alpha-guanidinylbutyl-Orn]-Tr...)
Affinity DataIC50: 101nMAssay Description:Displacement of [125I]NDP-alphaMSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50200359(Ac-c[Cys-His-D-Nal(2)'-Cys]-N-alpha-guanidinylbuty...)
Affinity DataIC50: 209nMAssay Description:Displacement of [125I]NDP-alphaMSH from human MC5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50200358(Ac-c[Glu-His-D-Phe-N-alpha-guanidinylbutyl-Orn]-Tr...)
Affinity DataIC50: 750nMAssay Description:Displacement of [125I]NDP-alphaMSH from human MC1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50200361(Ac-c[Cys-His-D-Phe-Cys]-N-alpha-guanidinylbutyl-Tr...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]NDP-alphaMSH from human MC1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50200357(Ac-c[Glu-His-D-Nal(2)'-N-alpha-guanidinylbutyl-Orn...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]NDP-alphaMSH from human MC3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50200358(Ac-c[Glu-His-D-Phe-N-alpha-guanidinylbutyl-Orn]-Tr...)
Affinity DataEC50: >1.00E+3nMAssay Description:Displacement of [125I]NDP-alphaMSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50200358(Ac-c[Glu-His-D-Phe-N-alpha-guanidinylbutyl-Orn]-Tr...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]NDP-alphaMSH from human MC3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50200356(Ac-c[Cys-His-D-Phe-Cys]-N-alpha-guanidinylbutyl-D-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]NDP-alphaMSH from human MC3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50200355(Ac-c[Glu-His-D-Phe-N-alpha-guanidinylbutyl-Dab]-Tr...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]NDP-alphaMSH from human MC1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50200355(Ac-c[Glu-His-D-Phe-N-alpha-guanidinylbutyl-Dab]-Tr...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]NDP-alphaMSH from human MC3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50200361(Ac-c[Cys-His-D-Phe-Cys]-N-alpha-guanidinylbutyl-Tr...)
Affinity DataEC50: >1.00E+3nMAssay Description:Displacement of [125I]NDP-alphaMSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50200354(Ac-c[Cys-His-D-Phe-N-alpha-guanidinylbutyl-D-Cys]-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]NDP-alphaMSH from human MC1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50200356(Ac-c[Cys-His-D-Phe-Cys]-N-alpha-guanidinylbutyl-D-...)
Affinity DataEC50: >1.00E+3nMAssay Description:Displacement of [125I]NDP-alphaMSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50200361(Ac-c[Cys-His-D-Phe-Cys]-N-alpha-guanidinylbutyl-Tr...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]NDP-alphaMSH from human MC3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50200359(Ac-c[Cys-His-D-Nal(2)'-Cys]-N-alpha-guanidinylbuty...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]NDP-alphaMSH from human MC1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50200357(Ac-c[Glu-His-D-Nal(2)'-N-alpha-guanidinylbutyl-Orn...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]NDP-alphaMSH from human MC1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed