Compile Data Set for Download or QSAR
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Found 30 Enz. Inhib. hit(s) with all data for entry = 50019299
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50203481(2-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohe...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [125]HEAT from human adrenergic alpha1d receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM82517(2-{4-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-butyl}-...)
Affinity DataKi:  0.260nMAssay Description:Displacement of [125]HEAT from human adrenergic alpha1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM82517(2-{4-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-butyl}-...)
Affinity DataKi:  0.300nMAssay Description:Displacement of [125]HEAT from human adrenergic alpha1d receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50203485(5,6-dichloro-2-(4-(4-(2-isopropoxyphenyl)piperazin...)
Affinity DataKi:  0.300nMAssay Description:Displacement of [125]HEAT from human adrenergic alpha1d receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50203486(2-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohe...)
Affinity DataKi:  0.400nMAssay Description:Displacement of [125]HEAT from human adrenergic alpha1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50203480(8-fluoro-2-(4-(4-(2-isopropoxyphenyl)piperazin-1-y...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [125]HEAT from human adrenergic alpha1d receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50203480(8-fluoro-2-(4-(4-(2-isopropoxyphenyl)piperazin-1-y...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [125]HEAT from human adrenergic alpha1d receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50203486(2-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohe...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [125]HEAT from human adrenergic alpha1d receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50203484(6-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohe...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [125]HEAT from human adrenergic alpha1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM82517(2-{4-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-butyl}-...)
Affinity DataKi:  0.960nMAssay Description:Displacement of [125]HEAT from human adrenergic alpha1b receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50203482(4-fluoro-2-(4-(4-(2-isopropoxyphenyl)piperazin-1-y...)
Affinity DataKi:  1nMAssay Description:Displacement of [125]HEAT from human adrenergic alpha1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50203482(4-fluoro-2-(4-(4-(2-isopropoxyphenyl)piperazin-1-y...)
Affinity DataKi:  1nMAssay Description:Displacement of [125]HEAT from human adrenergic alpha1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50203484(6-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohe...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [125]HEAT from human adrenergic alpha1d receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50203481(2-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohe...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [125]HEAT from human adrenergic alpha1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50203485(5,6-dichloro-2-(4-(4-(2-isopropoxyphenyl)piperazin...)
Affinity DataKi:  2.70nMAssay Description:Displacement of [125]HEAT from human adrenergic alpha1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50203480(8-fluoro-2-(4-(4-(2-isopropoxyphenyl)piperazin-1-y...)
Affinity DataKi:  3.90nMAssay Description:Displacement of [125]HEAT from human adrenergic alpha1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50203480(8-fluoro-2-(4-(4-(2-isopropoxyphenyl)piperazin-1-y...)
Affinity DataKi:  3.90nMAssay Description:Displacement of [125]HEAT from human adrenergic alpha1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50203482(4-fluoro-2-(4-(4-(2-isopropoxyphenyl)piperazin-1-y...)
Affinity DataKi:  14.9nMAssay Description:Displacement of [125]HEAT from human adrenergic alpha1d receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50203482(4-fluoro-2-(4-(4-(2-isopropoxyphenyl)piperazin-1-y...)
Affinity DataKi:  14.9nMAssay Description:Displacement of [125]HEAT from human adrenergic alpha1d receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50203481(2-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohe...)
Affinity DataKi:  15nMAssay Description:Displacement of [125]HEAT from human adrenergic alpha1b receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50203486(2-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohe...)
Affinity DataKi:  22.4nMAssay Description:Displacement of [125]HEAT from human adrenergic alpha1b receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50203483(4,5,6,7-tetrafluoro-2-(4-(4-(2-isopropoxyphenyl)pi...)
Affinity DataKi:  30.2nMAssay Description:Displacement of [125]HEAT from human adrenergic alpha1d receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50203483(4,5,6,7-tetrafluoro-2-(4-(4-(2-isopropoxyphenyl)pi...)
Affinity DataKi:  37.8nMAssay Description:Displacement of [125]HEAT from human adrenergic alpha1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50203484(6-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohe...)
Affinity DataKi:  44.6nMAssay Description:Displacement of [125]HEAT from human adrenergic alpha1b receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50203480(8-fluoro-2-(4-(4-(2-isopropoxyphenyl)piperazin-1-y...)
Affinity DataKi:  46.5nMAssay Description:Displacement of [125]HEAT from human adrenergic alpha1b receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50203480(8-fluoro-2-(4-(4-(2-isopropoxyphenyl)piperazin-1-y...)
Affinity DataKi:  46.5nMAssay Description:Displacement of [125]HEAT from human adrenergic alpha1b receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50203482(4-fluoro-2-(4-(4-(2-isopropoxyphenyl)piperazin-1-y...)
Affinity DataKi:  127nMAssay Description:Displacement of [125]HEAT from human adrenergic alpha1b receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50203482(4-fluoro-2-(4-(4-(2-isopropoxyphenyl)piperazin-1-y...)
Affinity DataKi:  127nMAssay Description:Displacement of [125]HEAT from human adrenergic alpha1b receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50203485(5,6-dichloro-2-(4-(4-(2-isopropoxyphenyl)piperazin...)
Affinity DataKi:  1.08E+3nMAssay Description:Displacement of [125]HEAT from human adrenergic alpha1b receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50203483(4,5,6,7-tetrafluoro-2-(4-(4-(2-isopropoxyphenyl)pi...)
Affinity DataKi:  4.11E+3nMAssay Description:Displacement of [125]HEAT from human adrenergic alpha1b receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed