Compile Data Set for Download or QSAR
Report error Found 70 Enz. Inhib. hit(s) with all data for entry = 1906
TargetAngiopoietin-1 receptor(Human)
Amgen

LigandChemical structure of BindingDB Monomer ID 14948BDBM14948(4-Methyl-3-(3-(2-(methylamino)pyrimidin-4-yl)pyrid...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

LigandChemical structure of BindingDB Monomer ID 14974BDBM14974(N-{3-[3-(dimethylamino)propyl]-5-(trifluoromethyl)...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 14974BDBM14974(N-{3-[3-(dimethylamino)propyl]-5-(trifluoromethyl)...)
Affinity DataIC50: 2nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 14948BDBM14948(4-Methyl-3-(3-(2-(methylamino)pyrimidin-4-yl)pyrid...)
Affinity DataIC50: 3nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

LigandChemical structure of BindingDB Monomer ID 14984BDBM14984(N-(5-cyclohexyl-2-methoxyphenyl)-4-methyl-3-({3-[2...)
Affinity DataIC50: 4nMpH: 7.5 T: 2°CAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

LigandChemical structure of BindingDB Monomer ID 14971BDBM14971(4-methyl-3-{[3-(pyrimidin-4-yl)pyridin-2-yl]amino}...)
Affinity DataIC50: 4nMpH: 7.5 T: 2°CAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 14971BDBM14971(4-methyl-3-{[3-(pyrimidin-4-yl)pyridin-2-yl]amino}...)
Affinity DataIC50: 4nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

LigandChemical structure of BindingDB Monomer ID 14995BDBM14995(N-(2-{[3-(dimethylamino)propyl](methyl)amino}-5-(t...)
Affinity DataIC50: 4nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

LigandChemical structure of BindingDB Monomer ID 15001BDBM15001(N-(2-((3-(Dimethylamino)propyl)(methyl)amino)-5-is...)
Affinity DataIC50: 6nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

LigandChemical structure of BindingDB Monomer ID 14983BDBM14983(4-methyl-3-({3-[2-(methylamino)pyrimidin-4-yl]pyri...)
Affinity DataIC50: 10nMpH: 7.5 T: 2°CAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

LigandChemical structure of BindingDB Monomer ID 14996BDBM14996(4-methyl-3-({3-[4-(methylamino)-1,3,5-triazin-2-yl...)
Affinity DataIC50: 10nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

LigandChemical structure of BindingDB Monomer ID 15002BDBM15002(N-(5-Cyclopropyl-2-((3-(dimethylamino)propyl)(meth...)
Affinity DataIC50: 13nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

LigandChemical structure of BindingDB Monomer ID 14985BDBM14985(N-(5-Cyclohexyl-2-methoxyphenyl)-4-methyl-3-(3-(4-...)
Affinity DataIC50: 22nMpH: 7.5 T: 2°CAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

LigandChemical structure of BindingDB Monomer ID 15000BDBM15000(N-(2-((3-(Dimethylamino)propyl)(methyl)amino)-5-(t...)
Affinity DataIC50: 30nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

LigandChemical structure of BindingDB Monomer ID 14991BDBM14991(4-chloro-3-({3-[2-(methylamino)pyrimidin-4-yl]pyri...)
Affinity DataIC50: 30nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 15019BDBM15019(N-(4-phenoxyphenyl)-2-[(pyridin-4-ylmethyl)amino]p...)
Affinity DataIC50: 38nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandChemical structure of BindingDB Monomer ID 15020BDBM15020(N-(4-phenoxyphenyl)-3-[(3-{4-[(3,4,5-trimethoxyphe...)
Affinity DataIC50: 38nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

LigandChemical structure of BindingDB Monomer ID 14992BDBM14992(4-Methyl-3-(3-(2-(methylamino)pyrimidin-4-yl)pyrid...)
Affinity DataIC50: 39nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

LigandChemical structure of BindingDB Monomer ID 14994BDBM14994(2-Fluoro-5-(3-(2-(methylamino)pyrimidin-4-yl)pyrid...)
Affinity DataIC50: 40nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

LigandChemical structure of BindingDB Monomer ID 14975BDBM14975(N-[2-methoxy-5-(trifluoromethyl)phenyl]-4-methyl-3...)
Affinity DataIC50: 43nMpH: 7.5 T: 2°CAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 14995BDBM14995(N-(2-{[3-(dimethylamino)propyl](methyl)amino}-5-(t...)
Affinity DataIC50: 46nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

LigandChemical structure of BindingDB Monomer ID 14999BDBM14999(2-Fluoro-5-(3-(4-(methylamino)-1,3,5-triazin-2-yl)...)
Affinity DataIC50: 53nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 14975BDBM14975(N-[2-methoxy-5-(trifluoromethyl)phenyl]-4-methyl-3...)
Affinity DataIC50: 58nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

LigandChemical structure of BindingDB Monomer ID 14998BDBM14998(N-(2-((3-(Dimethylamino)propyl)(methyl)amino)-5-(t...)
Affinity DataIC50: 59nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 14977BDBM14977(4-Methyl-3-(3-(pyrimidin-4-yl)pyridin-2-yloxy)-N-(...)
Affinity DataIC50: 59nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

LigandChemical structure of BindingDB Monomer ID 14986BDBM14986(N-(5-Cyclohexyl-2-methoxyphenyl)-4-methyl-3-(3-(2-...)
Affinity DataIC50: 62nMpH: 7.5 T: 2°CAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

LigandChemical structure of BindingDB Monomer ID 14990BDBM14990(4-fluoro-3-({3-[2-(methylamino)pyrimidin-4-yl]pyri...)
Affinity DataIC50: 62nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 15018BDBM15018(4-[2-(phenylamino)pyridin-3-yl]-N-(3,4,5-trimethox...)
Affinity DataIC50: 68nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 14984BDBM14984(N-(5-cyclohexyl-2-methoxyphenyl)-4-methyl-3-({3-[2...)
Affinity DataIC50: 70nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

LigandChemical structure of BindingDB Monomer ID 15020BDBM15020(N-(4-phenoxyphenyl)-3-[(3-{4-[(3,4,5-trimethoxyphe...)
Affinity DataIC50: 85nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 14996BDBM14996(4-methyl-3-({3-[4-(methylamino)-1,3,5-triazin-2-yl...)
Affinity DataIC50: 97nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

LigandChemical structure of BindingDB Monomer ID 14989BDBM14989(3-({3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl}...)
Affinity DataIC50: 99nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 14979BDBM14979(N-[2-methoxy-5-(trifluoromethyl)phenyl]-4-methyl-3...)
Affinity DataIC50: 100nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

LigandChemical structure of BindingDB Monomer ID 14979BDBM14979(N-[2-methoxy-5-(trifluoromethyl)phenyl]-4-methyl-3...)
Affinity DataIC50: 103nMpH: 7.5 T: 2°CAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

LigandChemical structure of BindingDB Monomer ID 14997BDBM14997(4-methyl-3-({3-[4-(methylamino)-1,3,5-triazin-2-yl...)
Affinity DataIC50: 108nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

LigandChemical structure of BindingDB Monomer ID 14977BDBM14977(4-Methyl-3-(3-(pyrimidin-4-yl)pyridin-2-yloxy)-N-(...)
Affinity DataIC50: 153nMpH: 7.5 T: 2°CAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 14973BDBM14973(4-methyl-3-{[3-(pyrimidin-4-yl)pyridin-2-yl]amino}...)
Affinity DataIC50: 177nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

LigandChemical structure of BindingDB Monomer ID 14976BDBM14976(4-methyl-N-[2-(piperidin-1-yl)-5-(trifluoromethyl)...)
Affinity DataIC50: 181nMpH: 7.5 T: 2°CAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 14983BDBM14983(4-methyl-3-({3-[2-(methylamino)pyrimidin-4-yl]pyri...)
Affinity DataIC50: 310nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

LigandChemical structure of BindingDB Monomer ID 14980BDBM14980(4-Methyl-N-(2-(piperidin-1-yl)-5-(trifluoromethyl)...)
Affinity DataIC50: 366nMpH: 7.5 T: 2°CAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

LigandChemical structure of BindingDB Monomer ID 14993BDBM14993(2-methyl-3-({3-[2-(methylamino)pyrimidin-4-yl]pyri...)
Affinity DataIC50: 388nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

LigandChemical structure of BindingDB Monomer ID 14982BDBM14982(4-methyl-N-[2-(morpholin-4-yl)-5-(trifluoromethyl)...)
Affinity DataIC50: 399nMpH: 7.5 T: 2°CAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 14972BDBM14972(4-Methyl-N-phenyl-3-(3-(pyrimidin-4-yl)pyridin-2-y...)
Affinity DataIC50: 435nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 14992BDBM14992(4-Methyl-3-(3-(2-(methylamino)pyrimidin-4-yl)pyrid...)
Affinity DataIC50: 461nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

LigandChemical structure of BindingDB Monomer ID 14973BDBM14973(4-methyl-3-{[3-(pyrimidin-4-yl)pyridin-2-yl]amino}...)
Affinity DataIC50: 504nMpH: 7.5 T: 2°CAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 14991BDBM14991(4-chloro-3-({3-[2-(methylamino)pyrimidin-4-yl]pyri...)
Affinity DataIC50: 675nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 14978BDBM14978(4-Methyl-3-(3-(pyrimidin-4-yl)pyridin-2-yloxy)-N-(...)
Affinity DataIC50: 705nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

LigandChemical structure of BindingDB Monomer ID 14972BDBM14972(4-Methyl-N-phenyl-3-(3-(pyrimidin-4-yl)pyridin-2-y...)
Affinity DataIC50: 1.22E+3nMpH: 7.5 T: 2°CAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 14980BDBM14980(4-Methyl-N-(2-(piperidin-1-yl)-5-(trifluoromethyl)...)
Affinity DataIC50: 1.30E+3nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 14990BDBM14990(4-fluoro-3-({3-[2-(methylamino)pyrimidin-4-yl]pyri...)
Affinity DataIC50: 2.00E+3nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2007
Entry Details Article
PubMed
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