Compile Data Set for Download or QSAR
maximum 50k data
Found 10 Enz. Inhib. hit(s) with all data for entry = 50041524
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50204825(AcDRGDS | CHEMBL241297)
Affinity DataIC50:  20nMAssay Description:Inhibition of integrin alpha-v-beta-3 receptor-mediated human SK-MEL-24 cell adhesion to fibronectin by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50204820((S)-N-benzyl-3-{[(R)-1-(4-guanidino-butyryl)-pyrro...)
Affinity DataIC50:  26nMAssay Description:Inhibition of integrin alpha-v-beta-3 receptor-mediated human SK-MEL-24 cell adhesion to fibronectin by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50204824((S)-4-benzylcarbamoyl-4-{[(R)-1-(3-guanidino-propi...)
Affinity DataIC50:  35nMAssay Description:Inhibition of integrin alpha-v-beta-3 receptor-mediated human SK-MEL-24 cell adhesion to fibronectin by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50204822((S)-N-benzyl-3-({(R)-1-[(S)-5-guanidino-2-(toluene...)
Affinity DataIC50:  150nMAssay Description:Inhibition of integrin alpha-v-beta-3 receptor-mediated human SK-MEL-24 cell adhesion to fibronectin by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50204827(3-{[(R)-1-(4-guanidino-butyryl)-pyrrolidine-2-carb...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of integrin alpha-v-beta-3 receptor-mediated human SK-MEL-24 cell adhesion to fibronectin by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50204828((S)-4-benzylcarbamoyl-4-{[(R)-1-(4-guanidino-butyr...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of integrin alpha-v-beta-3 receptor-mediated human SK-MEL-24 cell adhesion to fibronectin by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50204826((S)-3-{[(R)-1-(4-guanidino-butyryl)-pyrrolidine-2-...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of integrin alpha-v-beta-3 receptor-mediated human SK-MEL-24 cell adhesion to fibronectin by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50204821((S)-N-benzyl-3-{[(R)-1-(3-guanidino-propionyl)-pyr...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of integrin alpha-v-beta-3 receptor-mediated human SK-MEL-24 cell adhesion to fibronectin by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50204823((S)-N-benzyl-3-({(S)-1-[(S)-5-guanidino-2-(toluene...)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of integrin alpha-v-beta-3 receptor-mediated human SK-MEL-24 cell adhesion to fibronectin by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50204819((S)-N-benzyl-3-{[(R)-1-(5-guanidino-pentanoyl)-pyr...)
Affinity DataIC50:  2.30E+5nMAssay Description:Inhibition of integrin alpha-v-beta-3 receptor-mediated human SK-MEL-24 cell adhesion to fibronectin by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed