Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50019220
TargetAdenosine receptor A2a(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50202991(7-(2-{4-[2-fluoro-4-(2-methoxy-ethoxy)-phenyl]-pip...)
Affinity DataKi:  0.400nMAssay Description:Binding affinity to human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50202994(7-{2-[4-(4-chloro-phenyl)-piperazin-1-yl]-ethyl}-2...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity to human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50203000(7-(2-{4-[4-(2-cyclopropoxy-ethoxy)-phenyl]-piperaz...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity to human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50202989(2-furan-2-yl-7-(2-{4-[4-(3-methoxy-propoxy)-phenyl...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity to human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50202990(SCH-412348 | 7-{2-[4-(2,4-difluoro-phenyl)-piperaz...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity to human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50202996(7-{2-[4-(2-fluoro-phenyl)-piperazin-1-yl]-ethyl}-2...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity to human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50202985(2-furan-2-yl-7-{2-[4-(2,3,4-trifluoro-phenyl)-pipe...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity to human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50202998(2-(4-{4-[2-(5-amino-2-furan-2-yl-pyrazolo[4,3-e][1...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity to human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50203001(1-(4-{4-[2-(5-amino-2-furan-2-yl-pyrazolo[4,3-e][1...)
Affinity DataKi:  0.800nMAssay Description:Binding affinity to human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50202992(7-{2-[4-(4-fluoro-phenyl)-piperazin-1-yl]-ethyl}-2...)
Affinity DataKi:  1nMAssay Description:Binding affinity to human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50202999(2-furan-2-yl-7-{2-[4-(2,4,6-trifluoro-phenyl)-pipe...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity to human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50202986(SCH-420814 | 7-(2-(4-(2,4-difluorophenyl)piperazin...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity to human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50202997(4-{4-[2-(5-amino-2-furan-2-yl-pyrazolo[4,3-e][1,2,...)
Affinity DataKi:  1.30nMAssay Description:Binding affinity to human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50202988(7-{2-[4-(3,4-difluoro-phenyl)-piperazin-1-yl]-ethy...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity to human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50202987(7-{2-[4-(4-ethoxy-phenyl)-piperazin-1-yl]-ethyl}-2...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity to human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50202993(2-furan-2-yl-7-[2-(4-phenyl-piperazin-1-yl)-ethyl]...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity to human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50202983(2-furan-2-yl-7-(2-{4-[4-(2-methoxy-propoxy)-phenyl...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity to human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50202984(4-{4-[2-(5-amino-2-furan-2-yl-pyrazolo[4,3-e][1,2,...)
Affinity DataKi:  2.10nMAssay Description:Binding affinity to human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50202995(2-furan-2-yl-7-{2-[4-(4-methanesulfinylmethoxy-phe...)
Affinity DataKi:  2.20nMAssay Description:Binding affinity to human adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50202986(SCH-420814 | 7-(2-(4-(2,4-difluorophenyl)piperazin...)
Affinity DataKi:  2.5nMAssay Description:Binding affinity to rat adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50202986(SCH-420814 | 7-(2-(4-(2,4-difluorophenyl)piperazin...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to human adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50202986(SCH-420814 | 7-(2-(4-(2,4-difluorophenyl)piperazin...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50202986(SCH-420814 | 7-(2-(4-(2,4-difluorophenyl)piperazin...)
Affinity DataKi: >1.70E+3nMAssay Description:Binding affinity to human adenosine A2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed