Compile Data Set for Download or QSAR
maximum 50k data
Found 33 Enz. Inhib. hit(s) with all data for entry = 2603
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM22496(3-(4-{[(3-phenoxyphenyl)methyl]amino}phenyl)propan...)
Affinity DataEC50:  79nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM22528(3-(4-{[(4-phenoxyphenyl)methyl]amino}phenyl)propan...)
Affinity DataEC50:  195nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM22498(3-(3-{[(3-phenoxyphenyl)methyl]amino}phenyl)propan...)
Affinity DataEC50:  398nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM22499(4-(4-{[(3-phenoxyphenyl)methyl]amino}phenyl)butano...)
Affinity DataEC50:  3.16E+3nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM22500(2-(4-{[(3-phenoxyphenyl)methyl]amino}phenyl)propan...)
Affinity DataEC50:  1.66E+4nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM22501(2-(4-{[(3-phenoxyphenyl)methyl]amino}phenyl)acetic...)
Affinity DataEC50:  3.98E+3nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM22502(3-(4-{[(4-phenylphenyl)methyl]amino}phenyl)propano...)
Affinity DataEC50:  251nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM22503(2-(4-{[(4-phenylphenyl)methyl]amino}phenyl)cyclopr...)
Affinity DataEC50:  40nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM22504(3-(3-{[(4-phenylphenyl)methyl]amino}phenyl)propano...)
Affinity DataEC50:  501nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM22505(4-(4-{[(4-phenylphenyl)methyl]amino}phenyl)butanoi...)
Affinity DataEC50:  1.59E+3nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM22506(2-(4-{[(4-phenylphenyl)methyl]amino}phenyl)propano...)
Affinity DataEC50: >3.16E+4nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM22507(2-(4-{[(4-phenylphenyl)methyl]amino}phenyl)acetic ...)
Affinity DataEC50:  1.23E+4nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM22508(3-(4-{[(3,4-dichlorophenyl)methyl]amino}phenyl)pro...)
Affinity DataEC50:  251nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM22509(3-{4-[(naphthalen-2-ylmethyl)amino]phenyl}propanoi...)
Affinity DataEC50:  794nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM22510(3-(4-{[(3-bromophenyl)methyl]amino}phenyl)propanoi...)
Affinity DataEC50:  794nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM22511(3-(4-{[(5-chlorothiophen-2-yl)methyl]amino}phenyl)...)
Affinity DataEC50:  2.00E+3nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM22512(3-[4-({[4-(trifluoromethyl)phenyl]methyl}amino)phe...)
Affinity DataEC50:  2.00E+3nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM22513(3-(4-{[(2-chlorophenyl)methyl]amino}phenyl)propano...)
Affinity DataEC50:  3.98E+3nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM22514(3-(4-{[(4-methylphenyl)methyl]amino}phenyl)propano...)
Affinity DataEC50:  3.98E+3nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM22515(3-(4-{[(3-fluorophenyl)methyl]amino}phenyl)propano...)
Affinity DataEC50:  5.01E+3nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM22516(3-[4-({[2-chloro-5-(trifluoromethyl)pyridin-3-yl]m...)
Affinity DataEC50:  5.01E+3nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM22517(3-[4-(benzylamino)phenyl]propanoic acid | carboxyl...)
Affinity DataEC50:  7.94E+3nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM22518(3-{4-[(pyridin-3-ylmethyl)amino]phenyl}propanoic a...)
Affinity DataEC50: >3.16E+4nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM22519(3-{4-[({4-[(dimethylamino)methyl]phenyl}methyl)ami...)
Affinity DataEC50: >3.16E+4nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM22520(3-{4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]phenyl}...)
Affinity DataEC50: >3.16E+4nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM22521(4-({[4-(2-carboxyethyl)phenyl]amino}methyl)benzoic...)
Affinity DataEC50: >3.16E+4nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM22522(3-(4-{[(4-hydroxyphenyl)methyl]amino}phenyl)propan...)
Affinity DataEC50: >3.16E+4nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM22523(3-(4-{[(4-cyanophenyl)methyl]amino}phenyl)propanoi...)
Affinity DataEC50: >3.16E+4nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM22524(3-(4-{[(4-methoxyphenyl)methyl]amino}phenyl)propan...)
Affinity DataEC50:  1.26E+3nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM22525(3-(4-{[(3-carbamoylphenyl)methyl]amino}phenyl)prop...)
Affinity DataEC50: >3.16E+4nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM22526(3-{4-[(1H-imidazol-2-ylmethyl)amino]phenyl}propano...)
Affinity DataEC50: >3.16E+4nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM22527(3-(4-{[(3-methanesulfonamidophenyl)methyl]amino}ph...)
Affinity DataEC50: >3.16E+4nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM22497(2-(4-{[(3-phenoxyphenyl)methyl]amino}phenyl)cyclop...)
Affinity DataEC50:  50nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed