TargetAlpha-2A adrenergic receptor [16-465](Rattus norvegicus (rat))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to adrenergic alpha2A receptor in Sprague-Dawley rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of [3H]noradrenaline uptake in Sprague-Dawley rat brain synaptosomesMore data for this Ligand-Target Pair