Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50019212
Target5-hydroxytryptamine receptor 2A(Rat)
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50202762(N-(4-(3-(4-m-tolylpiperazin-1-yl)propylthio)phenyl...)
Affinity DataKi:  6.09nMAssay Description:Displacement of [3H]ketanserin from rat cloned 5HT2A receptor expressed in NIH-3T3-GF6 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50202763(1-(3-(phenylthio)propyl)-4-m-tolylpiperazine | CHE...)
Affinity DataKi:  13.6nMAssay Description:Displacement of [3H]ketanserin from rat cloned 5HT2A receptor expressed in NIH-3T3-GF6 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50202761(N-(4-(3-(4-o-tolylpiperazin-1-yl)propylthio)phenyl...)
Affinity DataKi:  21.1nMAssay Description:Displacement of [3H]ketanserin from rat cloned 5HT2A receptor expressed in NIH-3T3-GF6 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50202764(1-(3-(4-nitrophenylthio)propyl)-4-m-tolylpiperazin...)
Affinity DataKi:  21.1nMAssay Description:Displacement of [3H]ketanserin from rat cloned 5HT2A receptor expressed in NIH-3T3-GF6 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed